CAS 1423715-09-6

Benzoic acid, 3-​(4-​morpholinylsulfonyl)​-​, (2E)​-​2-​[1-​(5-​chloro-​2-​hydroxyphenyl)​ethylidene]​hydrazide

CAS: 1423715-09-6

Formula: C₁₉H₂₀ClN₃O₅S

Purezza: %

Colore e forma: Solid

Peso molecolare: 437.8972

Ref: IN-DA009CK9

SP2509

CAS: 1423715-09-6

SP2509

Purezza: ≥98%

Peso molecolare: 437.9g/mol

Ref: 54-BUP10444

SP2509

CAS: 1423715-09-6

SP2509 is a specific histone demethylase LSD1 inhibitor(IC50 =13 nM).

Formula: C₁₉H₂₀ClN₃O₅S

Purezza: 98.82% - 99.53%

Colore e forma: Solid

Peso molecolare: 437.9

Ref: TM-T2304

SP 2509

CAS: 1423715-09-6

Lysine-specific demethylase 1 ( LSD1) antagonist

Formula: C₁₉H₂₀ClN₃O₅S

Purezza: (Hplc) Min. 98.0%

Colore e forma: Powder

Peso molecolare: 437.9 g/mol

Ref: 3D-BS168098

SP 2509

Prodotto controllato

CAS: 1423715-09-6

Applications SP 2509 reduces the effect of the LSD1 binding to CoREST, resulting in increased methylation of H3K4 and driving increased expression of p21, p27 and CCAAT/enhancer binding protein α in acute myeloid leukemia cells. Anti-leukemia agent.
References Sorna, V. et al.: J. Med. Chem., 56, 9496 (2013); Fiskus, W. et al.: Leukemia, 11, 2155 (2014);

Formula: C₁₉H₂₀ClN₃O₅S

Colore e forma: Neat

Peso molecolare: 437.9

Ref: TR-S679000