CAS 59-33-6

Maleato di pirilamina

Descrizione:

Maleato di pirilamina è un composto antistaminico utilizzato principalmente per alleviare reazioni allergiche e sintomi come la febbre da fieno e l'orticaria. È classificato come un antistaminico di prima generazione, il che significa che può attraversare la barriera ematoencefalica, portando spesso a effetti sedativi. La struttura chimica di Maleato di pirilamina consiste in un anello di piridina e un gruppo amminico, contribuendo alla sua attività farmacologica bloccando i recettori H1 dell'istamina. La forma di sale maleato ne migliora la solubilità e la stabilità. Maleato di pirilamina è tipicamente somministrato per via orale ed è disponibile in varie formulazioni, tra cui compresse e sciroppi. Gli effetti collaterali comuni possono includere sonnolenza, secchezza delle fauci e vertigini, che sono caratteristici di molti antistaminici di prima generazione. È importante utilizzare questo farmaco sotto supervisione medica, specialmente in individui con condizioni preesistenti o in coloro che assumono altri farmaci, a causa di potenziali interazioni e controindicazioni. In generale, Maleato di pirilamina rappresenta un'opzione efficace per gestire i sintomi allergici, sebbene si consiglia cautela riguardo alle sue proprietà sedative.

Formula: C₂₁H₂₇N₃O₅

InChI: InChI=1/C17H23N3O.C4H4O4/c1-19(2)12-13-20(17-6-4-5-11-18-17)14-15-7-9-16(21-3)10-8-15;5-3(6)1-2-4(7)8/h4-11H,12-14H2,1-3H3;1-2H,(H,5,6)(H,7,8)/p-2/b;2-1-

InChI key: InChIKey=JXYWFNAQESKDNC-BTJKTKAUSA-N

SMILES: C(=C\C(O)=O)\C(O)=O.N(CC1=CC=C(OC)C=C1)(CCN(C)C)C2=CC=CC=N2

Sinonimi:

• 1,2-Ethanediamine, N-[(4-methoxyphenyl)methyl]-N',N'-dimethyl-N-2-pyridinyl-, (2Z)-2-butenedioate (1:1)
• 1,2-Ethanediamine, N-[(4-methoxyphenyl)methyl]-N',N'-dimethyl-N-2-pyridinyl-, (Z)-2-butenedioate (1:1)
• 1,2-Ethanediamine, N1-[(4-methoxyphenyl)methyl]-N2,N2-dimethyl-N1-2-pyridinyl-, (2Z)-2-butenedioate (1:1)
• 1,2-Ethanediamine, N¹-[(4-methoxyphenyl)methyl]-N²,N²-dimethyl-N¹-2-pyridinyl-, (2Z)-2-butenedioate (1:1)
• 2-[(2-Dimethylaminoethyl)(p-methoxybenzyl)amino]-pyridine maleate
• 2-[[2-(Dimethylamino)ethyl](p-methoxybenzyl)amino]pyridine Bimaleate
• AH
• Anisopyradamine
• Antamine
• Anthisan maleate
• Antihist
• Antisan
• Diaminide maleate
• Enrumay
• Histalet Forte
• Histalon
• Histan
• Histapyran
• Histatex
• Histavet P
• Maleate De Mepyramine
• Maleato De Mepiramina
• Maleinsaeure-(2-(N-(2-Dimethylamino-Aethyl)-N-(P-Methoxy-Benzyl)-Amino)-Pyridin) - Salz
• Mepyramine hydrogen maleinate
• Mepyramine maleate
• Mepyraminmaleat
• Minihist
• N-(4-methoxybenzyl)-N',N'-dimethyl-N-(pyridin-2-yl)ethane-1,2-diamine
• N-(4-methoxybenzyl)-N',N'-dimethyl-N-pyridin-2-ylethane-1,2-diamine (2E)-but-2-enedioate
• N-(4-methoxybenzyl)-N',N'-dimethyl-N-pyridin-2-ylethane-1,2-diamine (2Z)-but-2-enedioate
• N-p-Methoxybenzyl-N',N'-dimethyl-N-α-pyridylethylenediamine maleate
• Neo-Antergan maleate
• Neoantergan maleate
• Nsc 3604
• Paramal
• Paraminyl
• Paraminyl maleate
• Parmal
• Prefrin A
• Pymafed
• Pyra Maleate
• Pyramal
• Pyranilamine maleate
• Pyraninyl
• Pyranisamine maleate
• Pyridine, 2-[[2-(dimethylamino)ethyl](p-methoxybenzyl)amino]-, maleate (1:1)
• Pyrilamine Maleate
• Renstamin
• Stamine
• Stangen
• Stangen maleate
• Statomin maleate
• Thylogen
• Thylogen maleate
• N-[4-METHOXY-PHENYL]METHYL-N',N'-DIMETHYL-N[2-PYRIDINYL]-1,2-ETHANEDIAMINE MALEATE SALT
• diaminidemaleate
• MEPYRAMINE MALEATE SALT
• 2-((2-(dimethylamino)ethyl)(p-methoxybenzyl)amino)-pyridinmaleate(1:1)
• (z)-2-butenedioat
• n-((4-methoxyphenyl)methyl)-n,n’-dimethyl-n-2-pyridinyl-2-ethanediamine
• PYRILAMINE MALEATE SALT
• anthisanmaleate
• 2-ethanediamine,n-[(4-methoxyphenyl)methyl]-n’,n’-dimethyl-n-2-pyridinyl-(
• 2-((2-(dimethylamino)ethyl)(p-methoxybenzyl)amino)pyridinebimaleate
• N-(P-METHOXYBENZYL)-N',N'-DIMETHYL-N-2-PYRIDYLETHYLENEDIAMINE MALEATE

