
Enzima
Gli inibitori enzimatici sono molecole che si legano agli enzimi e ne diminuiscono l'attività. Questi inibitori sono ampiamente utilizzati nella ricerca per studiare la cinetica enzimatica, la regolazione e il ruolo di specifici enzimi nelle vie metaboliche. Gli inibitori enzimatici sono anche fondamentali nello sviluppo di farmaci, poiché molti agenti terapeutici agiscono inibendo enzimi coinvolti in processi patologici. Mirando agli enzimi, questi inibitori possono modulare le vie biochimiche e offrire potenziali trattamenti per varie malattie. Presso CymitQuimica, offriamo una vasta selezione di inibitori enzimatici di alta qualità per supportare le tue ricerche in biochimica, farmacologia e scoperta di farmaci.
Sottocategorie di "Enzima"
- Anidrasi carbonica(192 prodotti)
- Idrossilasi(35 prodotti)
- MPO(2 prodotti)
- Riduttasi(50 prodotti)
- Tirosinasi(72 prodotti)
Trovati 3614 prodotti di "Enzima"
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Tyrosinase-IN-7
CAS:Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.Formula:C15H10O5Purezza:99%Colore e forma:SolidPeso molecolare:270.24hCAI/II-IN-2
CAS:hCAI/II-IN-2 (2b) inhibits hCA I/II (Ki: 40.97 nM, 15.15 nM) and IX (61.88 nM), fights AMS with anti-hypoxic effects, but has low cellular activity.Formula:C12H12N4O5S2Colore e forma:SolidPeso molecolare:356.38hCAXII-IN-4
CAS:hCAXII-IN-4 is a selective and potent CA XII inhibitor with a Ki value of 6.4 nM for human CA XII.Formula:C22H27N5O6SColore e forma:SolidPeso molecolare:489.54PPIE Protein, Human, Recombinant (His)
Peptidyl-prolyl cis-trans isomerase E, also known as Cyclophilin E, Cyclophilin-33, Rotamase E, CYP33, PPIE, is an enzyme which belongs to the cyclophilin-typeColore e forma:Lyophilized PowderPeso molecolare:34 KDa (reducing condition)DTP348
CAS:DTP348: Oral carbonic anhydrase IX inhibitor & hypoxic cell radiosensitizer with sulfamide & 5-nitroimidazole components.Formula:C6H11N5O4SColore e forma:SolidPeso molecolare:249.25hCAXII-IN-2
CAS:hCAXII-IN-2 is a potent inhibitor of hCA XII (Ki: 84.2 nM) and hCA IX (Ki: 268.5 nM), with low activity on hCA I/II.Formula:C21H18ClN3O4Colore e forma:SolidPeso molecolare:411.84CK1 δ/CSNK1D Protein, Human, Recombinant (Baculovirus, His)
<p>Expression system: Baculovirus<br>Length: 1-415, Full Length<br>Activity: Not Tested</p>Purezza:85%Colore e forma:Odour Lyophilized PowderhCAII-IN-1
CAS:hCAII-IN-1 (7f) inhibits CA II/IX with Kis 1.2 nM/113.6 nM, potential for cancer treatment.Formula:C21H21BrN6O4SColore e forma:SolidPeso molecolare:533.4hCAIX-IN-6
CAS:6B and 14g inhibit tumor-associated HCA IX with low nanomolar potency; 6K targets HCA XII. All are potential cancer drug leads.Formula:C18H12N2O4SColore e forma:SolidPeso molecolare:352.36hCAI/II-IN-3
CAS:"hCAI/II-IN-3 (compound 5b) is a potent dual hCA I/II inhibitor with Ki: 51.25nM (I), 13.15nM (II), helps treat AMS."Formula:C16H18N4O4S2Colore e forma:SolidPeso molecolare:394.47hCAIX-IN-10
CAS:"hCAIX-IN-10 (6i) selectively inhibits carbonic anhydrase IX/XII (Ki: 61.5/586.8 nM), markers in tumor cells, affecting acid-base balance."Formula:C28H21N3O3SColore e forma:SolidPeso molecolare:479.55Quinethazone
CAS:Quinethazone is a thiazide diuretic used to treat hypertension. Common side effects include dizziness, dry mouth, nausea, and low potassium levels.Formula:C10H12ClN3O3SColore e forma:Fibrous Crystals From 50% Acetone Physical Description Fibrous Crystals Or White Powder (Ntp 1992)Peso molecolare:289.74SU 10603
CAS:SU 10603 is a specific inhibitor of 17α-hydroxylase (also known as CYP17A1 and P450c17) used to study steroid hormone synthesis.Formula:C15H12ClNOPurezza:99.93% - 99.96%Colore e forma:SolidPeso molecolare:257.72L 645151
CAS:L 645151 is an inhibitor of lipophilic CA.Formula:C12H14N2O4S2Colore e forma:SolidPeso molecolare:314.38LP-533401
CAS:LP-533401 is an inhibitor of Tryptophan hydroxylase 1. It is used for regulates serotonin production in the gut.Formula:C27H22F4N4O3Purezza:98%Colore e forma:SolidPeso molecolare:526.48(R)-Nepicastat HCl
CAS:<p>(R)-Nepicastat HCl (RS-25560-198 HCl), R-enantiomer, inhibits bovine/human dopamine-β-hydroxylase (IC50: 25.1/18.3 nM); not affecting other enzymes/receptors.</p>Formula:C14H15F2N3S·HClPurezza:98%Colore e forma:SolidPeso molecolare:331.81GV2-20
CAS:GV2-20 is an effective carbonic anhydrase 2 inhibitors.Formula:C15H13N3O6Purezza:98%Colore e forma:SolidPeso molecolare:331.28L-693612
CAS:L-693612 is an inhibitor of carbonic anhydrase.Formula:C14H24N2O5S3Purezza:98%Colore e forma:SolidPeso molecolare:396.55hCAXII-IN-5
CAS:hCAXII-IN-5, or compound 6o, is a potent, selective hCAXII inhibitor with Ki values: hCAI & II >10000, hCAIX 286.1, hCAXII 1.0 nM.Formula:C23H22N2O4Colore e forma:SolidPeso molecolare:390.43Carbonic anhydrase inhibitor 14
CAS:CA inhibitor 14 blocks hCA I/II/IX/XII (K i of 1203/99.7/9.4/27.7 nM) and CDK2 (IC50: 20.3 μM), showing antitumor effects.Formula:C18H17N7O2SColore e forma:SolidPeso molecolare:395.44
