
cAMP
cAMP è un secondo messaggero importante in molti processi biologici, inclusa la regolazione del metabolismo, l'espressione genica e la crescita cellulare. Nella via di segnalazione MAPK, cAMP può modulare l'attività di diverse chinasi, inclusa la PKA, che a sua volta influenza la cascata MAPK. La disregolazione della segnalazione di cAMP è implicata in varie malattie, tra cui il cancro e i disturbi cardiovascolari. Presso CymitQuimica, offriamo una varietà di modulatori di cAMP per supportare la tua ricerca sulla trasduzione del segnale, il metabolismo e la patologia delle malattie.
Trovati 46 prodotti di "cAMP"
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JNJ-39758979
CAS:JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).Formula:C11H19N5Purezza:98.33% - 99.62%Colore e forma:SolidPeso molecolare:221.3Ref: TM-T11723L
1mg46,00€5mg92,00€10mg147,00€25mg241,00€50mg350,00€100mg515,00€200mg700,00€1mL*10mM (DMSO)100,00€HJC0197
CAS:HJC0197 is a selective Epac antagonist; blocks cAMP-induced activation with IC50=5.9 μM for Epac2.Formula:C19H21N3OSPurezza:98.05%Colore e forma:SolidPeso molecolare:339.45Ref: TM-T15485
2mg38,00€5mg54,00€10mg86,00€25mg135,00€50mg188,00€100mg283,00€200mg426,00€1mL*10mM (DMSO)64,00€Bithionol
CAS:Bithionol (Actamer), formerly marketed as an active ingredient in various topical drug products, was shown to be a potent photosensitizer with the potential toFormula:C12H6Cl4O2SPurezza:99.04%Colore e forma:White Or Grayish-White Crystalline Powder Phenolic Odor (Ntp 1992)Peso molecolare:356.05CE3F4
CAS:CE3F4 is a selective antagonist of exchange protein directly activated by cAMP (Epac1; IC50s of 10.7 μM and 66 μM for Epac1 and Epac2(B), respectively).Formula:C11H10Br2FNOPurezza:97.15% - 98.06%Colore e forma:SolidPeso molecolare:351.01Mirabegron
CAS:Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.Formula:C21H24N4O2SPurezza:99.64%Colore e forma:Light Yellow To Yellow SolidPeso molecolare:396.51Bucladesine sodium
CAS:Bucladesine sodium (DC2797) is a cAMP analog with cell-permeable properties.Formula:C18H23N5NaO8PPurezza:96.56% - 99.76%Colore e forma:White PowderPeso molecolare:491.37A-3 hydrochloride
CAS:A-3 hydrochloride: potent, reversible kinase antagonist; permeable; inhibits PKC, CKI, PKA, CKII, MLCK; Ki: 4.3-80 μM.
Formula:C12H14Cl2N2O2SPurezza:99.32%Colore e forma:SolidPeso molecolare:321.22MR-L2
CAS:MR-L2 is a reversible and noncompetitive allosteric activator of long-isoform phosphodiesterase-4 (PDE4).Formula:C19H16Cl3FN4OPurezza:98.09% - 98.94%Colore e forma:SolidPeso molecolare:441.71Ref: TM-T12103
1mg138,00€2mg197,00€5mg334,00€10mg500,00€25mg807,00€50mg1.099,00€100mg1.485,00€500mg2.962,00€1mL*10mM (DMSO)358,00€ESI-05
CAS:ESI-05 (NSC-116966) is a specific 0.4 μM IC50 EPAC2 antagonist that blocks cAMP-induced EPAC2 and Rap1 activation.Formula:C16H18O2SPurezza:97.22%Colore e forma:SolidPeso molecolare:274.38OX04528
CAS:OX04528 is an orally active and potent GPR84 biased agonist.OX04528 inhibits cAMP signaling and may be useful in cancer research.Formula:C16H13F6NO2Purezza:99.74%Colore e forma:SoildPeso molecolare:365.27MRS-1706
CAS:MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.Formula:C27H29N5O5Purezza:99.00%Colore e forma:SolidPeso molecolare:503.55Ref: TM-T16136
1mg37,00€5mg79,00€10mg119,00€25mg235,00€50mg376,00€100mg603,00€200mg848,00€1mL*10mM (DMSO)88,00€BC 11-38
CAS:BC 11-38 is a potent, selective PDE biodepressant which is mainly effective against PDE11 (IC50 : 0.28 μM).Formula:C15H16N2OS2Purezza:98.95% - 99.28%Colore e forma:SolidPeso molecolare:304.43Ref: TM-T21865
1mg34,00€5mg66,00€10mg92,00€25mg192,00€50mg313,00€100mg500,00€200mg708,00€1mL*10mM (DMSO)77,00€Adenosine 3'-monophosphate (sodium salt hydrate)
Adenosine 3'-monophosphate (sodium salt hydrate) (3'-AMP) is a nucleotide and cAMP-generating agonist that elevates cAMP levels in NG108-15 cells.Formula:C10H15N5NaO8PColore e forma:SolidPeso molecolare:387.222-PCCA hydrochloride
CAS:2-PCCA hydrochloride, a racemate, is a potent and selective GPR88 receptor agonist showing inhibition of GPR88-mediated cAMP production in HEK293 cells with anFormula:C30H39Cl2N3OPurezza:97.54% - 99.07%Colore e forma:SoildPeso molecolare:528.56Ref: TM-T80666
1mg86,00€5mg183,00€10mg259,00€25mg416,00€50mg550,00€100mg752,00€200mg1.008,00€1mL*10mM (DMSO)215,00€GLP-1R modulator L7-028
CAS:GLP-1R modulator L7-028 is a variant modulator that enhances affinity for GLP-1 and cAMP signaling.Formula:C24H28N2O3Purezza:98.76% - >99.99%Colore e forma:SolidPeso molecolare:392.49Anti-Cathelicidin/Camp Polyclonal Antibody
Antibody Type: Rabbit Polyclonal
Application: ELISA,ICC/IF,IF,IHC-Fr,IHC-P
Reactivity: (predicted:Mouse,Rat)Colore e forma:LiquidPeso molecolare:Theoretical: 19 kDa.Glaucine
CAS:Glaucine: antitussive, antioxidative, antiviral, may fight arthritis, boosts IL-10, hinders breast cancer cell spread by inhibiting MMP-9 and NF-κB.
Formula:C21H25NO4Purezza:99.42% - 99.56%Colore e forma:SolidPeso molecolare:355.43Pinoresinol 4-O-β-D-glucopyranoside
CAS:(+)-Pinoresinol-β-D-glucoside, also known as (+)-pinor, is a major active lignan furanoid found in Forsythia.Formula:C26H32O11Purezza:99.32% - >99.99%Colore e forma:SolidPeso molecolare:520.53Ref: TM-T4S0792
1mg50,00€5mg96,00€10mg161,00€25mg264,00€50mg370,00€100mg522,00€200mg707,00€1mL*10mM (DMSO)127,00€Ro 20-1724
CAS:Ro 20-1724 (4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone) is a widely used inhibitor of cyclic nucleotide phosphodiesterase with IC50 of 2.0 μM and Ki of 3.1Formula:C15H22N2O3Purezza:98.82% - 99.79%Colore e forma:SolidPeso molecolare:278.35SAX-187
CAS:SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.Formula:C15H13ClN4O2S2Purezza:97.82% - 98%Colore e forma:SolidPeso molecolare:380.87Ref: TM-T3183
1mg79,00€5mg152,00€10mg245,00€25mg398,00€50mg532,00€100mg735,00€200mg973,00€1mL*10mM (DMSO)166,00€

