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Canale del potassio

Canale del potassio

I canali del potassio sono un gruppo diversificato di proteine di membrana che facilitano il flusso di ioni potassio (K+) attraverso la membrana cellulare. Questi canali svolgono un ruolo cruciale nel mantenimento del potenziale di membrana a riposo, nella regolazione del volume cellulare e nel controllo dell'eccitabilità dei neuroni e delle cellule muscolari. I canali del potassio sono coinvolti in vari processi fisiologici, tra cui la regolazione del ritmo cardiaco, la secrezione di insulina e il rilascio di neurotrasmettitori. La disfunzione dei canali del potassio è legata a condizioni come aritmie, epilessia e ipertensione. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei canali del potassio per supportare la tua ricerca in elettrofisiologia, salute cardiovascolare e neurobiologia.

Trovati 283 prodotti di "Canale del potassio"

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  • Oxybutynin

    CAS:
    Oxybutynin (Ditropan) is a synthetic anticholinergic agent that is used for treatment of urinary incontinence and overactive bladder syndrome.
    Formula:C22H31NO3
    Purezza:97.81% - 99.57%
    Colore e forma:White To Off-White Crystalline Powder
    Peso molecolare:357.49

    Ref: TM-T1049L

    1g
    138,00€
    50mg
    39,00€
    100mg
    49,00€
    500mg
    92,00€
    1mL*10mM (DMSO)
    56,00€
  • Clofilium tosylate

    CAS:
    Clofilium tosylate is a potassium channel blocker, induces apoptosis on human promyelocytic leukemia (HL-60) cells.
    Formula:C28H44ClNO3S
    Purezza:99.68% - >99.99%
    Colore e forma:Solid
    Peso molecolare:510.17

    Ref: TM-T14982

    2mg
    34,00€
    5mg
    50,00€
    10mg
    84,00€
    25mg
    158,00€
    50mg
    284,00€
    100mg
    424,00€
    1mL*10mM (DMSO)
    57,00€
  • VU591 hydrochloride

    CAS:
    VU591 hydrochloride is a selective Kir1.1 (ROMK) blocker with IC50 of 0.24 μM, not affecting Kir7.1, Kir2.1, Kir2.3, or Kir4.1, similar to VU 590.
    Formula:C16H13ClN6O5
    Purezza:98.93% - 99.22%
    Colore e forma:Solid
    Peso molecolare:404.76

    Ref: TM-T13320

    1mg
    34,00€
    5mg
    71,00€
    10mg
    105,00€
    25mg
    215,00€
    50mg
    366,00€
    100mg
    512,00€
    200mg
    695,00€
    1mL*10mM (DMSO)
    79,00€
  • Glipizide

    CAS:
    Glipizide (CP 28720) is a short-acting, second-generation sulfonylurea with hypoglycemic activity.
    Formula:C21H27N5O4S
    Purezza:99.67% - 99.75%
    Colore e forma:Solid
    Peso molecolare:445.54

    Ref: TM-T1603

    1g
    58,00€
    500mg
    46,00€
  • NS13001

    CAS:
    NS13001, an oral SK channel modulator, shows promise for SCA2 therapy; EC50: 1.8 µM (SK2), 0.14 µM (SK3).
    Formula:C17H16ClN7
    Purezza:99.55%
    Colore e forma:Solid
    Peso molecolare:353.81

    Ref: TM-T16345

    2mg
    49,00€
    5mg
    97,00€
    10mg
    170,00€
    25mg
    305,00€
    50mg
    432,00€
    100mg
    622,00€
    1mL*10mM (DMSO)
    96,00€
  • Mefloquine hydrochloride

    CAS:
    Mefloquine hydrochloride (Mefloquin hydrochloride) is a quinoline derivative used for the prevention and therapy of P. falciparum malaria.
    Formula:C17H17ClF6N2O
    Purezza:99% - 99.99%
    Colore e forma:Off-White To Yellow Solid
    Peso molecolare:414.77

    Ref: TM-T0860

    25mg
    34,00€
    50mg
    47,00€
    100mg
    56,00€
    200mg
    74,00€
    500mg
    92,00€
    1mL*10mM (DMSO)
    52,00€
  • Dronedarone hydrochloride

    CAS:
    Dronedarone hydrochloride (SR33589) is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.
    Formula:C31H44N2O5S·HCl
    Purezza:99.61%
    Colore e forma:Solid
    Peso molecolare:593.22

    Ref: TM-T1073

    5mg
    38,00€
    10mg
    52,00€
    25mg
    87,00€
    50mg
    117,00€
    100mg
    170,00€
    200mg
    250,00€
    500mg
    424,00€
    1mL*10mM (DMSO)
    55,00€
  • Indapamide

    CAS:
    Indapamide (Noranat) is a non-thiazide sulphonamide diuretic compound, generally used in the treatment of hypertension, as well as decompensated cardiac failure.
    Formula:C16H16ClN3O3S
    Purezza:98.97% - 99.83%
    Colore e forma:Solid
    Peso molecolare:365.83

    Ref: TM-T1498

    1mL*10mM (DMSO)
    35,00€
  • IK1 inhibitor PA-6

    CAS:
    IK1 inhibitor PA-6 (PA-6) is a selective and potent inhibitor of IK1 (KIR2.x ion-channel-carried inward rectifier current)(IC50 of 12-15 nM for human and mouse
    Formula:C31H32N4O2
    Purezza:98.9%
    Colore e forma:Solid
    Peso molecolare:492.61

    Ref: TM-T15555

    2mg
    38,00€
    5mg
    56,00€
    10mg
    98,00€
    25mg
    178,00€
    50mg
    303,00€
    100mg
    444,00€
    1mL*10mM (DMSO)
    63,00€
  • Minoxidil

