Enzima
Gli inibitori enzimatici sono molecole che si legano agli enzimi e ne diminuiscono l'attività. Questi inibitori sono ampiamente utilizzati nella ricerca per studiare la cinetica enzimatica, la regolazione e il ruolo di specifici enzimi nelle vie metaboliche. Gli inibitori enzimatici sono anche fondamentali nello sviluppo di farmaci, poiché molti agenti terapeutici agiscono inibendo enzimi coinvolti in processi patologici. Mirando agli enzimi, questi inibitori possono modulare le vie biochimiche e offrire potenziali trattamenti per varie malattie. Presso CymitQuimica, offriamo una vasta selezione di inibitori enzimatici di alta qualità per supportare le tue ricerche in biochimica, farmacologia e scoperta di farmaci.
Sottocategorie di "Enzima"
- Anidrasi carbonica(189 prodotti)
- Idrossilasi(35 prodotti)
- MPO(2 prodotti)
- Riduttasi(50 prodotti)
- Tirosinasi(72 prodotti)
Trovati 3610 prodotti di "Enzima"
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Phenylsulfamide
CAS:<p>Phenylsulfamide (Compound 10), acting as an inhibitor of human carbonic anhydrase-II (hCA-II), exhibits a dissociation constant (Kd) of 45.50 μM and an</p>Formula:C6H8N2O2SColore e forma:SolidPeso molecolare:172.2Tyrosinase-IN-38
Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.Colore e forma:Odour SolidCarbonic anhydrase inhibitor 31
Carbonic anhydrase inhibitor31 is an mtCA2 inhibitor (Ki: 5.2 nM) that can be used in antituberculosis research.Formula:C24H20N6O5SColore e forma:SolidPeso molecolare:504.12159VM4-037
CAS:VM4-037 is a PET imaging agent used for carbonic anhydrase IX.Formula:C26H29FN6O7S2Colore e forma:SolidPeso molecolare:620.675,6-Dihydro-2H-pyran-2-one
CAS:5,6-Dihydro-2H-pyran-2-one is a carbonic anhydrase 1/9 inhibitor that inhibits KB cell viability.Formula:C5H6O2Colore e forma:SolidPeso molecolare:98.1TPH1-IN-1
TPH1-IN-1 (compound 40) is a xanthine derivative that serves as an inhibitor of tryptophan hydroxylase TPH1, with an IC50 of 110.1 nM.Formula:C21H18N6O4SColore e forma:SolidPeso molecolare:450.47hCAIX-IN-17
hCA IX-IN-1 inhibits hCA I/II/IX/XII with Ki of 331.4/28.4/9.4/17.8 nM, has anticancer properties.Formula:C19H18N2O3SColore e forma:SolidPeso molecolare:354.42Peroxidase, from horseradish, approx. 200 U/mg
CAS:Purezza:≥ 150U/mgColore e forma:Beige to light-brown, reddish brown or dark brown lyophilised powderPeso molecolare:-DOTA-XYIMSR-01
CAS:DOTA-XYIMSR-01 is a molecular probe targeting CAIX, capable of being labeled with 177Lu for the treatment and localization of malignant gliomas. The uptake of [177Lu]Lu-XYIMSR-01 in U87MG tumors is 6.19% injected dose per gram (% ID/g), with a tumor-to-muscle uptake ratio of 20.14. In an orthotopic glioma model, co-administration with temozolomide significantly enhances survival rates and inhibits tumor growth in mice. DOTA-XYIMSR-01 shows potential for research in the field of cancer treatment.Formula:C61H88N16O22S2Colore e forma:SolidPeso molecolare:1461.57hCAIX-IN-19
<p>hCAIX-IN-19 is a sulfonamide inhibitor with an inhibition constant (KI) of 6.2 nM for hCAIX, exhibiting significant selectivity towards hCAIX over hCAI (hCA I/</p>Colore e forma:Odour SolidCAIX/CAXII-IN-4
<p>CAIX/CAXII-IN-4 (Compound 7h) is an inhibitor of carbonic anhydrase (CA) that binds to CAIX, CA XII, and CAII with Ki values of 1.324 μM, 0.435 μM, and 3.035 μM, respectively. This compound exhibits broad-spectrum anti-tumor activity and inhibits the proliferation of central nervous system tumor cells U251, with a GI50 of 0.361 μM.</p>Formula:C23H21N5O3SColore e forma:SolidPeso molecolare:447.51Tyrosinase-IN-32
<p>Tyrosinase-IN-32 (compound 11), a hydroxamate-based alkaloid extracted from black pepper (Piper nigrum L.), functions as an inhibitor of mushroom tyrosinase. In addition to its inhibitory properties, it exhibits antioxidant activity.</p>Formula:C15H19NO3Colore e forma:SolidPeso molecolare:261.32Dorzolamide
CAS:<p>Dorzolamide is an anti-glaucoma agent and is a carbonic anhydrase inhibitor.</p>Formula:C10H16N2O4S3Purezza:98%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:324.44
