Canale TRP/TRPV
canali TRP (Transient Receptor Potential), inclusa la sottofamiglia TRPV, sono un gruppo di canali ionici coinvolti in vari processi sensoriali, come la percezione della temperatura, la sensazione del dolore e l'osmoregolazione. I canali TRP sono ampiamente espressi in diversi tessuti e svolgono un ruolo nelle risposte fisiologiche agli stimoli ambientali. In particolare, i canali TRPV sono coinvolti nel rilevamento dei cambiamenti di temperatura e sono implicati in condizioni come il dolore cronico, l'infiammazione e il cancro. Presso CymitQuimica, offriamo una gamma completa di modulatori dei canali TRP/TRPV per supportare la tua ricerca in biologia sensoriale, gestione del dolore e trasduzione del segnale.
Trovati 93 prodotti di "Canale TRP/TRPV"
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(Z)-Capsaicin
CAS:<p>(Z)-Capsaicin (Zucapsaicin) is a medication used to treat osteoarthritis of the knee and Others neuropathic pain.(Z)-Capsaicin is a synthetic cis isomer of</p>Formula:C18H27NO3Purezza:97.33% - 98.91%Colore e forma:SolidPeso molecolare:305.41Vocacapsaicin hydrochloride
CAS:<p>Vocacapsaicin hydrochloride (CA-008 hydrochloride) is a non-opioid TRPV1 agonist, a raw material for capsaicin, and is used for pain relief.</p>Formula:C26H42ClN3O4Purezza:99.66% - 99.80%Colore e forma:SolidPeso molecolare:496.08TRPV4 agonist-1 free base
CAS:<p>TRPV4 agonist-1 free base (OUN67600) is an agonist of transient receptor potential vanilloid 4 (TRPV4;EC50 of 60 nM, in the hTRPV4 Ca2+ assay).</p>Formula:C25H22F2N4O2Purezza:99.79%Colore e forma:SolidPeso molecolare:448.46BI-749327
CAS:<p>BI-749327 is a high selectivity and orally bioavailable antagonist of TRPC6 (IC50s: 13 nM, 19 nM and 15 nM for mouse, human and guinea pig TRPC6).</p>Formula:C23H21F3N4O2Purezza:99.68%Colore e forma:SolidPeso molecolare:442.43IA-Alkyne
CAS:<p>IA-Alkyne: TRPC agonist, cysteine-reactivity probe, potential in respiratory infection study.</p>Formula:C8H12INOPurezza:99.76%Colore e forma:SolidPeso molecolare:265.09GFB-8438
CAS:<p>GFB-8438 is a potent and subtype selective inhibitor of TRPC5(IC50s of 0.18 and 0.29 μM of hTRPC5 and hTRPC4, respectively).</p>Formula:C16H14ClF3N4O2Purezza:99.58%Colore e forma:SolidPeso molecolare:386.76PF-04745637
CAS:<p>PF-04745637 is a potent and selective TRPA1 antagonist with an IC50 of 17 nM[1].</p>Formula:C27H32ClF3N2O2Purezza:98.88% - 99.3%Colore e forma:SolidPeso molecolare:509Oleoyl Serotonin
CAS:<p>Oleoyl Serotonin is an antagonist of hTRPV1 with an IC50 of 2.57 μM.</p>Formula:C28H44N2O2Purezza:99.88%Colore e forma:SolidPeso molecolare:440.66L-R4W2
CAS:<p>Vanilloid TRPV1 (VR1) receptor antagonist peptide (IC50 ~ 0.1 μM); blocks Ca2+ currents in dorsal root ganglion neurons. Analgesic in vivo.</p>Formula:C46H71N21O6Purezza:98%Colore e forma:SolidPeso molecolare:1014.2TRPA1-IN-2
