Somatostatina
La somatostatina è un ormone peptidico che inibisce il rilascio di diversi altri ormoni, tra cui l'ormone della crescita, l'insulina e il glucagone. Agisce legandosi ai recettori della somatostatina, che sono recettori accoppiati alle proteine G espressi in vari tessuti. Gli analoghi della somatostatina sono utilizzati nel trattamento dell'acromegalia, dei tumori neuroendocrini e dei disturbi gastrointestinali. Questi analoghi sono anche strumenti preziosi per lo studio della secrezione ormonale e della segnalazione. Presso CymitQuimica, offriamo una gamma completa di analoghi della somatostatina di alta qualità per supportare la tua ricerca in endocrinologia, regolazione ormonale e sviluppo terapeutico.
Trovati 54 prodotti di "Somatostatina"
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(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid
CAS:(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.Formula:C20H29N3O8Purezza:99.72%Colore e forma:SoildPeso molecolare:439.46Somatostatin acetate
<p>Somatostatin acetate is an endogenously secreted inhibitor of cell proliferation with potential antitumor activity for the study of cancer and neurological disorders.</p>Purezza:99.11%Colore e forma:Odour SolidCortistatin 14, human, rat acetate
Cortistatin 14, human, rat acetate is a neuropeptide having structural similarity to somatostatin-14 and shows anticonvulsive, neuroprotective effects andFormula:C80H112N18O19S2Purezza:97.86%Colore e forma:SolidPeso molecolare:1693.98Cortistatin-14 acetate
<p>Cortistatin-14 acetate, a neuropeptide have structural similarity to somatostatin-14, binds and exerts its function via the somatostatin receptors (sst1-sst5).</p>Formula:C83H118N20O20S2Purezza:98.24% - 99.63%Colore e forma:SoildPeso molecolare:1780.08Seglitide acetate
CAS:<p>Seglitide acetate (MK-678) is a selective agonist of sst2 somatostatin receptor.</p>Formula:C46H60N8O9Purezza:98.87%Colore e forma:SolidPeso molecolare:869.02Seglitide
CAS:<p>Peptide agonist targets sst2/sst5 receptors. IC50/Kd: sst1 >1000, sst2 = 0.2-1.5, sst3 = 27-36, sst4 >127, sst5 = 0.06-23 nM.</p>Formula:C44H56N8O7Purezza:98%Colore e forma:SolidPeso molecolare:808.98Ilatreotide
CAS:Ilatreotide is a Amadori compound of octreotide.Formula:C61H86N10O20S2Purezza:98%Colore e forma:SolidPeso molecolare:1343.53CYN 154806
CAS:CYN 154806: potent sst2 antagonist; pIC50: 8.58 (sst2), 5.41 (sst1), 6.07 (sst3), 5.76 (sst4), 6.48 (sst5).Formula:C56H68N12O14S2Purezza:98%Colore e forma:SolidPeso molecolare:1197.34Cortistatin 14, human, rat
CAS:Cortistatin 14: a neuropeptide similar to somatostatin; induces sleep, depresses neuronal activity; found in cortex, hippocampus.Formula:C81H113N19O19S2Purezza:98%Colore e forma:SolidPeso molecolare:1721.01Veldoreotide
CAS:Veldoreotide (Somatoprim): a somatostatin analogue targeting receptors 2, 4, 5, reduces GH in pituitary adenomas.Formula:C60H74N12O10Purezza:98%Colore e forma:SolidPeso molecolare:1123.3Somatostatin(3-6)
CAS:Somatostatin(3-6) is a somatostatin fragment.Formula:C22H34N6O6SColore e forma:SolidPeso molecolare:510.61MMC(TMZ)-TOC TFA
MMC(TMZ)-TOC TFA exhibits high binding affinity and selectivity for the somatostatin receptor subtype 2 (SSTR2). It targets the delivery of TMZ to SSTR2-positive tumor cells, making MMC(TMZ)-TOC TFA useful for cancer research.Formula:C74H99F3N20O21S2Colore e forma:SolidPeso molecolare:1725.82Somatostatin
CAS:Somatostatin: a peptide hormone inhibiting growth hormone, insulin, and glucagon; secreted by hypothalamus and pancreatic D cells.Purezza:98%Colore e forma:PowderPeso molecolare:1637.88CH 275
CAS:Potent sst1 agonist with 30.9 nM IC50; selective over sst2-5; inhibits somatostatin in rat nucleus accumbens.Formula:C74H96N14O15S2Purezza:98%Colore e forma:SolidPeso molecolare:1485.8MMC(TMZ)-TOC
