Endocrinologia/Ormoni
Gli inibitori dell'endocrinologia/oromone sono composti che bloccano l'azione degli ormoni o interferiscono con le vie di segnalazione ormonale. Questi inibitori sono fondamentali per studiare la regolazione dei sistemi endocrini e per sviluppare trattamenti per malattie correlate agli ormoni, come il diabete, i disturbi della tiroide e i tumori ormono-dipendenti. Modulando l'attività ormonale, questi inibitori possono aiutare a chiarire le complesse interazioni all'interno del sistema endocrino. Presso CymitQuimica, offriamo un'ampia gamma di inibitori di alta qualità per endocrinologia/oromone per supportare le tue ricerche in endocrinologia, farmacologia e scienze mediche.
Sottocategorie di "Endocrinologia/Ormoni"
- Recettore degli androgeni(229 prodotti)
- Annessina A(16 prodotti)
- Aromatasi(22 prodotti)
- Recettore degli estrogeni/progestogeni(57 prodotti)
- GPR(1 prodotti)
- Recettore dei glucocorticoidi(166 prodotti)
- LHRH(1 prodotti)
- Recettore degli oppioidi(326 prodotti)
- Recettore della prostaglandina(122 prodotti)
- RAAS(90 prodotti)
- Riduttasi(50 prodotti)
- Somatostatina(57 prodotti)
- Recettore dell'ormone tiroideo (THR)(32 prodotti)
- Recettore della vasopressina(48 prodotti)
Mostrare 6 più sottocategorie
Trovati 3371 prodotti di "Endocrinologia/Ormoni"
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DPP-4/GPR119 modulator 1
CAS:Orally active DPP-4 inhibitor/GPR119 agonist, Compound 22 lowers glucose, moderate hERG inhibition, IC50 4.9 µM, for diabetes research.Formula:C30H39ClN10O3Colore e forma:SolidPeso molecolare:623.15(d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin
CAS:(d(CH2)51,Tyr(Me)2, Orn8)-Oxytocin (OVT) is an antagonist of the oxytocin receptor that finds application in the study of neurological diseases [1].Formula:C48H74N12O12S2Purezza:98%Colore e forma:SolidPeso molecolare:1075.3Bexirestrant
CAS:Bexirestrant is an orally active ER-α degrader commonly employed in the research of antiestrogen and antineoplastic therapies.Formula:C29H26F3NO2Colore e forma:SolidPeso molecolare:477.527Ganoderic acid Df
CAS:<p>Ganoderic acid Df, a lanostane triterpenoid from Ganoderma lucidum, inhibits aldose reductase with IC50 of 22.8 μM.</p>Formula:C30H44O7Colore e forma:SolidPeso molecolare:516.67Deltorphin acetate
Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioidFormula:C46H66N10O12S2Purezza:98.93%Colore e forma:SolidPeso molecolare:1015.21Ref: TM-T20166L
1mg185,00€5mg415,00€10mg622,00€25mg1.119,00€50mg1.679,00€100mg2.520,00€200mg3.780,00€Inocoterone acetate
CAS:Inocoterone acetate is a nonsteroidal antiandrogen that binds to the androgen receptor and possesses antiandrogenic activity in animal models.Formula:C18H26O3Colore e forma:SolidPeso molecolare:290.40NH-3
CAS:NH-3, an orally active THR antagonist with a 55 nM IC50, blocks thyroid hormone binding and cofactor recruitment.Formula:C28H27NO6Purezza:97.79% - 99.40%Colore e forma:SolidPeso molecolare:473.52Ref: TM-T40548
1mg217,00€5mg550,00€10mg792,00€25mg1.206,00€50mg1.605,00€100mg2.175,00€500mg4.389,00€1mL*10mM (DMSO)492,00€AM-5262
CAS:AM-5262 is a potent GPR40 Full Agonist with improved rat PK profile and general selectivity profile.Formula:C33H35FO4Colore e forma:SolidPeso molecolare:514.63ER degrader 4