CAS:<p>TRPA1-IN-2 is a potent and orally active TRPA1 inhibitor with an IC50 value of 0.04 µM.TRPA1-IN-2 has anti-inflammatory activity.</p>Formula:C24H25F3N4OPurezza:98.05%Colore e forma:SoildPeso molecolare:442.48RN-1665
CAS:<p>RN-1665 is a potent and selective TRPV4 receptor antagonist.</p>Formula:C20H24F5N3O3S2Purezza:>99.99%Colore e forma:SoildPeso molecolare:513.54CBP-1008
<p>CBP-1008 is a dual-ligand peptide-drug conjugate (PDC) with MMAE, targeting folate receptor (FRα) and TRPV6. It exhibits high binding affinity to FRα and low affinity to TRPV6. CBP-1008 shows antitumor activity and can be utilized for research in advanced solid tumors such as colorectal cancer, breast cancer, non-small cell lung cancer, ovarian cancer, adrenocortical carcinoma, and follicular dendritic cell sarcoma.</p>Colore e forma:Odour SolidAP 18
CAS:<p>AP-18 is a potent and selective TRPA1 inhibitor.</p>Formula:C11H12ClNOPurezza:99.85% - 99.96%Colore e forma:SolidPeso molecolare:209.67TRPM8 antagonist 3
CAS:TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).Formula:C13H12N2O4SPurezza:99.74%Colore e forma:SolidPeso molecolare:292.31GSK2798745
CAS:GSK2798745 is an orally active transient receptor potential vanilloid 4 (TRPV4) ion channel blocker (IC50s: 1.8 and 1.6 nM for hTRPV4 and rTRPV4).Formula:C25H28N6O3Colore e forma:SolidPeso molecolare:460.53Resolvin D2
CAS:<p>Resolvin D2 (RvD2) is a TRPV1 inhibitor and pro-ablative mediator with anti-inflammatory, anti-infective and pro-ablative effects.</p>Formula:C22H32O5Purezza:98%Colore e forma:SolidPeso molecolare:376.49NGD-8243
CAS:<p>NGD-8243 (N-[4-(trifluoromethyl)phenyl]-7-[3-(trifluoromethyl)pyridin-2-yl]quinazolin-4-amine) is a TRPV1 inhibitor and can be used in studies for prevention</p>Formula:C21H12F6N4Purezza:95.26%Colore e forma:SolidPeso molecolare:434.34(S)-ABT 102
CAS:<p>N-[(1S)-1H-inden-1-yl]-N'-indazol-4-ylurea is a strong TRPV1 blocker with a 123 nM IC50 against capsaicin.</p>Formula:C21H24N4OPurezza:99.65% - 99.77%Colore e forma:SoildPeso molecolare:348.44BTD
CAS:<p>BTD is a TRPC5 activator that activates heteromeric channel complexes composed of TRPC5 and its closest relatives TRPC1 or TRPC4.</p>Formula:C24H33N3O4SColore e forma:SolidPeso molecolare:459.6Phenazopyridine
CAS:<p>Phenazopyridine is an orally administered azo dye with local analgesic effects on urinary tract infections,. against SARM1 and TRPM8.</p>Formula:C11H11N5Purezza:99.98%Colore e forma:SolidPeso molecolare:213.24ASP7663
CAS:ASP7663 is a TRPA1 Receptor Agonist and exhibiting an abdominal analgesic effect in vivo.Formula:C14H14FNO3Purezza:98.61%Colore e forma:SolidPeso molecolare:263.26PF-4840154
CAS:<p>PF-4840154: potent TrpA1 agonist; EC50 of 97 nM (rat) & 23 nM (human); triggers nociception in mice.</p>Formula:C26H38N6O2Purezza:>99.99%Colore e forma:SolidPeso molecolare:466.62GSK2193874
CAS:<p>GSK2193874 was identified as a selective, orally active TRPV4 blocker.</p>Formula:C37H38BrF3N4OPurezza:98.79% - ≥95%Colore e forma:SolidPeso molecolare:691.62JNJ-17203212
