Recettore della vasopressina
I recettori della vasopressina sono una famiglia di recettori accoppiati alle proteine G che mediano gli effetti della vasopressina, un ormone coinvolto nella regolazione dell'equilibrio idrico, della pressione sanguigna e della funzione renale. Gli agonisti e antagonisti dei recettori della vasopressina sono studiati per il loro ruolo nel trattamento di condizioni come il diabete insipido, l'iponatriemia e l'insufficienza cardiaca. Questi recettori sono anche obiettivi importanti nella ricerca sull'equilibrio dei fluidi e sulla salute cardiovascolare. Presso CymitQuimica, offriamo una selezione di modulatori dei recettori della vasopressina di alta qualità per supportare la tua ricerca in endocrinologia, nefrologia e biologia cardiovascolare.
Trovati 46 prodotti di "Recettore della vasopressina"
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Invopressin
CAS:<p>Invopressin (Compound 42), a vasopressin V1A receptor partial agonist (EC50: 1.0 nM), is utilized in research related to cirrhosis conditions such as bacterial</p>Formula:C110H161N31O27S2Purezza:98%Colore e forma:SolidPeso molecolare:2413.78[Deamino-Pen1,Val4,D-Arg8]-vasopressin
CAS:[Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an antagonist of arginine-vasopressin (AVP).Formula:C48H69N13O11S2Purezza:98%Colore e forma:SolidPeso molecolare:1068.27Val9-Oxytocin
CAS:Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete antagonist of the vasopressin (V1a) receptor.Formula:C46H72N12O12S2Purezza:98%Colore e forma:SolidPeso molecolare:1049.27(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
CAS:(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].Formula:C52H76N14O11S2Purezza:98%Colore e forma:SolidPeso molecolare:1137.38V1a/V2 antagonist 1
V1a/V2 antagonist 1 (Compound 18j) is an orally active dual-target antagonist of V1a and V2 receptors, exhibiting high binding affinity toward these receptors [Ki values are hV1a: 0.13 nM, hV2: 0.53 nM, and mV1a: 0.5 nM; IC50 for hV1a is 2.2 nM]. This compound can inhibit oxytocin-induced scratching behavior in mice.Formula:C25H26ClN5O3Colore e forma:SolidPeso molecolare:479.96d[Leu4,Lys8]-VP
CAS:Vasopressin V1B agonist; Ki: 0.16nM V1B, 64nM oxytocin; weak antidiuretic/vasopressor; minimal oxytocic action.Formula:C47H67N11O11S2Purezza:98%Colore e forma:SolidPeso molecolare:1026.2d[Cha4]-AVP TFA
d[Cha4]-AVP TFA: potent, selective V1b agonist, K i 1.2 nM, favors V1b over V1a, V2, oxytocin receptors.Formula:C52H72F3N13O13S2Colore e forma:SolidPeso molecolare:1208.33Atosiban
CAS:Atosiban (RW22164), an oxytocin/vasopressin inhibitor, halts premature labor as an intravenous tocolytic, reducing uterine contractions rapidly.Formula:C43H67N11O12S2Purezza:98%Colore e forma:SolidPeso molecolare:994.19Fedovapagon
CAS:<p>Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.</p>Formula:C27H34N4O3Purezza:99.33%Colore e forma:SolidPeso molecolare:462.58Argipressin
CAS:Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.Formula:C46H65N15O12S2Purezza:98%Colore e forma:White PowderPeso molecolare:1084.23Conopressin S acetate(111317-90-9 free base)
Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1bFormula:C43H77N17O12S2Purezza:99.79%Colore e forma:SolidPeso molecolare:1088.32Desmopressin acetate (16679-58-6 free base)
CAS:Desmopressin (16679-58-6), a synthetic vasopressin analog, treats nocturia, enuresis, and diabetes insipidus by reducing urine production.Formula:C48H68N14O14S2Purezza:98.84% - >99.99%Colore e forma:SolidPeso molecolare:1129.26Fuscoside
CAS:Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.Formula:C26H31N3O4Purezza:98.13% - 99.66%Colore e forma:SolidPeso molecolare:449.54d[Cha4]-AVP acetate(500170-27-4 free base)
'd[Cha4]-AVP acetate: strong V1B agonist, weak on V1A/Oxytocin/V2. Boosts ACTH, corticosterone; low blood pressure effect.'Formula:C52H75N13O13S2Purezza:99.86%Colore e forma:SolidPeso molecolare:1154.37Atosiban acetate
CAS:Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin.Formula:C45H71N11O14S2Purezza:99.84% - 99.92%Colore e forma:SolidPeso molecolare:1054.24Ref: TM-T5148
5mg73,00€10mg115,00€25mg170,00€50mg207,00€100mg268,00€500mg660,00€1mL*10mM (DMSO)134,00€Mozavaptan
CAS:Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.Formula:C27H29N3O2Purezza:98.98% - 99.12%Colore e forma:SolidPeso molecolare:427.54LIXIVAPTAN
CAS:Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)Formula:C27H21ClFN3O2Purezza:98.36%Colore e forma:SolidPeso molecolare:473.93Ref: TM-T7303
2mg37,00€5mg70,00€10mg104,00€25mg216,00€50mg354,00€100mg550,00€200mg785,00€1mL*10mM (DMSO)73,00€Felypressin
CAS:Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.Formula:C46H65N13O11S2Purezza:99.65%Colore e forma:SolidPeso molecolare:1040.22Conivaptan hydrochloride
CAS:<p>Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and</p>Formula:C32H26N4O2·HClPurezza:98.33% - 99.86%Colore e forma:SolidPeso molecolare:535.04Tolvaptan
CAS:<p>Tolvaptan (OPC-41061) is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.</p>Formula:C26H25ClN2O3Purezza:99.78% - >99.99%Colore e forma:SolidPeso molecolare:448.94
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