MMC(TMZ)-TOC exhibits a high binding affinity and selectivity for somatostatin receptor subtype 2 (SSTR2). It is designed to target and deliver TMZ specifically to SSTR2-positive tumor cells. MMC(TMZ)-TOC is applicable for cancer research.Formula:C72H98N20O19S2Peso molecolare:1610.67585Somatostatin-28 (1-14)
CAS:Somatostatin-28 (1-14) is a truncated neuropeptide from prosomatostatin cleavage.Formula:C61H105N23O21SPurezza:98%Colore e forma:SolidPeso molecolare:1528.71Cortistatin 29
Cortistatin 29: neuropeptide, relieves neuropathic pain, binds SS receptors (IC50: 2.8-13.7 nM), anti-fibrotic.Formula:C161H242N46O41S2Colore e forma:SolidPeso molecolare:3539.77Satoreotide
CAS:Satoreotide (JR11) is an SSTR2 antagonist, typically conjugated with radiolabeled chelators for use in neuroendocrine tumor imaging [1].Formula:C58H72ClN15O14S2Colore e forma:SolidPeso molecolare:1302.87L-796,778
CAS:<p>L-796,778 is an SST3 agonist and a selective ligand of SST3, which can increase the level of cAMP in the body.</p>Formula:C29H40N6O7Purezza:96.20%Colore e forma:SolidPeso molecolare:584.66BIM-23190 hydrochloride
<p>BIM-23190 hydrochloride, somatostatin analog, SSRT2/5 agonist, Ki: 0.34 nM (SSTR2), 11.1 nM (SSTR5). Used in cancer, acromegaly research.</p>Colore e forma:LiquidDOTA-JR11
CAS:DOTA-JR11 is a somatostatin receptor 2 (SSTR2) antagonist that can be radiolabeled with 68Ga.Formula:C74H98ClN19O21S2Colore e forma:SolidPeso molecolare:1689.27Dotanoc
CAS:Dotanoc is a ligand to make gallium Ga 68-DOTANOC, which is a gallium Ga 68-radiolabeled analog of somatostatin.Formula:C69H94N14O17S2Colore e forma:SolidPeso molecolare:1455.71Cyclic SSTR agonist octreotide
Cyclic SSTR agonist octreotide is a Octreotide , serving as the cyclic Somatostatin Receptor SSTR agonist [1] .Formula:C53H71N11O14S2Colore e forma:SolidPeso molecolare:1150.33Cyclosomatostatin TFA
Cyclosomatostatin TFA blocks SST receptor, reduces CRC cell growth, ALDH+ size, and sphere-formation.Formula:C46H58F3N7O8Colore e forma:SolidPeso molecolare:893.99L-796,778 acetate
L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for sst1, sst2, sst4 and sst5, IC50 is >1000nM.Formula:C31H44N6O9Purezza:98%Colore e forma:SoildPeso molecolare:644.72Tau conotoxin CnVA
CAS:Tau conotoxin CnVA, a small peptide found in the venom of Conus consors (cone snail), is a member of the T1 cone snail peptide superfamily. It demonstrates high selectivity for the somatostatin sst3 receptor with a Ki value of 1.5 µM. Tau conotoxin CnVA is unique as the only known toxin interacting with this subfamily of G protein-coupled receptors (GPCR). This compound is useful for research related to diseases associated with the sst3 receptor, such as pancreatic cancer or pituitary adenomas.Formula:C72H116N24O17S4Colore e forma:SolidPeso molecolare:1718.1SSTR4 agonist-1
CAS:<p>SSTR4agonist-1 (Compound 47) is a selective agonist of the somatostatin receptor 4 (SSTR4), with an EC50 of 4.7 nM. It has a half-life of over 130 minutes in human liver microsomes.</p>Formula:C16H23N3O2Colore e forma:SolidPeso molecolare:289.37Ref: 4Z-PS-219001
5mgPrezzo su richiesta10mgPrezzo su richiesta25mgPrezzo su richiesta50mgPrezzo su richiesta100mgPrezzo su richiestaL-797,591 hydrochloride
L-797,591 HCl activates SSTR1, boosts p-ERK5 with AG1478, and enhances p38 phosphorylation, reversible by AG1478.Formula:C38H50ClN5O2Purezza:98.65% - >99.99%Colore e forma:SoildPeso molecolare:644.30Neuronostatin-13 (human)
CAS:Neuronostatin-13: human-conserved, 13-amino-acid peptide with amidated C-terminus.Formula:C64H110N20O16Purezza:98%Colore e forma:SolidPeso molecolare:1415.68[D-Trp8,Tyr11] Somatostatin
CAS:[D-Trp8,Tyr11] Somatostatin, an analogue of the hormone somatostatin that modulates numerous bodily functions, is characterized by the substitution of DTrp8,Formula:C76H104N18O20S2Peso molecolare:1653.88[Tyr11]-Somatostatin
CAS:[Tyr11]-Somatostatin, a neuroactive peptide, aids proteomics research and modulates retinal function.Formula:C76H104N18O20S2Peso molecolare:1653.89DOTA-EB-TATE