CAS:JNJ-17203212 is a potent and selective antagonist of TRPV1 (human TRPV1 and rat TRPV1, IC50 of 65 nM and 102 nM).Formula:C17H15F6N5OPurezza:99.18%Colore e forma:SolidPeso molecolare:419.32M8-B Hydrochloride
CAS:<p>M8-B Hydrochloride is a selective transient receptor potential melastatin-8 (TRPM8) channel antagonist.</p>Formula:C22H25ClN2O3SPurezza:99.33%Colore e forma:SolidPeso molecolare:432.96SB-366791
CAS:<p>SB-366791 is a new and selective cinnamide TRPV1 antagonist.</p>Formula:C16H14ClNO2Purezza:99.51%Colore e forma:SolidPeso molecolare:287.74Ononetin
CAS:<p>Ononetin (2',4'-Dihydroxy-2-(4-methoxyphenyl)acetophenone) is a TRPM3 channel blocker(IC50: 0.3 μM).</p>Formula:C15H14O4Purezza:98.06%Colore e forma:SolidPeso molecolare:258.27Evifacotrep
CAS:<p>Evifacotrep: TRPC5 antagonist for neurological disease research (WO2020061162, compound 100).</p>Formula:C18H12ClF4N5O2Purezza:98.6%Colore e forma:SolidPeso molecolare:441.77HC067047 Hydrochloride(883031-03-6 free base)
CAS:HC-067047 hydrochloride, a TRPV4 antagonist, selectively inhibits human, rat, and mouse currents with IC50s: 486 nM, 133 nM, and 17 nM.Formula:C26H29ClF3N3O2Purezza:99.95%Colore e forma:SolidPeso molecolare:507.98HC-030031
CAS:<p>HC-030031 (TOSLAB 829227) is a potent TRPA1 inhibitor, which antagonizes AITC- and formalin-evoked calcium influx with IC50s of 6.2 and 5.3 μM, respectively.</p>Formula:C18H21N5O3Purezza:99.69% - ≥95%Colore e forma:SolidPeso molecolare:355.39ML204
CAS:<p>ML204 is a novel potent antagonist that selectively modulates native TRPC4/C5 ion channels.</p>Formula:C15H18N2Purezza:98.1% - 99.72%Colore e forma:SolidPeso molecolare:226.32RN-1734
CAS:<p>RN-1734 is selective TRPV4 channel antagonist(IC50 of 2.3 μM,5.9 μM,3.2 μM for hTRPV4, mTRPV4 and rTRPV4,respectively)</p>Formula:C14H22Cl2N2O2SPurezza:99.1% - 99.3%Colore e forma:SolidPeso molecolare:353.31AMG 333
CAS:<p>AMG 333 is TRPM8 antagonist with an IC50 of 13 nM,a Clinical Candidate for the Treatment of Migraine.</p>Formula:C20H12F5N3O4Purezza:99.95%Colore e forma:SolidPeso molecolare:453.32Chembridge-5861528
CAS:<p>Chembridge-5861528 (TCS 5861528) is a TRPA1 channel blocker that antagonizes AITC- and 4-HNE-evoked calcium influx with IC50 values of 14.3 and 18.7 μM.</p>Formula:C19H23N5O3Purezza:99.97%Colore e forma:SolidPeso molecolare:369.42RQ-00203078
CAS:<p>RQ-00203078 is a highly selective, potent and orally available TRPM8 antagonist.</p>Formula:C21H13ClF6N2O5SPurezza:98% - 99.6%Colore e forma:SolidPeso molecolare:554.85A-967079
CAS:<p>A 967079 is a potent, selective, and bioavailable inhibitor of the TRPA1 channel, with IC50 values of 67 and 289 nM for the human and rat isoforms, respectively</p>Formula:C12H14FNOPurezza:98.34% - 99.75%Colore e forma:SolidPeso molecolare:207.24ICILIN
CAS:<p>ICILIN (AG-3-5) is a synthetic TRPM8 ion channel super-agonist.</p>Formula:C16H13N3O4Purezza:98.45% - ≥95%Colore e forma:Light Yellow SolidPeso molecolare:311.29HC-067047
