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Recettore degli androgeni

Recettore degli androgeni

Il recettore degli androgeni (AR) è un recettore ormonale nucleare che viene attivato dal legame con gli androgeni, come il testosterone e il diidrotestosterone. Questo recettore svolge un ruolo cruciale nello sviluppo e nel mantenimento delle caratteristiche maschili, nonché nella regolazione di diversi processi fisiologici, tra cui la crescita muscolare, la libido e la densità ossea. Gli inibitori del recettore degli androgeni sono ampiamente studiati nel contesto del cancro alla prostata, dove la segnalazione dell'AR è spesso sovraregolata. Presso CymitQuimica, offriamo una gamma di modulatori del recettore degli androgeni di alta qualità per supportare la tua ricerca in endocrinologia, biologia del cancro e regolazione ormonale.

Trovati 229 prodotti di "Recettore degli androgeni"

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  • Inocoterone acetate

    CAS:
    Inocoterone acetate is a nonsteroidal antiandrogen that binds to the androgen receptor and possesses antiandrogenic activity in animal models.
    Formula:C18H26O3
    Colore e forma:Solid
    Peso molecolare:290.40
  • Linuron

    CAS:
    Linuron herbicide disrupts photosynthesis and acts as an androgen receptor antagonist.
    Formula:C9H10Cl2N2O2
    Purezza:99.08%
    Colore e forma:White Crystalline Solid Linuron Is A Colorless Crystals Non Corrosive Used As An Herbicide
    Peso molecolare:249.09
  • Enzalutamide-d3

    CAS:
    Enzalutamide D3 is a deuterium labeled Enzalutamide . Enzalutamide is an androgen receptor (AR) antagonist with an IC50 of 36 nM in LNCaP prostate cells.
    Formula:C21H16F4N4O2S
    Colore e forma:Solid
    Peso molecolare:467.45
  • Anti-Androgen receptor Antibody (8R912)


    Anti-Androgen receptor Antibody (8R912) is a Mouse antibody targeting Androgen receptor. Anti-Androgen receptor Antibody (8R912) can be used in ICC/IF.
    Colore e forma:Odour Liquid
  • Anti-Androgen receptor Antibody (7Q574)


    Anti-Androgen receptor Antibody (7Q574) is an antibody targeting Androgen receptor. Anti-Androgen receptor Antibody (7Q574) can be used in ELISA, WB, IHC.
    Colore e forma:Odour Liquid
  • MK-0773

    CAS:
    MK-0773 (PF-05314882) is a selective androgen receptor modulator that binds to AR (IC50: 6.6 nM) for the study of diseases caused by endocrine abnormalities.
    Formula:C27H34FN5O2
    Purezza:98.38% - 99.14%
    Colore e forma:Solid
    Peso molecolare:479.59
  • Anti-Androgen receptor Antibody (8H883)


    Anti-Androgen receptor Antibody (8H883) is an antibody targeting Androgen receptor. Anti-Androgen receptor Antibody (8H883) can be used in ELISA, IHC.
    Colore e forma:Odour Liquid
  • ARD-1676

    CAS:
    <p>ARD-1676 is an orally administered androgen receptor (AR) PROTAC degrader that combines an AR ligand with a cereblon ligand.</p>
    Formula:C44H46ClN7O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:788.33
  • Alternariol (Standard)

    CAS:
    Alternariol (Standard) is the standard substance of Alternariol, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Alternariol (AOH), a mycotoxin synthesized by Alternaria species, displays numerous therapeutic and biological effects, including phytotoxic, cytotoxic, anti-HIV, anti-cancer, and anti-microbial properties. It functions by inhibiting the catalytic activity of topoisomerase I and II enzymes.
    Formula:C14H10O5
    Peso molecolare:258.23
  • Estradiol valerate

    CAS:
    β-estradiol 17-valerate (EV) is a synthetic estrogen. In hormone replacement therapy drugs, it is widely used in combination with other steroid hormones.
    Formula:C23H32O3
    Purezza:99.11% - 99.9%
    Colore e forma:Na
    Peso molecolare:356.51
  • Tricaprin (Standard)

    CAS:
    Tricaprin (Standard) is the standard substance of Tricaprin, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Glycerol Tridecanoate is an orally active precursor (DA precursor) of caprylic acid that can be hydrolyzed to caprylic acid. It is a major component of medium chain triglycerides (MCT) and has antiandrogenic and antihyperglycemic properties. It can be used as an additive in food, pharmaceuticals and cosmetics.
    Formula:C33H62O6
    Colore e forma:Solid
    Peso molecolare:554.84
  • Dehydroepiandrosterone-d2

    CAS:
    Dehydroepiandrosterone-d2 is a deuterated compound of Dehydroepiandrosterone.
    Formula:C19H26D2O2
    Colore e forma:Solid
    Peso molecolare:290.44
  • Rezvilutamide

    CAS:
    Rezvilutamide (SHR3680) is an orally available androgen receptor inhibitor that crosses the blood-brain barrier and has antitumor activity.
    Formula:C22H20F3N3O4S
    Purezza:99.96% - 99.97%
    Colore e forma:Solid
    Peso molecolare:479.47
  • D4-abiraterone

    CAS:
    D4-abiraterone is the active metabolite of abiraterone.Δ4-Abiraterone is a inhibitor of CYP17A1, 3β-HSD and SRD5A, and an antagonist of the androgen receptor.
    Formula:C24H29NO
    Purezza:99.75% - 99.8%
    Colore e forma:Solid
    Peso molecolare:347.49
  • Leelamine hydrochloride

    CAS:
    Leelamine hydrochloride, a pine bark extract, inhibits androgen receptor and CB1, reducing lipid synthesis in prostate cancer.
    Formula:C20H32ClN
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:321.93
  • (Rac)-PF-998425

    CAS:
    (Rac)-PF-998425: nonsteroidal AR antagonist, potent & selective, IC50: 26 nM (binding), 90 nM (cellular), potential for androgenetic alopecia study.
    Formula:C14H14F3NO
    Colore e forma:Solid
    Peso molecolare:269.267
  • Apalutamide-13C-d3


    Apalutamide-13C-d3 is a 13C and 2H labeled Apalutamide. Apalutamide is an androgen receptor (AR) antagonist, used in research on prostate diseases.
    Formula:CC20H12F4N5O2SD3
    Colore e forma:Solid
    Peso molecolare:481.45
  • Fenarimol

    CAS:
    Fenarimol, a pyrimidine-type fungicide, exhibits potent inhibitory activity against BR biosynthesis.
    Formula:C17H12Cl2N2O
    Colore e forma:Solid
    Peso molecolare:331.2
  • Darolutamide

    CAS:
    Darolutamide (BAY-1841788) is an androgen receptor (AR) antagonist that blocks AR nuclear translocation (Ki: 11 nM).
    Formula:C19H19ClN6O2
    Purezza:97.36% - >99.99%
    Colore e forma:Solid
    Peso molecolare:398.85
  • 3-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile

    CAS:
    3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.
    Formula:C18H14N4O
    Purezza:98.41%
    Colore e forma:Solid
    Peso molecolare:302.33