Pyrilamine Maleate

CAS: 59-33-6, 91-84-9

Formula: C₁₇H₂₃N₃O·C₄H₄O₄

Purezza: >98.0%(T)(HPLC)

Colore e forma: White to Almost white powder to crystal

Peso molecolare: 401.46

Ref: 3B-P2369

Pyrilamine maleate

CAS: 59-33-6

Selective inverse agonist for the H-1 histamine receptor

Formula: C₁₇H₂₃N₃O·C₄H₄O₄

Peso molecolare: 401.46

Ref: 02-J63247

Mepyramine Maleate

CAS: 59-33-6

Colore e forma: Neat

Ref: 61-FOR0559.00

MEPYRAMINE MALEATE CRS

CAS: 59-33-6

MEPYRAMINE MALEATE CRS

Ref: 41-M0500000

Pyrilamine Maleate

CAS: 59-33-6

Compounds containing an unfused pyridine ring in the structure, nesoi

Formula: C₁₇H₂₃N₃O·C₄H₄O₄

Colore e forma: Powder

Peso molecolare: 401.19507

Ref: 45-1588004

1,2-Ethanediamine,N-[(4-methoxyphenyl)methyl]-N',N'-dimethyl-N-2-pyridinyl-,(2Z)-2-butenedioate (1:1)

CAS: 59-33-6

Formula: C₂₁H₂₇N₃O₅

Purezza: 98%

Colore e forma: Solid

Peso molecolare: 401.4562

Ref: IN-DA00IAHB

Mepyramine maleate

CAS: 59-33-6

Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.

Formula: C₂₁H₂₇N₃O₅

Purezza: 99.51% - 99.7%

Colore e forma: White Crystalline Powder

Peso molecolare: 401.47

Ref: TM-T1232

Mepyramine Maleate

CAS: 59-33-6

Formula: C₁₇H₂₃N₃O·C₄H₄O₄

Colore e forma: White To Off-White Solid

Peso molecolare: 285.39 116.07

Ref: 4Z-M-179001

Mepyramine maleate

CAS: 59-33-6

Mepyramine maleate

Purezza: ≥98%

Peso molecolare: 401.47g/mol

Ref: 54-BUP18353

Pyrilamine maleate salt

CAS: 59-33-6

Formula: C₁₇H₂₃N₃O·C₄H₄O₄

Purezza: ≥ 98.0%

Colore e forma: White to off-white crystalline powder

Peso molecolare: 401.46

Ref: 7W-GP6304

N1-(4-Methoxybenzyl)-N2,N2-Dimethyl-N1-(Pyridin-2-Yl)Ethane-1,2-Diamine Maleate

CAS: 59-33-6

N1-(4-Methoxybenzyl)-N2,N2-Dimethyl-N1-(Pyridin-2-Yl)Ethane-1,2-Diamine Maleate

Purezza: 98%

Peso molecolare: 401.46g/mol

Ref: 54-OR1030388

Mepyramine maleate

Prodotto controllato

CAS: 59-33-6

Formula: C₁₇H₂₃N₃O·C₄H₄O₄

Colore e forma: Neat

Peso molecolare: 401.46

Ref: 04-C14896000

Mepyramine Maleate

Prodotto controllato

CAS: 59-33-6

Formula: C₁₇H₂₃N₃O·C₄H₄O₄

Colore e forma: Neat

Peso molecolare: 401.46

Ref: 86-MM0559.00

Pyrilamine Maleate Salt

Prodotto controllato

CAS: 59-33-6

Applications Antihistaminic.
References Watanabe, T., et al.: Brain Res., 295, 13 (1984), Nakazato, E., et al.: Life Sci., 67, 1139 (2000), Masuoka, T., et al.: Brain Res. Bull., 73, 231 (2007),

Formula: C₁₇H₂₃N₃O·C₄H₄O₄

Colore e forma: White

Peso molecolare: 401.46

Ref: TR-P997225

Pyrilamine maleate

CAS: 59-33-6

Pyrilamine maleate salt is a reagent used for optical rotation measurements. It is also known to be an antihistamine that has been shown to have mutagenic effects on Salmonella typhimurium and other bacteria. Pyrilamine maleate salt inhibits potassium ion transport across the cell membrane, which can lead to hyperpolarization of the cell membrane and inhibition of the uptake of sodium ions. This inhibition leads to an increase in intracellular sodium concentrations, which in turn leads to decreased ATP production.

Formula: C₁₇H₂₃N₃O•C₄H₄O₄

Purezza: Min. 95%

Colore e forma: Powder

Peso molecolare: 401.46 g/mol

Ref: 3D-FP27345

Pyrilamine-D6 Maleate Salt

Prodotto controllato

CAS: 59-33-6

Formula: C₁₇H₁₇D₆N₃O•C₄H₄O₄

Colore e forma: Neat

Peso molecolare: 407.5

Ref: TR-P997236