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Enzima

Enzima

Gli inibitori enzimatici sono molecole che si legano agli enzimi e ne diminuiscono l'attività. Questi inibitori sono ampiamente utilizzati nella ricerca per studiare la cinetica enzimatica, la regolazione e il ruolo di specifici enzimi nelle vie metaboliche. Gli inibitori enzimatici sono anche fondamentali nello sviluppo di farmaci, poiché molti agenti terapeutici agiscono inibendo enzimi coinvolti in processi patologici. Mirando agli enzimi, questi inibitori possono modulare le vie biochimiche e offrire potenziali trattamenti per varie malattie. Presso CymitQuimica, offriamo una vasta selezione di inibitori enzimatici di alta qualità per supportare le tue ricerche in biochimica, farmacologia e scoperta di farmaci.

Sottocategorie di "Enzima"

Trovati 3619 prodotti di "Enzima"

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  • hCAIX-IN-8

    CAS:
    hCAIX-IN-8, a selective hCAIX inhibitor, IC50: 0.024 μM. Also affects CAII, CAVA (IC50s: 1.99, 1.10 μM), limits cell migration, and induces apoptosis.
    Formula:C19H16N4O6
    Colore e forma:Solid
    Peso molecolare:396.35

    Ref: TM-T61852

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • PPIE Protein, Human, Recombinant (His)


    Peptidyl-prolyl cis-trans isomerase E, also known as Cyclophilin E, Cyclophilin-33, Rotamase E, CYP33, PPIE, is an enzyme which belongs to the cyclophilin-type
    Colore e forma:Lyophilized Powder
    Peso molecolare:34 KDa (reducing condition)

    Ref: TM-TMPJ-01389

    1mg
    2.535,00€
    5µg
    113,00€
    10µg
    178,00€
    20µg
    284,00€
    50µg
    523,00€
    100µg
    759,00€
    200µg
    1.103,00€
    500µg
    1.765,00€
  • (R)-Nepicastat HCl

    CAS:
    (R)-Nepicastat HCl (RS-25560-198 HCl), R-enantiomer, inhibits bovine/human dopamine-β-hydroxylase (IC50: 25.1/18.3 nM); not affecting other enzymes/receptors.
    Formula:C14H15F2N3S·HCl
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:331.81

    Ref: TM-T6356

    5mg
    126,00€
    10mg
    207,00€
    25mg
    389,00€
    50mg
    527,00€
    100mg
    770,00€
    1mL*10mM (DMSO)
    126,00€
  • hCA I-IN-2

    CAS:
    hCA I-IN-2 (6d) inhibits hCA I (Ki: 18.8 nM) more selectively over II, IX, XII (Ki: 375.1, 1721, 283.9 nM).
    Formula:C26H20BrN5O3S
    Colore e forma:Solid
    Peso molecolare:562.44

    Ref: TM-T63972

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Telotristat besilate

    CAS:
    Telotristat besilate is an inhibitor of tryptophan hydroxylase.
    Formula:C31H28ClF3N6O6S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:705.11

    Ref: TM-T26258

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • hCAIX-IN-11

    CAS:
    hCAIX-IN-11 inhibits carbonic anhydrases IX & XII with Ki of 32.7 nM & 623.5 nM, respectively.
    Formula:C21H15ClN4O3
    Colore e forma:Solid
    Peso molecolare:406.82

    Ref: TM-T62026

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • CDK2-IN-11

    CAS:
    CDK2-IN-11 inhibits CDK2 (IC50: 6.4 μM) and targets hCA II, IX, XII (Ki: 23.4-56.3 nM); suited for cancer research.
    Formula:C18H14ClN7O2S
    Colore e forma:Solid
    Peso molecolare:427.87

    Ref: TM-T62337

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • FC11409B

    CAS:
    FC11409B is a CAIX inhibitor, inhibiting breast cancer invasion and metastasis.
    Formula:C29H23BF4N2O3S
    Colore e forma:Solid
    Peso molecolare:566.38

    Ref: TM-T70821

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • hCAIX/XII-IN-6


    hCAIX/XII-IN-6: Oral carbonic anhydrase inhibitor, targets hCA I/II/IV/IX/XII, aids rheumatoid arthritis research. Ki: 6697/2950/4093/4.1/7.7 nM.
    Formula:C26H23N3O6S4
    Colore e forma:Solid
    Peso molecolare:601.74

