CAS 808-71-9

Idrioduro di penetamato

Descrizione:

Idrioduro di penetamato è un composto chimico utilizzato principalmente come antistaminico e agente antiallergico. È classificato come un composto di ammonio quaternario ed è noto per la sua capacità di inibire l'azione dell'istamina, alleviando così i sintomi allergici. La sostanza appare come una polvere cristallina bianca o bianco sporco ed è solubile in acqua, il che facilita il suo utilizzo in varie formulazioni farmaceutiche. Idrioduro di penetamato viene spesso somministrato sotto forma di compresse orali o soluzioni. Il suo meccanismo d'azione implica il blocco dei recettori H1, responsabili della mediazione delle risposte allergiche. Inoltre, può presentare effetti sedativi lievi, rendendolo utile nel trattamento di condizioni come la rinite allergica e l'orticaria. I profili di sicurezza ed efficacia sono ben documentati, ma come tutti i farmaci, può avere effetti collaterali, tra cui sonnolenza o secchezza delle fauci. Devono essere seguite linee guida adeguate per il dosaggio e la somministrazione per minimizzare gli effetti avversi e garantire l'efficacia terapeutica.

Formula: C₂₂H₃₁N₃O₄S·HI

InChI: InChI=1S/C22H31N3O4S.HI/c1-5-24(6-2)12-13-29-21(28)18-22(3,4)30-20-17(19(27)25(18)20)23-16(26)14-15-10-8-7-9-11-15;/h7-11,17-18,20H,5-6,12-14H2,1-4H3,(H,23,26);1H/t17-,18+,20-;/m1./s1

InChI key: InChIKey=XWRCFDRXQPRCCO-FLQNVMKHSA-N

SMILES: C(OCCN(CC)CC)(=O)[C@@H]1N2[C@@]([C@H](NC(CC3=CC=CC=C3)=O)C2=O)(SC1(C)C)[H].I

Sinonimi:

• 2-(diethylamino)ethyl (2S,5R,6R)-3,3-dimethyl-7-oxo-6-[(phenylacetyl)amino]-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylate hydroiodide (1:1)
• 4-Thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid, 3,3-dimethyl-7-oxo-6-(2-phenylacetamido)-, 2-(diethylamino)ethyl ester, monohydriodide
• 4-Thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid, 3,3-dimethyl-7-oxo-6-[(phenylacetyl)amino]- (2S,5R,6R)-, 2-(diethylamino)ethyl ester, monohydriodide
• 4-Thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid, 3,3-dimethyl-7-oxo-6-[(phenylacetyl)amino]- [2S-(2α,5α,6β)]-, 2-(diethylamino)ethyl ester, monohydriodide
• 4-Thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid, 3,3-dimethyl-7-oxo-6-[(phenylacetyl)amino]-, 2-(diethylamino)ethyl ester, hydriodide (1:1), (2S,5R,6R)-
• Alivin
• Benzylpenicillin β-diethylaminoethyl ester hydriodide
• Bronchocillin
• Bronchopen
• Broncopen
• Deripen
• Diethylaminoethyl ester penicillin hydriodide
• Eficillin
• Ephicillin hydriodide
• Estopen
• Leocillin
• Mamyzin
• Neo-Penil
• Penethacillin
• Penethamate Hydriodide
• Penethecillin
• Penicillin G diethylaminoethyl ester hydriodide
• Penicillin G, 2-(diethylamino)ethyl ester, hydriodide
• Penicillin, 2-(diethylamino)ethyl ester, hydriodide
• Pulmaxil N
• Pulmo 500

Penethacillin Hydroiodide (Penethamate Hydroiodide)

CAS: 808-71-9

Formula: C₂₂H₃₁N₃O₄SHI

Colore e forma: White To Off-White Solid

Peso molecolare: 433.57 127.91

Ref: 4Z-P-182001

Benzylpenicillin Diethylaminoethyl Ester Hydroiodide

Prodotto controllato

CAS: 808-71-9

Applications Benzylpenicillin Diethylaminoethyl Ester Hydroiodide is a prodrug of Benzylpenicillin. It is an antimicrobial/antibacterial agent that is used primarily in the treatment of bovine mastitis.
References Sandgren, C. et al.: Veterin. J., 175, 108 (2008); McDougall, S. et al.: J. Dairy, Sci., 92, 4421 (2009);

Formula: C₂₂H₃₂IN₃O₄S

Colore e forma: Neat

Peso molecolare: 561.48

Ref: TR-B288590

Benzylpenicillin diethylaminoethyl ester hydroiodide

CAS: 808-71-9

Benzylpenicillin diethylaminoethyl ester hydroiodide is a potent broad-spectrum antimicrobial agent that inhibits the growth of bacteria by inhibiting protein synthesis. It is used to treat microbial infections and has been shown to be effective against Streptococcus species, including Streptococcus pneumoniae, Streptococcus pyogenes, and Streptococcus viridans. Benzylpenicillin diethylaminoethyl ester hydroiodide binds to the 50S ribosome subunit of bacteria and prevents the formation of an antibiotic-inhibitor complex with the enzyme cell wall synthesis that is required for cell wall biosynthesis. This binding prevents protein synthesis and cell division.

Formula: C₂₂H₃₂IN₃O₄S

Purezza: Min. 95%

Peso molecolare: 561.5 g/mol

Ref: 3D-AAA80871

Penethamate hydriodide

CAS: 808-71-9

Penethamate hydriodide is a diethylaminoethyl ester prodrug of penicillin, utilized via intramuscular injection to treat mastitis in cattle.

Formula: C₂₂H₃₂IN₃O₄S

Colore e forma: Solid

Peso molecolare: 561.477

Ref: TM-T206114