CAS:<p>HC-067047 is a potent and selective TRPV4 antagonist.Also inhibits the endogenous TRPV4-mediated response to 4α-PDH .</p>Formula:C26H28F3N3O2Purezza:99.45% - 99.97%Colore e forma:SolidPeso molecolare:471.51AM-0902
CAS:<p>AM-0902 is a potent and specific TRPA1 antagonist (IC50s: 71/131 nM for rTRPA1 and hTRPA1).</p>Formula:C17H15ClN6O2Purezza:>99.99%Colore e forma:SolidPeso molecolare:370.79SB 452533
CAS:<p>SB 452533 is an antagonist of the vanilloid receptor 1(pKb: 7.8).</p>Formula:C18H22BrN3OPurezza:99.87%Colore e forma:SolidPeso molecolare:376.29Pico145
CAS:<p>Pico145 (HC-608) is a remarkable inhibitor of TRPC1/4/5 channels.</p>Formula:C23H20ClF3N4O5Purezza:99.06%Colore e forma:SolidPeso molecolare:524.88TRPM4-IN-1
CAS:<p>TRPM4-IN-1 (4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid) is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.</p>Formula:C15H11Cl2NO4Purezza:97.22%Colore e forma:SolidPeso molecolare:340.16MK6-83
CAS:<p>MK6-83 is the transient receptor potential channel ML3 agonist.</p>Formula:C16H20N2O2S2Purezza:99.5%Colore e forma:SolidPeso molecolare:336.479-Phenanthrol
CAS:<p>9-Phenanthrol is inhibitor of the transient receptor potential melastatin 4 (TRPM) channel, a Ca2+ -activated non-selective cation channel.</p>Formula:C14H10OPurezza:98.48%Colore e forma:SolidPeso molecolare:194.23TC-I2000
CAS:<p>TC-I2000 is an TRPM8 channel blocker. Inhibits icilin-induced TRPM8 channel activation in rTRPM8-expressing CHO cells with IC50 of 53 nM.</p>Formula:C23H18F4N2OPurezza:99.778%Colore e forma:SolidPeso molecolare:414.4ML204 hydrochloride
CAS:<p>ML204 hydrochloride (ML204 HCl) is a TRPC4/TRPC5 channel antagonist.</p>Formula:C15H19ClN2Colore e forma:SolidPeso molecolare:262.78WS-12
CAS:WS-12 is a potent TRPM8 agonist that acts as a cooling agent (EC50 : 193 nM)Formula:C18H27NO2Purezza:99.99%Colore e forma:Whitish To White Solid CrystallinePeso molecolare:289.41Pyr10
CAS:<p>Pyr10, a pyrazole derivative, selectively inhibits TRPC3, not STIM1/Orai1, with IC50 of 0.72 μM in TRPC3-HEK293, and 13.08 μM in BRL-2H3 cells.</p>Formula:C18H13F6N3O2SPurezza:99.69% - 99.7%Colore e forma:SolidPeso molecolare:449.37SB-705498
CAS:<p>SB705498 is a TRPV1 antagonist for hTRPV1. SB-705498 has been investigated for the treatment of Rhinitis, Chronic Cough, and Non-allergic Rhinitis.</p>Formula:C17H16BrF3N4OPurezza:99.57% - ≥95%Colore e forma:SolidPeso molecolare:429.23Vanilloid receptor antagonist 1
CAS:<p>Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) is a potent vanilloid receptor TRPV1 antagonist.</p>Formula:C18H15N3O2Purezza:98.14%Colore e forma:SolidPeso molecolare:305.33AMG9810
CAS:<p>AMG 9810 blocks capsaicin's action on TRPV1; human IC50=24.5 nM, rat IC50=85.6 nM.</p>Formula:C21H23NO3Purezza:99.79% - 99.95%Colore e forma:SolidPeso molecolare:337.41Optovin
CAS:<p>Optovin is a TRPA1 activator, which is reversibly photoactivated.</p>Formula:C15H13N3OS2Purezza:99.47% - 99.67%Colore e forma:SolidPeso molecolare:315.41MDR-652
