Recettore della prostaglandina
I recettori delle prostaglandine sono un gruppo di recettori accoppiati alle proteine G che mediano gli effetti delle prostaglandine, composti lipidici coinvolti in una vasta gamma di processi fisiologici, tra cui infiammazione, dolore, febbre e regolazione del flusso sanguigno. I modulatori dei recettori delle prostaglandine sono studiati per il loro ruolo nella gestione delle condizioni infiammatorie, delle malattie cardiovascolari e della salute riproduttiva. Questi recettori sono obiettivi chiave nello sviluppo di farmaci anti-infiammatori e analgesici. Presso CymitQuimica, offriamo una selezione di modulatori dei recettori delle prostaglandine di alta qualità per supportare la tua ricerca in endocrinologia, infiammazione e farmacologia.
Trovati 122 prodotti di "Recettore della prostaglandina"
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EP2 receptor antagonist-2
CAS:<p>CID891729, an EP2 receptor blocker, hinders PGE2 activation and reduces NMDA-induced LDH release.</p>Formula:C15H14F3N3OPurezza:99.95%Colore e forma:SolidPeso molecolare:309.29Isbogrel
CAS:Isbogrel (CV4151) is a TXA2 synthase inhibitor for researching arrhythmias, ischemic attacks, and thrombosis.Formula:C18H19NO2Purezza:99.58%Colore e forma:SolidPeso molecolare:281.35TG6-129
CAS:<p>TG6-129 is an EP2 receptor antagonist, blocking PGE2 effects, reducing inflammatory markers with 1.6 µM IC50.</p>Formula:C20H18FN5O3S3Purezza:99.55%Colore e forma:SolidPeso molecolare:491.58Omidenepag isopropyl
CAS:Omidenepag isopropyl (DE-117) is a prostaglandin EP2 receptor agonist used in the study of glaucoma and hypertension.Formula:C26H28N6O4SPurezza:99.86%Colore e forma:SolidPeso molecolare:520.6Prostaglandin D3
CAS:Prostaglandin D3 (PGD3) functions as an inhibitor of platelet aggregation and modulates autonomic neurotransmission in humans [1].Formula:C20H30O5Purezza:98%Colore e forma:SolidPeso molecolare:350.45AGN 210676
CAS:AGN 210676 is a selective agonist of prostaglandin EP2(EC50 : 5 nM).Formula:C23H29NO5SPurezza:98%Colore e forma:SolidPeso molecolare:431.55EP4 receptor antagonist 1
CAS:EP4 antagonist 1: inhibits human/mouse EP4 receptors (IC50: 6.1/16.2 nM), selective over EP1-EP3 (>10 μM). For cancer immunotherapy.Formula:C23H21F3N4O3Purezza:99.53%Colore e forma:SolidPeso molecolare:458.43TCS 2510
CAS:<p>TCS 2510 (CAY10598) 是一种选择性 PGE2 和 EP4 受体激动剂，可增强细胞内 cAMP 浓度和活性 β-caten 的丰度。TCS 2510 抑制TNF-α 产生，可用于研究代谢紊乱带来的疾病。</p>Formula:C21H29N5O2Purezza:98%Colore e forma:SolidPeso molecolare:383.49(+)-Fluprostenol
CAS:(+)-Fluprostenol (AL-5848), an analogue of prostaglandin F2 alpha, is a prostaglandin F2α receptor PTGFR agonist and decreases the expression of OviductalFormula:C23H29F3O6Purezza:97.35%Colore e forma:SolidPeso molecolare:458.47Ref: TM-T21224
1mg85,00€5mg180,00€10mg298,00€25mg550,00€50mg792,00€100mg1.093,00€200mg1.454,00€1mL*10mM (DMSO)187,00€BAY 73-1449
CAS:BAY 73-1449 is a selective and potent antagonist of the prostacyclin receptor(IC50<0.1 nM).Formula:C26H23N3O3Purezza:99.77%Colore e forma:SolidPeso molecolare:425.48Ref: TM-T26745
1mg44,00€5mg90,00€10mg136,00€25mg227,00€50mg325,00€100mg434,00€200mg585,00€1mL*10mM (DMSO)94,00€DG-041