DOTA-EB-TATE is formed by combining the SST peptide derivative DOTA-octreotate with an Evans blue analog (EB). This peptide drug conjugate (PDC) enhances the pharmacokinetics of SSTR2 analogs and reduces PRRT toxicity. Additionally, DOTA-EB-TATE serves in the synthesis/research of radiopharmaceutical conjugates (RDC).Formula:C105H133N21O30S5Peso molecolare:2329.63Cortistatin-14
CAS:Cortistatin-14, a neuropeptide structurally similar to growth inhibitor-14, is used to study sepsis-induced cognitive impairment.Formula:C81H114N20O18S2Purezza:98.06% - 98.23%Colore e forma:SolidPeso molecolare:1720.03Cyclosomatostatin Acetate
<p>Cyclosomatostatin Acetate is an effective antagonist of the somatostatin receptor.Cyclosomatostatin Acetate inhibits SSTR1 signaling and decreases cell</p>Formula:C46H61N7O8Purezza:98.83%Colore e forma:SolidPeso molecolare:840.02L803
CAS:L803 is a selective somatostatin receptor type 4 (SST4) agonist that can inhibit L-type calcium channel currents (ICa). It holds potential for research into degenerative diseases of retinal ganglion cells (RGC), such as glaucoma.Formula:C50H80N13O19PColore e forma:SolidPeso molecolare:1198.22Somatostatin 1-28 acetate
Somatostatin 1-28 acetate circulates in human plasma.Purezza:99.22%Colore e forma:Soild(D-Phe5,Cys6,11,N-Me-D-Trp8)-Somatostatin-14 (5-12) amide
CAS:Somatostatin analog (Compound 4) with Kd: SSTR5-0.61nM, SSTR3-11.05nM, SSTR2-23.5nM, SSTR1-1.2µM, SSTR4->1µM.Formula:C50H67N11O10S2Peso molecolare:1046.26[Tyr1]-Somatostatin-14
CAS:[Tyr1]-Somatostatin-14 could binds to SSTR2.Formula:C82H108N18O20S2Peso molecolare:1729.99Anti-Somatostatin Antibody (9L93)
Anti-Somatostatin Antibody (9L93) is a Rabbit antibody targeting Somatostatin. Anti-Somatostatin Antibody (9L93) can be used in ELISA.Colore e forma:Odour LiquidLanreotide
CAS:Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.Formula:C54H69N11O10S2Colore e forma:SolidPeso molecolare:1096.32BIM-23190 aceate
<p>BIM-23190 aceate, a somatostatin analog, a selective agonist of SSTR2 and SSTR5. BIM-23190 can be used in cancer and acromegaly studies.</p>Formula:C59H83N13O14S2Purezza:99.7%Colore e forma:SolidPeso molecolare:1262.5Paltusotine
CAS:Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.Formula:C27H22F2N4OPurezza:99.91%Colore e forma:SolidPeso molecolare:456.49Pasireotide Acetate
CAS:The pKi of Pasireotide (SOM230) acetate for sst1, 2, 3, 4, and 5 were 8.2, 9.0, 9.1, less than 7.0, and 9.9, respectively.Cost-effective and quality-assured.Formula:C60H70N10O11Purezza:98.64% - 99.92%Colore e forma:SolidPeso molecolare:1107.26Ref: 4Z-PS-219002
5mgPrezzo su richiesta10mgPrezzo su richiesta25mgPrezzo su richiesta50mgPrezzo su richiesta100mgPrezzo su richiestaOctreotide Acetate
CAS:Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.Formula:C51H70N10O12S2Purezza:99.03% - 99.87%Colore e forma:Less To Off-White Lyophilised Solid Colourless To Off-White Lyophilised SolidPeso molecolare:1079.3FK962
CAS:FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.Formula:C14H17FN2O2Purezza:99.89%Colore e forma:SolidPeso molecolare:264.3Somatostatin Impurity 2 (13-Dha) Trifluoroacetate
Formula:C76H102N18O18S2·C2HF3O2Peso molecolare:1619.88 114.02Ref: 4Z-PS-219003
5mgPrezzo su richiesta10mgPrezzo su richiesta25mgPrezzo su richiesta50mgPrezzo su richiesta100mgPrezzo su richiestaCYN 154806 TFA
CAS:CYN 154806 TFA: cyclic octapeptide, selective somatostatin sst2 antagonist; pIC50: sst2 - 8.58, sst1 - 5.41, sst3 - 6.07, sst4 - 5.76, sst5 - 6.48.Formula:C58H69F3N12O16S2Purezza:99.7%Colore e forma:SolidPeso molecolare:1311.36Edotreotide
CAS:Edotreotide (SMT-487) is an Indicator and Reagent. It also is used in the Diagnosis and Staging of Tumors Expressing Somatostatin Receptors.Formula:C65H92N14O18S2Purezza:96.95%Colore e forma:SolidPeso molecolare:1421.64
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