CAS:<p>MDR-652 is a highly specific and efficacious agonist of nonpungent transient receptor potential vanilloid 1 (TRPV1) with Ki value of 11.4 nM and 23.8 nM for</p>Formula:C22H23ClFN3O2SPurezza:99.96%Colore e forma:SolidPeso molecolare:447.95RN-1747
CAS:<p>RN-1747: TRPV4 agonist (EC50: human 0.77 μM, mouse 4.0 μM, rat 4.1 μM), TRPM8 antagonist (IC50: 4 μM).</p>Formula:C17H18ClN3O4SPurezza:99.29%Colore e forma:SolidPeso molecolare:395.86AMTB hydrochloride
CAS:<p>AMTB HCl: Novel TRPM8 blocker, relieves pain, treats urinary issues, moderates bladder reflexes in rats.</p>Formula:C23H27ClN2O2SPurezza:99.08%Colore e forma:SolidPeso molecolare:430.99TRPM8 antagonist 2
CAS:<p>TRPM8 antagonist 2 is a potent and selective TRPM8 antagonist with an IC50 of 0.2 nM. TRPM8 antagonist 2 is used in the research of neuropathic pain syndromes.</p>Formula:C26H26N2O2Purezza:98.1%Colore e forma:SolidPeso molecolare:398.5AC1903
CAS:<p>AC1903 is a specific inhibitor of TRPC5 channel, and has been shown to suppress severe proteinuria and prevent podocyte loss.</p>Formula:C19H17N3OPurezza:98.45%Colore e forma:SolidPeso molecolare:303.36cim0216
CAS:<p>CIM0216 is a synthetic TRPM3 activator whose potency and apparent affinity greatly exceeds that of the canonical TRPM3 agonist.</p>Formula:C21H21N3O2Purezza:99.87%Colore e forma:SolidPeso molecolare:347.41AMG 517
CAS:<p>AMG 517 is an effective and specific TRPV1 antagonist, antagonizes proton (IC50: 0.76 nM), capsaicin (IC50: 0.62 nM) and heat activation (IC50: 1.3 nM) of TRPV1</p>Formula:C20H13F3N4O2SPurezza:99.77% - 99.85%Colore e forma:SolidPeso molecolare:430.4JNJ-28583113
CAS:<p>JNJ-28583113 is a TRPM2 antagonist, inducing phosphorylation of GSK3α and β subunits, protecting cells from oxidative stress-induced cell death.</p>Formula:C19H21F3N2O2Purezza:98.57%Colore e forma:SolidPeso molecolare:366.38SAR7334
CAS:<p>SAR7334 (TRCP6-IN-1) is a potent and specific inhibitor of TRPC6(IC50 of 7.9 nM).</p>Formula:C21H22ClN3OPurezza:99.62% - 99.71%Colore e forma:SolidPeso molecolare:367.87N-Oleoyl Valine
CAS:N-Oleoyl valine, an N-acyl amine, antagonizes TRPV3 for thermoregulation; rises post-cold exposure; elevates in mouse lung injury.Formula:C23H43NO3Peso molecolare:381.59JYL 1421
CAS:<p>JYL 1421 (SC 0030) is an antagonist of TRPV1 receptor (IC50 = 8 nM).</p>Formula:C20H26FN3O2S2Purezza:98.83%Colore e forma:SolidPeso molecolare:423.57AM12
CAS:AM12 inhibits Lanthanide-evoked TRPC5 activity (IC50: 0.28 μM).Formula:C15H9BrO5Purezza:98%Colore e forma:SolidPeso molecolare:349.13TRPC6-PAM-C20
CAS:<p>TRPC6-PAM-C20, a selective enhancer for TRPC6, boosts calcium in HEK cells and OAG-related platelet clumping, EC50: 2.37μM.</p>Formula:C22H21NO4Purezza:98.16%Colore e forma:SolidPeso molecolare:363.41D-3263 hydrochloride