CAS:ER degrader 4, a selective and orally active compound, effectively degrades estrogen receptors and exhibits anti-tumor activity [1].Formula:C26H19FO4SColore e forma:SolidPeso molecolare:446.49Leumorphin, human
CAS:Leumorphin, human, is a potent agonist of the kappa opioid receptor (κ opioid receptor) and inhibits the contraction of the guinea pig ileum's myenteric plexus-Formula:C150H224N42O46Purezza:98%Colore e forma:SolidPeso molecolare:3351.64Saprisartan
CAS:Saprisartan (GR-138950, GR-138950X) is an AT1 receptor antagonist used for the treatment of heart failure and blood pressure.Formula:C25H22BrF3N4O4SColore e forma:SolidPeso molecolare:611.43AH 7563
CAS:AH 7563 is structurally classified as an opioid compound with analgesic properties. In mice, its ED50 for pain relief was 15.3 mg/kg when administered orally in the Phenylquinone test, and 15.5 mg/kg when injected subcutaneously in the Hot plate test.Formula:C16H24N2OColore e forma:SolidPeso molecolare:260.38U-48520
CAS:U-48520 is an agonist of the μ-opioid receptor (μ-opioid receptor) with an EC50 of 1561 nM.Formula:C16H23ClN2OColore e forma:SolidPeso molecolare:294.82(-)-9-Hydroxycorynantheidine
CAS:(-)-9-Hydroxycorynantheidine (9-O-Desmethyl mitragynine) is a demethylated analog of Mitragynine, functioning as a selective and partial agonist for the μ-opioid receptor (μ-opioid receptor). This compound inhibits electrically stimulated twitch contractions in the guinea pig ileum.Formula:C22H28N2O4Colore e forma:SolidPeso molecolare:384.47Antidiabetic agent 15
<p>Antidiabetic agent 15 (compound 1B15) acts as a dual inhibitor of AT1R and NEP, reducing oxidative stress and restoring mitochondrial membrane potential.</p>Formula:C26H23NO5Colore e forma:SolidPeso molecolare:429.15762Nurr1 agonist 12
Nurr1 agonist 12 (Compound 37) acts as an agonist of the nuclear receptor-related protein 1 (Nurr1), enhancing its transcriptional activity with an EC50 of 0.06 μM. It stimulates human response elements NBRE, NurRE, and DR5 with EC50 values of 0.07 μM, 0.027 μM, and 0.014 μM, respectively. Additionally, Nurr1 agonist 12 induces the expression of neurotrophic genes regulated by Nurr1, such as tyrosine hydroxylase (TH), SOD1/2, BDNF, Sestrin 3, and BIRC5 (Survivin). The compound also demonstrates neuroprotective effects against neurotoxicity caused by Paraquat.Formula:C18H12ClN3OColore e forma:SolidPeso molecolare:321.76MOR agonist-2
Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM.Formula:C37H47Cl2N5O3Purezza:98%Colore e forma:SolidPeso molecolare:680.71WAY-298630
CAS:Fluorophenoxy benzimidazole, a CRTH2 blocker, IC50 < 10 μM for rhinitis, COPD, arthritis, eczema, conjunctivitis.Formula:C17H15FN2O3SPurezza:97.84%Colore e forma:SolidPeso molecolare:346.38Pro8-Oxytocin TFA
<p>Pro8-Oxytocin TFA, a modified oxytocin (OXT) ligand, exhibits greater potency and efficacy than the standard mammalian OXT ligand, Leu8-Oxytocin, at primate</p>Formula:C42H62N12O12S2·xC2HF3O2Purezza:98%Colore e forma:SolidMyrciacetin
CAS:Myrciacetin from Rhododendron inhibits rat aldose reductase with IC50 of 13 μM.Formula:C17H16O6Colore e forma:SolidPeso molecolare:316.309