    CAS:
    Minoxidil (U10858) is an orally administered vasodilator with hair growth stimulatory and antihypertensive effects.
    Formula:C9H15N5O
    Purezza:99.885% - >99.99%
    Colore e forma:Crystals From Methanol-Acetonitrile Solid
    Peso molecolare:209.25

    Ref: TM-T0451

    1g
    55,00€
    1mL*10mM (DMSO)
    55,00€
  • Eleclazine hydrochloride

    CAS:
    Eleclazine hydrochloride (GS 6615 hydrochloride) is a novel inhibitor of late Na+ current (IC50: 0.7 uM).
    Formula:C21H17ClF3N3O3
    Purezza:99.86%
    Colore e forma:Solid
    Peso molecolare:451.83

    Ref: TM-T15207

    1mg
    62,00€
    5mg
    116,00€
    10mg
    170,00€
    25mg
    283,00€
    50mg
    424,00€
    100mg
    562,00€
    200mg
    743,00€
    1mL*10mM (DMSO)
    128,00€
  • Ketanserin

    CAS:
    Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.
    Formula:C22H22FN3O3
    Purezza:99.19% - 99.73%
    Colore e forma:Solid
    Peso molecolare:395.43

    Ref: TM-T1066

    25mg
    34,00€
    100mg
    50,00€
    200mg
    92,00€
    500mg
    133,00€
    1mL*10mM (DMSO)
    50,00€
  • Ropivacaine

    CAS:
    Ropivacaine (LEA-103 HCl) is a local anaesthetic drug belonging to the amino amide group.
    Formula:C17H26N2O
    Purezza:97.75% - >99.99%
    Colore e forma:Solid
    Peso molecolare:274.40

    Ref: TM-T0386L

    10mg
    46,00€
    25mg
    60,00€
    50mg
    77,00€
    100mg
    90,00€
    1mL*10mM (DMSO)
    50,00€
  • DCPIB

    CAS:

    DCPIB, a known specific and potent inhibitor of volume-regulated anion channels (VRAC),DCPIB displayed superior selectivity toward TRESK with an IC50 of 0.14 μM

    Formula:C22H28Cl2O4
    Purezza:99.79% - 99.87%
    Colore e forma:Solid
    Peso molecolare:427.36

    Ref: TM-T10979

    2mg
    43,00€
    5mg
    64,00€
    10mg
    97,00€
    25mg
    197,00€
    50mg
    334,00€
    100mg
    537,00€
    200mg
    748,00€
  • BMS-394136

    CAS:
    BMS-394136 (BMS 394136) is a KV1.5 antagonist for the treatment of cardiovascular diseases such as arrhythmias and atrial fibrillation.
    Formula:C24H21Cl2FN4O
    Purezza:98.59% - 99.95%
    Colore e forma:Solid
    Peso molecolare:471.35

    Ref: TM-T30520

    1mg
    248,00€
    5mg
    613,00€
    10mg
    873,00€
    25mg
    1.311,00€
    50mg
    1.768,00€
    100mg
    2.365,00€
    500mg
    4.684,00€
  • VU0134992 hydrochloride

    CAS:
    VU0134992 hydrochloride is the first subtype-preferring, orally active and selective blocker of Kir4.1 potassium channel pore(IC50 : 0.97 μM).
    Formula:C20H32BrClN2O2
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:447.84

    Ref: TM-T13316

    5mg
    37,00€
    10mg
    59,00€
    25mg
    104,00€
    50mg
    170,00€
    100mg
    283,00€
    200mg
    437,00€
    1mL*10mM (DMSO)
    42,00€
  • Tannic acid

    CAS:
    Tannic acid (Gallotannic acid) is a novel hERG channel blocker.
    Formula:C76H52O46
    Purezza:AR - AR
    Colore e forma:Light Yellow To Light Brown Solid Solid Particulate/Powder
    Peso molecolare:1701.2

    Ref: TM-T0801

    1g
    37,00€
    5g
    52,00€
    10g
    66,00€
    25g
    87,00€
  • Repaglinide

    CAS:
    Repaglinide, a benzoic acid derivative, stimulates insulin, treats type 2 diabetes, and may rarely cause acute liver injury.
    Formula:C27H36N2O4
    Purezza:99.73% - >99.99%
    Colore e forma:White To Off-White Solid
    Peso molecolare:452.59

    Ref: TM-T1088

    10mg
    35,00€
    25mg
    50,00€
    50mg
    59,00€
    100mg
    87,00€
    500mg
    164,00€
    1mL*10mM (DMSO)
    59,00€
  • Glibenclamide

    CAS:
    Glibenclamide (Glyburide) is an antidiabetic sulfonylurea derivative with actions similar to those of chlorpropamide.
    Formula:C23H28ClN3O5S
    Purezza:99.05% - 99.75%
    Colore e forma:Solid
    Peso molecolare:494.00

    Ref: TM-T1634

    1g
    58,00€
    500mg
    49,00€
    1mL*10mM (DMSO)
    55,00€
  • Tertiapin-Q

    CAS:
    Tertiapin-Q is a bee toxin derivative that inhibits BK-type K(+) channels in a concentration-dependent manner, inhibiting efflux to K(+).
    Formula:C106H175N35O24S4
    Purezza:98.06% - 98.09%
    Colore e forma:Solid
    Peso molecolare:2452

    Ref: TM-TP2114

    1mg
    137,00€
    5mg
    295,00€
    10mg
    442,00€
    25mg
    708,00€
    50mg
    964,00€
    100mg
    1.288,00€