CAS:<p>D-3263 hydrochloride (D3263 HCl salt) is enteric-coated, orally bioavailable transient receptor potential melatonin member 8 (TRPM8) agonist.</p>Formula:C21H32ClN3O3Purezza:99.93%Colore e forma:SolidPeso molecolare:409.95TRPV3 antagonist 74a
CAS:<p>TRPV3 antagonist 74a (TRPV3 74a) is a specific TRPV3 antagonist for the study of neurological disorders.</p>Formula:C17H17F3N2O2Purezza:≥98.0%Colore e forma:SolidPeso molecolare:338.32GSK1702934A
CAS:GSK1702934A is a TRPC3 agonist with pro-arrhythmic and positive inotropic effects and is used in the study of diabetes mellitus.Formula:C22H25N3O2SPurezza:98.15%Colore e forma:SolidPeso molecolare:395.52TRPM4-IN-2
CAS:NBA, or TRPM4-IN-2, is a potent TRPM4 inhibitor with IC50 of 0.16 μM, used in prostate and colorectal cancer research.Formula:C19H14ClNO4Purezza:99.21%Colore e forma:SolidPeso molecolare:355.77Asivatrep
CAS:<p>Asivatrep (PAC14028) is a selective and potent antagonist of transient receptor potential vanilloid subtype 1 (TRPV1) for the study of atopic dermatitis.</p>Formula:C21H22F5N3O3SPurezza:95.13%Colore e forma:SolidPeso molecolare:491.48RN9893
CAS:RN9893 is a selective and potent TRPV4 receptor antagonist with IC50 values of 320, 420 and 660 nM for TRPV4 receptors in mouse, human and rat, respectively.Formula:C21H23F3N4O5SPurezza:99.99%Colore e forma:SolidPeso molecolare:500.49TRPV4 agonist-1
CAS:<p>TRPV4 agonist-1 is an agonist of TRPV4 (EC50: 60 nM in the hTRPV4 Ca2+ assay).</p>Formula:C25H23ClF2N4O2Purezza:98%Colore e forma:SolidPeso molecolare:484.93ABT 102
CAS:<p>ABT 102 (CHEMBL398338) is a selective antagonist of transient receptor potential vanilloid 1 (TRPV1) receptor.</p>Formula:C21H24N4OPurezza:98.38% - 99.86%Colore e forma:SolidPeso molecolare:348.44Mavatrep
CAS:<p>Mavatrep (JNJ-39439335) is a selective antagonist of TRPV1 with Ki of 6.5 nM and can be used for studies about inflammatory pain.</p>Formula:C25H21F3N2OPurezza:98.51% - 99.31%Colore e forma:SolidPeso molecolare:422.44SET 2
CAS:<p>SET 2 is an antagonist of transient receptor potential vanilloid type 2(TRPV2) with an IC50 of 0.46 μM. SET 2 shows selectivity over TRPV1, TRPV3 and TRPV4.</p>Formula:C17H21F3N4O2SPurezza:99.77%Colore e forma:SolidPeso molecolare:402.43Elismetrep
CAS:<p>Elismetrep (MT-8554) is an orally available TRPM8 inhibitor with potential analgesic activity for the study of vasomotor symptoms in postmenopausal women.</p>Formula:C27H21F3N2O5SPurezza:99.37% - 99.93%Colore e forma:SolidPeso molecolare:542.53MSP3
CAS:<p>MSP3 is an agonist of TRPV1 (EC50 = 0.87 μM) and shows antinociceptive and neuroprotective effects.</p>Formula:C16H19NO3SPurezza:99.89%Colore e forma:SolidPeso molecolare:305.39HC-070
CAS:<p>HC-070 is a TRPC5 and TRPC4 antagonist (IC50 = 9.3 nM and 46 nM).</p>Formula:C22H20Cl2N4O4Purezza:98.48%Colore e forma:SolidPeso molecolare:475.32Pyr3
CAS:<p>Pyr3 selectively blocks TRPC3 channels, reducing Ca2+ influx; it's effective at 700 nM.</p>Formula:C16H11Cl3F3N3O3Purezza:98.04%Colore e forma:SolidPeso molecolare:456.63TC-I 2014
