
MAPK
Le MAPK sono una famiglia di chinasi proteiche coinvolte in una varietà di processi cellulari, tra cui crescita, proliferazione, differenziazione e risposte allo stress. La via di segnalazione MAPK è composta da diversi livelli, tra cui ERK, JNK e p38 MAPK, ciascuno con ruoli distinti nella funzione cellulare. La disregolazione della segnalazione MAPK è collegata al cancro, alle malattie infiammatorie e ai disturbi metabolici. Presso CymitQuimica, offriamo una vasta gamma di inibitori e attivatori delle MAPK per supportare la tua ricerca in biologia cellulare, trasduzione del segnale e meccanismi delle malattie.
Trovati 894 prodotti di "MAPK"
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SW-034538
CAS:SW-034538 is a TAO2 inhibitor (IC 50= 300 nM).Formula:C18H20N4O3S2Colore e forma:SolidPeso molecolare:404.51SB-747651A
CAS:SB-747651A: ATP-competitive MSK1 inhibitor (IC50=11nM), affects N-terminal domain, also hinders MSK2, PKA, PKB, RSK, p70S6K.Formula:C16H22N8OPurezza:98%Colore e forma:SolidPeso molecolare:342.4SB 204900
CAS:SB 204900 inhibit the release of histamine and TNF-α from RBL-2H3 cells.Formula:C18H17NO2Colore e forma:SolidPeso molecolare:279.33HPK1-IN-29
CAS:"HPK1-IN-29 suppresses HPK1, boosting anti-tumor immunity; potential for immune disease research."Formula:C26H18F3N5O2Colore e forma:SolidPeso molecolare:489.45EO 1428
CAS:p38α and p38β2 inhibitorFormula:C20H16BrClN2OPurezza:98%Colore e forma:SolidPeso molecolare:415.71DDO3711
CAS:"DDO3711, a PHORC, links an ASK1 inhibitor to a PP5 activator, inhibiting ASK1 (IC50=164.1 nM), dephosphorylating p-ASK1, and showing anti-cancer potential."Formula:C42H41N9O6Colore e forma:SolidPeso molecolare:767.83PD 334581
CAS:MEK1 inhibitorFormula:C20H19F3IN5O2Purezza:98%Colore e forma:SolidPeso molecolare:545.3p38α inhibitor 2
CAS:P38α Inhibitor 2, a potent and selective inhibitor of p38α MAPK, exhibits a pIC50 value of 9.6.Formula:C27H33N5O3Colore e forma:SolidPeso molecolare:475.58pan-KRAS-IN-16
CAS:3344 is an inhibitor of KRAS-effector interactions,with an affnity of 126nm.Formula:C24H26N2O3Purezza:98%Colore e forma:SolidPeso molecolare:390.47B-Raf IN 6
CAS:B-Raf IN 6: potent B-Raf kinase inhibitor, IC50 of 1.7 nM, doesn't target PXR, metabolically stable, potential in cancer research.Formula:C24H21F3N6O2S2Colore e forma:SolidPeso molecolare:546.59(R)-CE3F4
CAS:(R)-CE3F4 is a selective inhibitor of exchange protein directly activated by cAMP isoform 1 (Epac1)(IC50 of 4.2 μM),Formula:C11H10Br2FNOColore e forma:SolidPeso molecolare:351.01SR-3737
CAS:SR-3737 is potent both JNK3 and p38 inhibitor.Formula:C29H25FN4O4Purezza:98%Colore e forma:SolidPeso molecolare:512.53KRAS G12C inhibitor 29
CAS:KRAS G12C inhibitor 29 is an inhibitor of KRAS G12C and can be used to study cancer.Formula:C23H21ClFN5O2Colore e forma:SolidPeso molecolare:453.9BMS-214662 hydrochloride
CAS:BMS-214662: a farnesyltransferase inhibitor, nonsedating benzodiazepine, blocks Ras-related tumorigenesis.Formula:C25H24ClN5O2S2Colore e forma:SolidPeso molecolare:526.07K-Ras G12C-IN-3
CAS:K-Ras G12C-IN-3: novel, irreversible inhibitor of K-Ras G12C mutant protein for cancer treatment.Formula:C21H19Cl3N2O3Colore e forma:SolidPeso molecolare:453.758-CPT-2Me-cAMP, sodium salt
CAS:8-CPT-2Me-cAMP sodium activates Epac GEFS, targets Rap1/2, has 2.2 μM EC50 for Epac1, doesn't activate PKA, and prompts Ca2+ release in β-cells.Formula:C17H16ClN5NaO6PSColore e forma:SolidPeso molecolare:507.82SCH-53870
CAS:SCH-53870 inhibits p21-hRas nucleotide exchange in vitro.Formula:C18H18N2O4SColore e forma:SolidPeso molecolare:358.41KRAS inhibitor-16
CAS:KRAS inhibitor-16 blocks KRAS G12C and p-ERK in cancer cells; potential for pancreatic, colorectal, lung cancer treatment. IC50: 0.457 μM.Formula:C20H16Cl2FN3O2SColore e forma:SolidPeso molecolare:452.33SOS1-IN-12
CAS:SOS1-IN-12 is a potent inhibitor of SOS1, acting on SOS1 (Ki: 0.11 nM) and on pERK (IC50: 47 nM).Formula:C23H26F3N5Colore e forma:SolidPeso molecolare:429.48J30-8
CAS:J30-8 is a JNK3 inhibitor (IC50: 40 nM) with neuroprotective activity and can be used to study neurodegenerative diseases such as Alzheimer's disease.Formula:C17H9ClFN3O2SPurezza:99.90%Colore e forma:SolidPeso molecolare:373.79