CAS:DG-041: EP3 receptor antagonist, high affinity (IC50: 4.6 & 8.1 nM), inhibits PGE2 in platelets, blood-brain barrier permeable.Formula:C23H15Cl4FN2O3S2Purezza:99.77%Colore e forma:SolidPeso molecolare:592.32Ref: TM-T15108
1mg50,00€2mg66,00€5mg97,00€10mg159,00€25mg300,00€50mg540,00€100mg777,00€500mg1.605,00€1mL*10mM (DMSO)110,00€Vidupiprant
CAS:Vidupiprant (AMG 853) is an effective dual antagonist of CRTH2 and prostanoid D receptor with IC50s of 8 nM and 35 nM in human plasma.Formula:C28H27Cl2FN2O6SPurezza:98.88%Colore e forma:SolidPeso molecolare:609.49Ref: TM-T17232
1mg66,00€5mg144,00€10mg217,00€25mg396,00€50mg590,00€100mg840,00€500mg1.691,00€1mL*10mM (DMSO)188,00€16,16-Dimethyl prostaglandin E2
CAS:16,16-Dimethyl prostaglandin E2 regulates hematopoietic stem cells via EP2/EP4 and Wnt, taken orally.Formula:C22H36O5Purezza:98%Colore e forma:SolidPeso molecolare:380.52L-657926
CAS:L-657926 is a stereoselective antagonist of the thromboxane A2 (TxA2) receptor, composed of (-)-9-chlorobenzyl-6-fluoro-1,2,3,4-tetrahydrocarbazol-1-yl acetic acid and (+)-9-chlorobenzyl-6-fluoro-1,2,3,4-tetrahydrocarbazol-1-yl acetic acid. The IC50 values for the (-) and (+) configurations against TxA2 are 0.27 nM and 124 nM, respectively.Formula:C21H19ClFNO2Colore e forma:SolidPeso molecolare:371.832EP4 receptor agonist 3
CAS:<p>EP4 receptor agonist 3 is an activator of the EP4 receptor and is useful for research in the DSS-induced colitis mouse model.</p>Formula:C21H27F2NO4Colore e forma:SolidPeso molecolare:395.44Nocloprost
CAS:Nocloprost (SH 475) is a prostaglandin E2 (PGE2) analog, an EP1 and EP3 receptor agonist with local gastric protection and ulcer healing effects.Formula:C22H37ClO4Colore e forma:SolidPeso molecolare:400.98(+)-15-epi Cloprostenol
CAS:(+)-15-epi Cloprostenol is a synthetic analogue of prostaglandin F2α (PGF2α) and functions as a potent FP receptor agonist. The compound (+)-15-epi Cloprostenol is the 15(S) or 15β-hydroxy enantiomer of (+)-(+)-15-epi Cloprostenol. Compared to the 15(R)-(+)-15-epi Cloprostenol, this epimer exhibits significantly lower activity as an FP receptor ligand. However, the specific activity of this isomer remains inadequately studied.Formula:C22H29ClO6Peso molecolare:424.92(E/Z)-Ozagrel sodium
CAS:(E/Z)-Ozagrel (sodium) [(E/Z)-OKY-046 (sodium)] is a mixture of the EZ isomers of Ozagrel (sodium). It acts as a thromboxane A2 (TXA2) synthase inhibitor. As an antiplatelet agent, Ozagrel (sodium) selectively inhibits human platelet aggregation, with an IC50 of 53.12 μM.Formula:C13H11N2NaO2Colore e forma:SolidPeso molecolare:250.228MED 27
CAS:MED 27 is an inhibitor of thromboxane synthase and thromboxane A2 receptors. It effectively inhibits rat platelet aggregation at doses significantly lower than those required for acetylsalicylic acid.Formula:C24H25N5O5Colore e forma:SolidPeso molecolare:463.49Cloprostenol
CAS:Cloprostenol is a synthetic prostaglandin and PGF2α analogue used in animals to terminate pregnancy and induce corpus luteum dissolution.Formula:C22H29ClO6Purezza:99.81%Colore e forma:Clear Colorless To Light Yellowish LiquidPeso molecolare:424.92