CAS:<p>TC-I 2014 shows antiallodynic properties in pain models.</p>Formula:C23H19F6N3OPurezza:99.07%Colore e forma:SolidPeso molecolare:467.41Olvanil
CAS:<p>Olvanil (N-Vannilyloleoylamide) is a vanilloid receptor agonist with EC50 of 0.7nM.</p>Formula:C26H43NO3Purezza:99.58%Colore e forma:SolidPeso molecolare:417.62FEMA-4809
CAS:<p>FEMA-4809 activates TRPM8, the ion channel for cold sensation, and is used as a cooling agent.</p>Formula:C17H17N3O2SPurezza:99.9%Colore e forma:SolidPeso molecolare:327.4JT010
CAS:<p>JT010 is an effective agonist of TRPA1 (EC50 = 0.65 nM).</p>Formula:C16H19ClN2O3SPurezza:99.75%Colore e forma:SolidPeso molecolare:354.85GSK3395879
CAS:<p>GSK3395879 is a selective and orally bioavailable antagonist of transient receptor potential vanilloid-4 (TRPV4) (IC50: 1 nM for hTRPV4).</p>Formula:C20H15F4N3O5SPurezza:98%Colore e forma:SolidPeso molecolare:485.41Mesendogen
CAS:<p>Mesendogen is an inhibitor of transient receptor potential cation channel, subfamily M, member 6 (TRPM6) and 7 (TRPM7) and acts by inhibiting TRPM6/TRPM7</p>Formula:C18H16ClF3N2OSPurezza:99.66%Colore e forma:SolidPeso molecolare:400.85A-1165442
CAS:<p>A-1165442 is a competitive TRPV1 antagonist. For human TRPV, the IC50 values is 9 nM.</p>Formula:C22H20ClF2N3O2Colore e forma:SolidPeso molecolare:431.86MK-2295
CAS:<p>MK-2295 is a potent TRPV1 antagonist. MK-2295 can be used in studies about the treatment of chronic pain.</p>Formula:C27H31FN6O2Purezza:98.83% - 99.44%Colore e forma:SolidPeso molecolare:490.57PF-05105679
CAS:<p>PF-05105679 is a selective TRPM8 antagonist (IC50 = 103 nM). PF-05105679 can be used in research on cold-related pain.</p>Formula:C26H21FN2O3Purezza:99.84%Colore e forma:SolidPeso molecolare:428.45AMG-0347
CAS:<p>AMG-0347 inhibits TRPA1 ion channels in sensory neurons, blocking pain perception.</p>Formula:C24H26F3N3O2Purezza:99.93%Colore e forma:SolidPeso molecolare:445.48AMG2850
CAS:<p>AMG2850 is a potent, orally bioavailable, and selective antagonist of transient receptor potential melastatin 8 (TRPM8).</p>Formula:C19H17F6N3OPurezza:99.84%Colore e forma:SolidPeso molecolare:417.35TRPA1 Antagonist 1
CAS:<p>TRPA1 Antagonist 1 is an antagonist of TRPA1(IC50: 8 nM) and is a methylene phosphate prodrug which converts to its active parent drug.</p>Formula:C24H20F6N5Na2O7PSPurezza:98%Colore e forma:SolidPeso molecolare:713.45Apcin A HCL
CAS:<p>Apcin A HCL is an Apcin derivative. Apcin A HCL is an anaphase-promoting complex (APC) inhibitor. Apcin-A HCL interacts strongly with Cdc20, and inhibits the ubiquitination of Cdc20 substrates. Apcin-A HCL can be used to synthesize the PROTAC CP5V [1].</p>Formula:C10H15Cl4N5O2Purezza:99.30%Colore e forma:SolidPeso molecolare:379.07Motugivatrep
CAS:<p>Motugivatrep is a potent and selective TRPV1 antagonist that can be used to study TRPV1-related respiratory diseases.</p>Formula:C22H20F3NO3Purezza:99.22%Colore e forma:SolidPeso molecolare:403.39
