CAS 202646-80-8

FR194921

CAS: 202646-80-8

FR194921 is a selective, high-affinity antagonist of the adenosine A1 receptor. It has been shown to selectively bind to the adenosine A1 receptor and block its binding site. FR194921 is orally active and has shown potential in the treatment of Parkinson's disease, Alzheimer's disease, and schizophrenia. The molecular structure of FR194921 is similar to that of caffeine with a fluorine atom replacing one hydrogen atom on the methyl group. This chemical property may account for some of its pharmacological properties.
FR194921 binds to the adenosine A1 receptor at a different site than caffeine, which may explain why FR194921 does not have any stimulant effects.

Formula: C₂₃H₂₃N₅O

Purezza: Min. 95%

Peso molecolare: 385.5 g/mol

Ref: 3D-CIA64680

FR-194921

CAS: 202646-80-8

FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.

Formula: C₂₃H₂₃N₅O

Colore e forma: Solid

Peso molecolare: 385.46

Ref: TM-T27379