CAS 2305815-72-7

R8-T198wt

CAS: 2305815-72-7

Cell-permeable peptide blocking Pim-1 kinase, halts DU145 cell growth, causes G1 arrest and apoptosis, inert to RPWE-1 cells at 10-20 μM.

Formula: C₁₁₁H₂₁₁N₅₉O₂₆S

Purezza: 98%

Colore e forma: Solid

Peso molecolare: 2820.33

Ref: TM-TP2128

R8-T198wt

CAS: 2305815-72-7

R8-T198wt is a potent and selective inhibitor of the Pim-1 kinase. Inhibiting Pim-1 kinase has been shown to have anti-tumor activity in vitro and in vivo. It is also a potential treatment for diseases such as cancer, where the Pim-1 kinase is overexpressed. This drug is designed to inhibit the Pim-1 kinase by binding to a specific site on its ATP binding site. R8-T198wt is an ATP analog that binds to the ATP binding site of pim-1 kinase, thereby inhibiting its activity.

Formula: C₁₁₁H₂₁₁N₅₉O₂₆S

Purezza: Min. 95%

Peso molecolare: 2,820.3 g/mol

Ref: 3D-FSD81572