CAS 152542-00-2

Risperidone Related Compound G (3-{2-[4-(4-Fluoro-2-hydroxybenzoyl)piperidin-1-yl]ethyl}-2-methyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-one hydrochloride)

CAS: 152542-00-2

Compounds containing a pyrimidine ring, whether or not hydrogenated, or piperazine ring in the structure, nesoi

Formula: C₂₃H₂₈FN₃O₃

Colore e forma: Off-White Powder

Peso molecolare: 413.21147

Ref: 45-1604756

Risperidone USP Related Compound G (Free Form)

CAS: 152542-00-2

Formula: C₂₃H₂₈FN₃O₃

Colore e forma: White To Off-White Solid

Peso molecolare: 413.49

Ref: 4Z-R-0626

3-[2-[4-(4-Fluoro-2-hydroxybenzoyl)piperidin-1-yl]ethyl]-2-methyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-one

Prodotto controllato

CAS: 152542-00-2

Colore e forma: Neat

Ref: 86-MM0491.09

3-[2-[4-(4-Fluoro-2-hydroxybenzoyl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one Hydrochloride

Prodotto controllato

CAS: 152542-00-2

Applications Risperidone (R525000) metabolite.
References Meuldermans, W. et al.; Drug Metab. Dispos. 22, 129 (1994); Mannens, G. et al.; Drug Metab. Dispos. 21, 1134 (1993)

Formula: C₂₃H₂₈FN₃O₃·HCl

Colore e forma: Neat

Peso molecolare: 449.946

Ref: TR-F591875

Risperidone USP Related Compound G

CAS: 152542-00-2

Formula: C₂₃H₂₈FN₃O₃

Peso molecolare: 413.49

Ref: ST-EA-CP-R15019

3-[2-[4-(4-Fluoro-2-hydroxybenzoyl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one

Prodotto controllato

CAS: 152542-00-2

Applications 3-[2-[4-(4-Fluoro-2-hydroxybenzoyl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one is an intermediate used in the synthesis of Bicyclo Risperidone (B382800), which is an impurity of Risperidone (R525000); a combined serotonin (5-HT2) and dopamine (D2) receptor antagonist.
References Jannssen, P.A.J., et al.: J. Pharmacol. Exp. Ther., 244, 685 (1988); Gelders, Y.G., et al.: Pharmacopsychiatry, 23, 206 (1990); Green, B.: Curr. Med. Res. Opin., 16, 57 (2000)

Formula: C₂₃H₂₈FN₃O₃

Colore e forma: Neat

Peso molecolare: 413.49

Ref: TR-F591878

3-[2-[4-(4-Fluoro-2-hydroxybenzoyl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one

CAS: 152542-00-2

Paliperidone is a psychotropic drug that belongs to the class of antipsychotics. It is used in the treatment of schizophrenia and other psychotic disorders. Paliperidone is metabolized extensively by cytochrome P450 enzymes, primarily CYP2D6, into active metabolites with different pharmacokinetics. The drug binds to serotonin receptors and has been shown to have anti-inflammatory effects. Paliperidone also has an affinity for histamine receptors and H1 receptors, which may contribute to its antipsychotic activity and sedative effects respectively. Paliperidone can be administered as a salt or ester prodrug form, but the most common form commercially available is paliperidone palmitate (PP).

Formula: C₂₃H₂₈FN₃O₃

Purezza: Min. 95%

Peso molecolare: 413.49 g/mol

Ref: 3D-FF103471