
Recettore degli androgeni
Il recettore degli androgeni (AR) è un recettore ormonale nucleare che viene attivato dal legame con gli androgeni, come il testosterone e il diidrotestosterone. Questo recettore svolge un ruolo cruciale nello sviluppo e nel mantenimento delle caratteristiche maschili, nonché nella regolazione di diversi processi fisiologici, tra cui la crescita muscolare, la libido e la densità ossea. Gli inibitori del recettore degli androgeni sono ampiamente studiati nel contesto del cancro alla prostata, dove la segnalazione dell'AR è spesso sovraregolata. Presso CymitQuimica, offriamo una gamma di modulatori del recettore degli androgeni di alta qualità per supportare la tua ricerca in endocrinologia, biologia del cancro e regolazione ormonale.
Trovati 229 prodotti di "Recettore degli androgeni"
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Darolutamide
CAS:Darolutamide (BAY-1841788) is an androgen receptor (AR) antagonist that blocks AR nuclear translocation (Ki: 11 nM).Formula:C19H19ClN6O2Purezza:97.36% - >99.99%Colore e forma:SolidPeso molecolare:398.85Ref: TM-T6915
1mg50,00€2mg66,00€5mg100,00€10mg158,00€25mg250,00€50mg358,00€100mg512,00€200mg732,00€1mL*10mM (DMSO)101,00€Dimethylcurcumin
CAS:Dimethylcurcumin (ASC-J9) (ASC-J9) is an androgen receptor degradation enhancer.Formula:C23H24O6Purezza:97.36% - 98.96%Colore e forma:SolidPeso molecolare:396.43Testosterone acetate
CAS:Testosterone acetate (NSC-523836) is a hormone with in vitro antitumor activity.Formula:C21H30O3Purezza:99.6%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:330.46GSK-2881078
CAS:GSK-2881078 is a selective androgen receptor modulato (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting.Formula:C14H13F3N2O2SPurezza:98.16% - 98.81%Colore e forma:SolidPeso molecolare:330.33MI-136
CAS:MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.Formula:C23H21F3N6SPurezza:98.63% - 99.12%Colore e forma:SolidPeso molecolare:470.51Ref: TM-T6889
1mg47,00€5mg87,00€10mg147,00€25mg279,00€50mg472,00€100mg730,00€200mg1.017,00€1mL*10mM (DMSO)97,00€Nandrolone phenylpropionate
CAS:Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosisFormula:C27H34O3Purezza:99.2% - 99.46%Colore e forma:White Or Milky Crystalline PowderPeso molecolare:406.56YK11
CAS:YK11 is an androgen receptor partial agonist that activates androgen receptor transcriptional activity in HEK293 cells overexpressing androgen receptors when used at a concentration of 0.1 μM, with osteogenic activity.Formula:C25H34O6Purezza:98.91%Colore e forma:SoildPeso molecolare:430.533-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile
CAS:3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.Formula:C18H14N4OPurezza:98.41%Colore e forma:SolidPeso molecolare:302.332-hydroxy Flutamide
CAS:2-hydroxy Flutamide is competitive inhibition of androgen receptor (AR) for the treatment of prostate cancerFormula:C11H11F3N2O4Purezza:99.45% - 99.82%Colore e forma:SolidPeso molecolare:292.21Testosterone undecanoate
CAS:Testosterone undecanoate is a metabolite of Testosterone, which is a promising androgen for male hormonal contraception.Formula:C30H48O3Purezza:99.45% - 99.788%Colore e forma:White Crystalline PowderPeso molecolare:456.7Apalutamide
CAS:<p>Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.</p>Formula:C21H15F4N5O2SPurezza:99.03% - 99.91%Colore e forma:SolidPeso molecolare:477.43AH-3960
CAS:AH-3960 是一种甲状腺激素受体 1 (PTHR1) 激动剂。Formula:C13H22N4O3Purezza:98.44%Colore e forma:SolidPeso molecolare:282.34VPC-13163
CAS:VPC-13566 inhibits growth in LNCaP, Enzalutamide-resistant MR49F, lowers AR gene, PSA, TMPRSS2 expression, but not in AR-independent PC3 cells.Formula:C16H14N2Purezza:98.02%Colore e forma:SolidPeso molecolare:234.3Ref: TM-T29110
1mg85,00€2mg111,00€5mg177,00€10mg269,00€25mg429,00€50mg610,00€100mg820,00€200mg1.071,00€1mL*10mM (DMSO)165,00€S-23
CAS:S-23 ((S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide) is an oral selective androgen receptor modulator (Formula:C18H13ClF4N2O3Purezza:99.55%Colore e forma:SolidPeso molecolare:416.75Iprodione
CAS:Iprodione is a fungicide. Iprodione is also used in cannabis testing kits as a component of pesticide mixes.Formula:C13H13Cl2N3O3Purezza:98.82%Colore e forma:Colorless Crystals Cream To Colorless Odorless PowderPeso molecolare:330.17Bavdegalutamide
CAS:Bavdegalutamide (ARV-110) is a PROTAC degrader of androgen receptor (AR).Formula:C41H43ClFN9O6Purezza:97.17% - 99.04%Colore e forma:SolidPeso molecolare:812.29N-desmethyl Enzalutamide
CAS:N-desmethyl Enzalutamide (N-desmethyl MDV 3100) is the active Enzalutamide metabolite.It is the active metabolite of Enzalutamide.Formula:C20H14F4N4O2SPurezza:99.74%Colore e forma:SolidPeso molecolare:450.41Ref: TM-T19450
2mg34,00€5mg52,00€10mg74,00€25mg138,00€50mg255,00€100mg375,00€200mg532,00€1mL*10mM (DMSO)58,00€Enzalutamide carboxylic acid
CAS:<p>Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .</p>Formula:C20H13F4N3O3SPurezza:97.88%Colore e forma:SolidPeso molecolare:451.39Lupeol
CAS:Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.Formula:C30H50OPurezza:98% - 99.96%Colore e forma:Needles From Alcohol Acetone White PowderPeso molecolare:426.72VPC-13566
CAS:<p>VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the</p>Formula:C18H14N2Purezza:99.55%Colore e forma:SolidPeso molecolare:258.32
