CAS 1838622-25-5

EST73502

CAS: 1838622-25-5

EST73502 is a compound that functions as a dual agonist for the μ-opioid receptor (MOR) and an antagonist for the σ1 receptor (σ1R). It is selective, orally active, and possesses the ability to penetrate the blood-brain barrier (BBB). The compound exhibits a Ki value of 64 nM for the MOR and 118 nM for the σ1R. Additionally, EST73502 demonstrates antinociceptive activity [1].

Formula: C₁₉H₂₆F₂N₂O₂

Purezza: 98%

Colore e forma: Solid

Peso molecolare: 352.426

Ref: TM-T61240