
Enzima
Gli inibitori enzimatici sono molecole che si legano agli enzimi e ne diminuiscono l'attività. Questi inibitori sono ampiamente utilizzati nella ricerca per studiare la cinetica enzimatica, la regolazione e il ruolo di specifici enzimi nelle vie metaboliche. Gli inibitori enzimatici sono anche fondamentali nello sviluppo di farmaci, poiché molti agenti terapeutici agiscono inibendo enzimi coinvolti in processi patologici. Mirando agli enzimi, questi inibitori possono modulare le vie biochimiche e offrire potenziali trattamenti per varie malattie. Presso CymitQuimica, offriamo una vasta selezione di inibitori enzimatici di alta qualità per supportare le tue ricerche in biochimica, farmacologia e scoperta di farmaci.
Sottocategorie di "Enzima"
- Anidrasi carbonica(197 prodotti)
- Idrossilasi(35 prodotti)
- MPO(2 prodotti)
- Riduttasi(50 prodotti)
- Tirosinasi(71 prodotti)
Trovati 3618 prodotti di "Enzima"
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hCAXII-IN-2
CAS:hCAXII-IN-2 is a potent inhibitor of hCA XII (Ki: 84.2 nM) and hCA IX (Ki: 268.5 nM), with low activity on hCA I/II.Formula:C21H18ClN3O4Colore e forma:SolidPeso molecolare:411.84LP-533401
CAS:LP-533401 is an inhibitor of Tryptophan hydroxylase 1. It is used for regulates serotonin production in the gut.Formula:C27H22F4N4O3Purezza:98%Colore e forma:SolidPeso molecolare:526.48hCAII-IN-1
CAS:hCAII-IN-1 (7f) inhibits CA II/IX with Kis 1.2 nM/113.6 nM, potential for cancer treatment.Formula:C21H21BrN6O4SColore e forma:SolidPeso molecolare:533.4hCAIX-IN-6
CAS:6B and 14g inhibit tumor-associated HCA IX with low nanomolar potency; 6K targets HCA XII. All are potential cancer drug leads.Formula:C18H12N2O4SColore e forma:SolidPeso molecolare:352.36Fenprinast
CAS:Fenprinast is a tryptophan-like bronchodilator utilized in the study of allergic and exercise-induced asthma. It exhibits oral activity.Formula:C16H16ClN5OPeso molecolare:329.78hCAI/II-IN-1
CAS:hCAI/II-IN-1 (Compound 3h) is a human carbonic anhydrase I and II (hCA I/II) inhibitor that acts on hCA I (IC50: 0.047 μM) and hCA II (IC50: 0.024 μM).Formula:C18H29N5O3S3Colore e forma:SolidPeso molecolare:459.65AHR-15010
CAS:AHR-15010 is a novel anti-arthritic agent.Formula:C10H16N2O8S2Purezza:98%Colore e forma:SolidPeso molecolare:356.373-Allylphenol
CAS:3-Allylphenol is an inhibitor of dopamine β-hydroxylase (DBH; Ki = 12 mM).Formula:C9H10OColore e forma:SolidPeso molecolare:134.18hCAI/II-IN-3
CAS:"hCAI/II-IN-3 (compound 5b) is a potent dual hCA I/II inhibitor with Ki: 51.25nM (I), 13.15nM (II), helps treat AMS."Formula:C16H18N4O4S2Colore e forma:SolidPeso molecolare:394.47hCAIX-IN-10
CAS:"hCAIX-IN-10 (6i) selectively inhibits carbonic anhydrase IX/XII (Ki: 61.5/586.8 nM), markers in tumor cells, affecting acid-base balance."Formula:C28H21N3O3SColore e forma:SolidPeso molecolare:479.55Quinethazone
CAS:Quinethazone is a thiazide diuretic used to treat hypertension. Common side effects include dizziness, dry mouth, nausea, and low potassium levels.Formula:C10H12ClN3O3SColore e forma:Fibrous Crystals From 50% Acetone Physical Description Fibrous Crystals Or White Powder (Ntp 1992)Peso molecolare:289.74JM6
CAS:JM6 is a weak kynurenine 3-monooxygenase (KMO) inhibitor that acts on mouse KMO (IC50: 19.85 μM). JM6 can be used to study Alzheimer's disease.Formula:C23H26N4O6S2Colore e forma:SolidPeso molecolare:518.61hCAIX-IN-5
CAS:hCAIX-IN-5 was a selective hCAIX inhibitor, inhibiting hCAI, hCAII, hCAIV, and hCAIX with Ki values of >10000, >10000, 130.7, and 829.1 nM, respectively.Formula:C18H12FNO3Purezza:99.25%Colore e forma:SolidPeso molecolare:309.29Disulfamide
CAS:Disulfamide: Oral carbonic anhydrase inhibitor, IC50 0.07 μM, diuretic by blocking Na+/HCO3- reabsorption.Formula:C7H9ClN2O4S2Purezza:98.65%Colore e forma:SolidPeso molecolare:284.74hCAIX-IN-11
CAS:hCAIX-IN-11 inhibits carbonic anhydrases IX & XII with Ki of 32.7 nM & 623.5 nM, respectively.Formula:C21H15ClN4O3Colore e forma:SolidPeso molecolare:406.82PGDS Protein, Human, Recombinant
Hematopoietic Prostaglandin D Synthase (HPGDS) belongs to the GST superfamily and Sigma family.Colore e forma:Lyophilized PowderPeso molecolare:26 KDa (reducing condition)Ref: TM-TMPJ-00690
1mg2.911,00€5µg119,00€10µg188,00€20µg301,00€50µg551,00€100µg823,00€200µg1.205,00€500µg2.029,00€(R)-Nepicastat HCl
CAS:(R)-Nepicastat HCl (RS-25560-198 HCl), R-enantiomer, inhibits bovine/human dopamine-β-hydroxylase (IC50: 25.1/18.3 nM); not affecting other enzymes/receptors.Formula:C14H15F2N3S·HClPurezza:98%Colore e forma:SolidPeso molecolare:331.81CK1 δ/CSNK1D Protein, Human, Recombinant (Baculovirus, His)
<p>Expression system: Baculovirus<br>Length: 1-415, Full Length<br>Activity: Not Tested</p>Purezza:85%Colore e forma:Odour Lyophilized PowderRef: TM-TMPH-03771
1mg9.292,00€5µg999,00€10µg1.686,00€20µg2.863,00€50µg3.715,00€100µg4.577,00€200µg5.655,00€500µg7.509,00€hCAXII-IN-5
CAS:hCAXII-IN-5, or compound 6o, is a potent, selective hCAXII inhibitor with Ki values: hCAI & II >10000, hCAIX 286.1, hCAXII 1.0 nM.Formula:C23H22N2O4Colore e forma:SolidPeso molecolare:390.43L-693612 HCl
CAS:L-693612 HCl is an inhibitor of carbonic anhydrase.Formula:C14H25ClN2O5S3Purezza:98%Colore e forma:SolidPeso molecolare:433.01

