
RAAS
Gli inibitori del sistema renina-angiotensina-aldosterone (RAAS) sono composti che prendono di mira la via del RAAS, nota principalmente per il suo ruolo nella regolazione della pressione sanguigna e dell'equilibrio dei fluidi, ma che influenza anche l'angiogenesi. La via del RAAS può contribuire allo sviluppo di nuovi vasi sanguigni nei tumori, supportandone così la crescita. Inibire i componenti del RAAS può quindi avere effetti anti-angiogenici, rendendo questi inibitori preziosi nel trattamento di alcuni tumori e disturbi vascolari. Presso CymitQuimica, offriamo una gamma di inibitori di alta qualità del RAAS per supportare la tua ricerca in biologia cardiovascolare, oncologia e angiogenesi.
Trovati 92 prodotti per "RAAS".
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
[Sar1, Ile8]-Angiotensin II acetate
'[Sar1, Ile8]-Angiotensin II acetate triggers oxidases and prompts superoxide in muscles; has varied vascular impacts.Formula:C48H77N13O12Purezza:99.36%Colore e forma:SolidPeso molecolare:1028.2Ref: TM-T7575L1
2mg34,00€5mg46,00€10mg60,00€1mL*10mM (DMSO)90,00€25mg119,00€50mg192,00€100mg289,00€200mg415,00€Handle region peptide, rat
CAS:Rat handle region peptide acts as prorenin receptor blocker, curbs diabetic kidney disease, and reduces eye inflammation.Formula:C54H101N15O12SPurezza:98%Colore e forma:SolidPeso molecolare:1184.54Alunacedase alfa
CAS:Alunacedase alfa (APN-01) is an angiotensin-converting enzyme 2 with antiviral activity.Purezza:99.1% (SDS-PAGE); 99.9% (SEC-HPLC) - 99.1% (SDS-PAGE); 99.9% (SEC-HPLC)Colore e forma:LiquidPeso molecolare:85.03 kDaTRV056
CAS:TRV056 is a Gq-biased AT1R agonist effective in Gq-mediated signaling and a basis for similar drug development.Formula:C52H74N14O13Colore e forma:SolidPeso molecolare:1103.249[Sar1, Ile8]-Angiotensin II TFA
[Sar1,Ile8]-Angiotensin II (TFA) contracts arteries and affects cell growth in vascular muscle.Formula:C48H74F3N13O12Purezza:98%Colore e forma:SolidPeso molecolare:1082.18Evazarsen sodium
CAS:Evazarsen sodium, an angiotensinogen synthesis inhibitor, possesses antihypertensive properties [1].Formula:C296H414N86O146P20S19Na20Colore e forma:SolidPeso molecolare:9201.6TRV120055
CAS:TRV120055 is a Gq-biased agonist with 10x more efficacy on AT1R-Gq than AT1R-βarr2.Formula:C34H54N12O7Peso molecolare:742.883Angiotensin II (3-8), human TFA
Angiotensin II (3-8), human (TFA) is an angiotensin AT1 receptor agonist with less activity.Formula:C42H55F3N8O10Purezza:98%Colore e forma:SolidPeso molecolare:888.93Angiotensin II (1-4), human TFA
Angiotensin II is a potent direct vasoconstrictor, causing arteries and veins to constrict, so leading to an increase in blood pressure.Formula:C26H38F3N7O10Purezza:98%Colore e forma:SolidPeso molecolare:665.62A 779
CAS:A 779 is a potent antagonist of the G-protein-coupled receptor Mas, the Ang1-7 receptor, which is distinct from conventional AngII.Formula:C39H60N12O11Purezza:98%Colore e forma:SolidPeso molecolare:872.97Angiotensin II (1-4), human
CAS:Angiotensin II constricts blood vessels and boosts blood pressure by escalating norepinephrine release.Formula:C24H37N7O8Purezza:98%Colore e forma:SolidPeso molecolare:551.59PRO20
PRO20 is a specific and competitive antagonist of the (pro)renin receptor (PRR). It inhibits the calcium influx induced by Proproin with an IC50 value of 81 nmol/L. By blocking the binding of Prorenin to PRR, PRO20 inhibits the activation of the renin-angiotensin system (RAS), reducing the production of angiotensin II (Ang II) and exerting antihypertensive effects. PRO20 holds promise for research in antihypertensive agents.Colore e forma:Odour SolidSaralasin
CAS:Competitive non-selective angiotensin II antagonist.Formula:C42H65N13O10Purezza:98%Colore e forma:SolidPeso molecolare:912Angiotensin amide
CAS:Angiotensin amide, an octapeptide amide, can be used to increase blood pressure by vasoconstriction.Formula:C49H70N14O11Purezza:98%Colore e forma:SolidPeso molecolare:1031.17Angiogenin (108-122)
CAS:Angiogenin (108-122) peptide treats cancer, infectious, fibrotic, inflammatory, neurodegenerative, autoimmune, and heart diseases.Formula:C78H125N25O23Colore e forma:SolidPeso molecolare:1780.98Losartan (D4 Carboxylic Acid)
CAS:Losartan D4 Carboxylic Acid is the deuterium labeled Losartan, which is an angiotensin II receptor antagonist.Formula:C22H21ClN6O2Purezza:98%Colore e forma:SolidPeso molecolare:440.919PD 123319 ditrifluoroacetate
CAS:PD 123319 ditrifluoroacetate is a selective non-peptide AT2 receptor antagonist with IC50 of 34 nM.Formula:C35H34F6N4O7Purezza:98%Colore e forma:White SolidPeso molecolare:736.66Angiotensin II 5-valine
CAS:ngiotensin II 5-valine is an angiotensin II analog which is an agonist at angiotensin receptors.Formula:C49H69N13O12Purezza:98%Colore e forma:SolidPeso molecolare:N/AValsartan-D9
CAS:Valsartan D9: deuterium-labeled, angiotensin II receptor antagonist, treats hypertension & heart failure.Formula:C24H29N5O3Purezza:98%Colore e forma:SolidPeso molecolare:444.574Spirapril hydrochloride
CAS:Spirapril hydrochloride (SCH 33844 hydrochloride) is a potent angiotensin converting enzyme inhibitor with antihypertensive activity that competitively blocks the conversion of angiotensin I to angiotensin II, functions as an orally active proagent of spiraprilat, and is extensively utilized in cardiovascular research focused on hypertension and congestive heart failure pathophysiology and therapeutic intervention.Formula:C22H31ClN2O5S2Purezza:99.78%Colore e forma:White SolidPeso molecolare:503.07

