CAS 200940-22-3

2,3-Diidro-5-metil-N-[6-[(2-metil-3-piridinil)ossi]-3-piridinil]-6-(trifluorometil)-1H-indolo-1-carbossamide

Descrizione:

2,3-Diidro-5-metil-N-[6-[(2-metil-3-piridinil)ossi]-3-piridinil]-6-(trifluorometil)-1H-indolo-1-carbossamide, con numero CAS 200940-22-3, è un composto organico sintetico caratterizzato dalla sua complessa struttura molecolare, che include un nucleo di indolo, più anelli aromatici e vari gruppi funzionali come trifluorometile e carbossamide. Questo composto presenta proprietà tipiche dei derivati dell'indolo, inclusa una potenziale attività biologica, rendendolo di interesse nella ricerca farmaceutica. La presenza di anelli di piridina suggerisce possibili interazioni con bersagli biologici, influenzando potenzialmente la sua farmacocinetica e farmacodinamica. Inoltre, si sa che il gruppo trifluorometile migliora la lipofilia e la stabilità metabolica, il che può essere vantaggioso nel design dei farmaci. La solubilità, stabilità e reattività del composto dipenderebbero dai suoi specifici gruppi funzionali e dalla conformazione molecolare complessiva. Come molte molecole organiche complesse, la sua sintesi e caratterizzazione richiederebbero tecniche avanzate come la spettroscopia NMR, la spettrometria di massa e la cristallografia per confermare la sua struttura e purezza.

Formula: C₂₂H₁₉F₃N₄O₂

InChI: InChI=1S/C22H19F3N4O2/c1-13-10-15-7-9-29(18(15)11-17(13)22(23,24)25)21(30)28-16-5-6-20(27-12-16)31-19-4-3-8-26-14(19)2/h3-6,8,10-12H,7,9H2,1-2H3,(H,28,30)

InChI key: InChIKey=ZETBBVYSBABLHL-UHFFFAOYSA-N

SMILES: C(NC=1C=CC(OC2=C(C)N=CC=C2)=NC1)(=O)N3C=4C(=CC(C)=C(C(F)(F)F)C4)CC3

Sinonimi:

• 1H-Indole-1-carboxamide, 2,3-dihydro-5-methyl-N-[6-[(2-methyl-3-pyridinyl)oxy]-3-pyridinyl]-6-(trifluoromethyl)-
• 2,3-Dihydro-5-methyl-N-[6-[(2-methyl-3-pyridinyl)oxy]-3-pyridinyl]-6-(trifluoromethyl)-1H-indole-1-carboxamide
• Sb-243213

SB 243213

CAS: 200940-22-3

SB 243213

Purezza: ≥98%

Peso molecolare: 428.41g/mol

Ref: 54-BUP07457

SB 243213

CAS: 200940-22-3

SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.

Formula: C₂₂H₁₉F₃N₄O₂

Purezza: 98.78% - 99.86%

Colore e forma: Solid

Peso molecolare: 428.41

Ref: TM-T37816

SB 243213

CAS: 200940-22-3

SB 243213 is a compound that has been extensively studied for its effects on melanogenesis and pigmentation. It acts as an antagonist for the IL-1 receptor, specifically IL-1RA, and the 5-HT2C receptor in humans. This compound has potential applications in the diagnosis and treatment of conditions related to pigmentation disorders such as vitiligo and melasma. Additionally, SB 243213 has shown promising results in cancer research, particularly as an inhibitory factor for melanoma cells. It can also be used in the development of microcapsules for targeted drug delivery in diseases like diabetes. Although not a fluoroquinolone or steroidal compound itself, SB 243213 belongs to the class of research chemicals that have gained attention in various scientific fields.

Formula: C₂₂H₁₉F₃N₄O₂

Purezza: Min. 95%

Peso molecolare: 428.4 g/mol

Ref: 3D-AIA94022

SB 243213

CAS: 200940-22-3

SB 243213 is a cell-permeable, potent, and selective inhibitor of the Kv1.3 potassium channel that is used as a research tool in pharmacology and cell biology. SB 243213 is a peptide that binds to the receptor site on the Kv1.3 channel and blocks ion flow, thereby inhibiting this type of potassium channel. The binding affinity of SB 243213 to the Kv1.3 receptor site is greater than 10,000 times higher than its binding affinity for other ion channels such as the nicotinic acetylcholine receptors. This agent has been shown to be an activator of protein interactions in cells and has also been used as an antibody labeling reagent.

Formula: C₂₂H₁₉F₃N₄O₂

Purezza: Min. 95%

Peso molecolare: 428.4 g/mol

Ref: 3D-BS181806