CAS 1616340-94-3

Methyl Bictegravir

CAS: 1616340-94-3

Formula: C₂₂H₂₀F₃N₃O₅

Peso molecolare: 463.41

Ref: 4Z-B-167010

(2R,5S,13aR)-2,3,4,5,7,9,13,13a-Octahydro-8-methoxy-7,9-dioxo-N-[(2,4,6-trifluorophenyl)methyl]-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide-d2, 15N

Prodotto controllato

CAS: 1616340-94-3

Applications (2R,5S,13aR)-2,3,4,5,7,9,13,13a-Octahydro-8-methoxy-7,9-dioxo-N-[(2,4,6-trifluorophenyl)methyl]-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide-d2, 15N is an intermediate in the synthesis of Bictegravir-15N, d2 (B382096), which is the labeled version of Bictegravir, which is a novel, potent inhibitor of HIV-1 integrase with an IC50 of 7.5 nM.
References Tsiang M. et al.: Antimicrob Agents Chemother. 2016 Nov 21;60(12):7086-7097;

Formula: C₂₂D₂H₁₈F₃₁₅NN₂O₅

Colore e forma: Neat

Peso molecolare: 466.412

Ref: TR-M262872

Methyl Bictegravir

CAS: 1616340-94-3

Formula: C₂₂H₂₀F₃N₃O₅

Peso molecolare: 463.41

Ref: ST-EA-CP-B147010