CAS 83002-04-4

5-(1,1-Dimetileptil)-2-[(1R,2R,5R)-5-idrossi-2-(3-idrossipropil)cicloesil]fenolo

Descrizione:

La sostanza chimica nota come 5-(1,1-Dimetileptil)-2-[(1R,2R,5R)-5-idrossi-2-(3-idrossipropil)cicloesil]fenolo, con il numero CAS 83002-04-4, è un composto sintetico principalmente riconosciuto per la sua applicazione nel campo della ricerca sui cannabinoidi. Questo composto presenta una struttura molecolare complessa che include un gruppo fenolico e un moiety ciclopentilico, che contribuiscono alla sua potenziale attività biologica. È caratterizzato dalla sua natura idrofobica a causa della presenza di lunghe catene alchiliche, che possono influenzare la sua solubilità e interazione con le membrane biologiche. La stereochimica indicata dalla configurazione (1R,2R,5R) suggerisce disposizioni spaziali specifiche che possono influenzare le proprietà farmacologiche del composto. Come analogo dei cannabinoidi, può interagire con i recettori dei cannabinoidi nel corpo, influenzando potenzialmente vari processi fisiologici. Tuttavia, sono necessari studi dettagliati per comprendere appieno la sua efficacia, sicurezza e potenziali applicazioni terapeutiche.

Formula: C₂₄H₄₀O₃

InChI: InChI=1S/C24H40O3/c1-4-5-6-7-14-24(2,3)19-11-13-21(23(27)16-19)22-17-20(26)12-10-18(22)9-8-15-25/h11,13,16,18,20,22,25-27H,4-10,12,14-15,17H2,1-3H3/t18-,20-,22-/m1/s1

InChI key: InChIKey=YNZFFALZMRAPHQ-SYYKKAFVSA-N

SMILES: C(CCO)[C@H]1[C@@H](C[C@H](O)CC1)C2=C(O)C=C(C(CCCCCC)(C)C)C=C2

Sinonimi:

• (-)-Cp 55940
• 2-[(1S,2R,5S)-5-hydroxy-2-(3-hydroxypropyl)cyclohexyl]-5-(2-methyloctan-2-yl)phenol
• 5-(1,1-Dimethylheptyl)-2-[(1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohexyl]phenol
• 5-(1,1-dimethylheptyl)-2-[(1S,2R,5S)-5-hydroxy-2-(3-hydroxypropyl)cyclohexyl]phenol
• Phenol, 5-(1,1-dimethylheptyl)-2-[5-hydroxy-2-(3-hydroxypropyl)cyclohexyl]-, (1α,2β,5α)-(-)-
• phenol, 5-(1,1-dimethylheptyl)-2-[(1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohexyl]-
• phenol, 5-(1,1-dimethylheptyl)-2-[(1S,2R,5S)-5-hydroxy-2-(3-hydroxypropyl)cyclohexyl]-

CP-55940

CAS: 83002-04-4

Formula: C₂₄H₄₀O₃

Peso molecolare: 376.57

Ref: 7W-GL0738

(-)-CP 55,940 (10 mg/mL in methanol)

Prodotto controllato

CAS: 83002-04-4

Applications CP 55,940 is a cannabinoid agonist which is considerably more potent than Δ9-THC in both behavioral tests and receptor binding assays. Displays high and roughly equal affinity for both central and peripheral cannabinoid receptors (Ki = 0.6 - 5.0 and 0.7 - 2.6 nM at CB1 and CB2 respectively; EC50 values are 0.2, 0.3 and 5 nM at CB1, CB2 and GRP55 respectively).Controlled substance. Synthetic Cannabinoids
References Wiley, et al.: Neuropharmacology, 34, 669 (1995); Griffin, et al.: J. Pharmacol. Exp. Ther., 285, 553 (1998); Thomas, et al.: J. Pharmacol. Exp. Ther., 285, 285 (1998); Ryberg, et al.: Br. J. Pharmacol., 152, 1092 (2007);

Formula: C₂₄H₄₀O₃

Colore e forma: Single Solution

Peso molecolare: 376.57

Ref: TR-C781410

CP 55940

Prodotto controllato

CAS: 83002-04-4

CP 55940 is a cannabinoid receptor agonist that inhibits acetylcholine release in the brain and has been shown to cause neuronal death. CP 55940 binds to the α7 nicotinic acetylcholine receptor, which is important for memory and learning. The binding of this drug causes an increase in guanine nucleotide-binding protein (G protein) activity by reducing the rate of GTP hydrolysis, leading to inhibition of adenylyl cyclase activity and subsequent decrease in cAMP levels. CP 55940 has significant up-regulation of toll-like receptors following exposure, which leads to an increased immune response. This drug can also cause bowel disease or side effects such as seizures and psychotic symptoms. CP 55940 can interact with other drugs, including cannabinoids that may lead to serious side effects.

Formula: C₂₄H₄₀O₃

Purezza: Min. 95%

Peso molecolare: 376.57 g/mol

Ref: 3D-FD146910