CAS 713544-47-9

APETx2

CAS: 713544-47-9

ASIC3 inhibitor; IC50: 63 nM (rat), 175 nM (human). Blocks NaV1.8, NaV1.2; analgesic for acid/inflammatory pain.

Formula: C₁₉₆H₂₈₀N₅₄O₆₁S₆

Purezza: 98%

Colore e forma: Solid

Peso molecolare: 4561.06

Ref: TM-TP2081

APETx2

CAS: 713544-47-9

APETx2 is a peptide that belongs to the inhibitor class of protein interactions. It has been shown to inhibit the activation of beta-adrenergic receptors by preventing the binding of the ligand, which is a catecholamine. APETx2 also has been shown to be an activator for muscarinic acetylcholine receptors. This peptide is a high purity research tool that can be used as an antibody conjugate in immunohistochemical and immunoprecipitation assays.

Formula: C₁₉₆H₂₈₀N₅₄O₆₁S₆

Purezza: Min. 95%

Peso molecolare: 4,561 g/mol

Ref: 3D-APE-4472-S

APETx2

CAS: 713544-47-9

APETx2 is a drug that inhibits the activity of apetx2, a protein which is involved in the regulation of ion channels and endothelin-A receptors. APETx2 has been shown to inhibit the activity of channels involved in pain perception and may have therapeutic potential as a pressor agent. This drug has also been shown to have anti-inflammatory properties, which are likely due to its inhibition of EGF receptor activity. The mechanism of action for this drug remains unclear, but it may work by blocking the channel or receptor for EGF.

Formula: C₁₉₆H₂₈₀N₅₄O₆₁S₆

Purezza: Min. 95%

Peso molecolare: 4,561 g/mol

Ref: 3D-NDB54447