    Ref: TM-T72840

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • hCA IX-IN-2


    hCA IX-IN-2 is a highly potent and selective inhibitor of hCA IX, exhibiting an inhibition constant (K I) value of 32.1 nM and demonstrating anti-proliferative
    Formula:C23H24N2O4STe
    Colore e forma:Solid
    Peso molecolare:552.11

    Ref: TM-T73036

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • hCAIX-IN-5

    CAS:
    hCAIX-IN-5 was a selective hCAIX inhibitor, inhibiting hCAI, hCAII, hCAIV, and hCAIX with Ki values of >10000, >10000, 130.7, and 829.1 nM, respectively.
    Formula:C18H12FNO3
    Purezza:99.25%
    Colore e forma:Solid
    Peso molecolare:309.29

    Ref: TM-T60745

    1mg
    175,00€
    5mg
    434,00€
    10mg
    622,00€
    25mg
    973,00€
    50mg
    1.341,00€
    100mg
    1.773,00€
    500mg
    3.537,00€
  • hCAI/II-IN-1

    CAS:
    hCAI/II-IN-1 (Compound 3h) is a human carbonic anhydrase I and II (hCA I/II) inhibitor that acts on hCA I (IC50: 0.047 μM) and hCA II (IC50: 0.024 μM).
    Formula:C18H29N5O3S3
    Colore e forma:Solid
    Peso molecolare:459.65

    Ref: TM-T62892

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Phenylthiazolylthiourea

    CAS:
    Phenylthiazolylthiourea ia a dopamine-beta-hydroxylase inhibitor.
    Formula:C10H9N3S2
    Colore e forma:Solid
    Peso molecolare:235.33

    Ref: TM-T71936

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • hCAI/II-IN-3

    CAS:
    "hCAI/II-IN-3 (compound 5b) is a potent dual hCA I/II inhibitor with Ki: 51.25nM (I), 13.15nM (II), helps treat AMS."
    Formula:C16H18N4O4S2
    Colore e forma:Solid
    Peso molecolare:394.47

    Ref: TM-T61832

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • hCAXII-IN-3

    CAS:
    hCAXII-IN-3 (Compound 6o) is a selective inhibitor of human carbonic anhydrase XII (hCAXII) (Ki: 10.0 nM).
    Formula:C26H20BrN5O3S
    Colore e forma:Solid
    Peso molecolare:562.44

    Ref: TM-T63973

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • hCAI/II-IN-4

    CAS:
    hCAI/II-IN-4 inhibits hCA I & II (Ki: 16.95 & 15.22 nM), hCA IX (Ki: 27.04 nM), has anti-hypoxia benefits and is low-toxic for AMS research.
    Formula:C15H15N3O5S2
    Colore e forma:Solid
    Peso molecolare:381.43

    Ref: TM-T61635

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • hCAXII-IN-5

    CAS:
    hCAXII-IN-5, or compound 6o, is a potent, selective hCAXII inhibitor with Ki values: hCAI & II >10000, hCAIX 286.1, hCAXII 1.0 nM.
    Formula:C23H22N2O4
    Colore e forma:Solid
    Peso molecolare:390.43

    Ref: TM-T61769

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • JM6

    CAS:
    JM6 is a weak kynurenine 3-monooxygenase (KMO) inhibitor that acts on mouse KMO (IC50: 19.85 μM). JM6 can be used to study Alzheimer's disease.
    Formula:C23H26N4O6S2
    Colore e forma:Solid
    Peso molecolare:518.61

    Ref: TM-T63613

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Tyrosinase-IN-7

    CAS:
    Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.
    Formula:C15H10O5
    Purezza:99%
    Colore e forma:Solid
    Peso molecolare:270.24

    Ref: TM-T72786

    1mg
    60,00€
    5mg
    130,00€
    10mg
    200,00€
    25mg
    401,00€
    50mg
    645,00€
    100mg
    1.018,00€
    200mg
    1.378,00€
  • hCAIX-IN-10

    CAS:
    "hCAIX-IN-10 (6i) selectively inhibits carbonic anhydrase IX/XII (Ki: 61.5/586.8 nM), markers in tumor cells, affecting acid-base balance."
    Formula:C28H21N3O3S
    Colore e forma:Solid
    Peso molecolare:479.55

    Ref: TM-T63158

    25mg
    1.927,00€
    50mg
    2.507,00€
    100mg
    3.168,00€