
Canale del potassio
I canali del potassio sono un gruppo diversificato di proteine di membrana che facilitano il flusso di ioni potassio (K+) attraverso la membrana cellulare. Questi canali svolgono un ruolo cruciale nel mantenimento del potenziale di membrana a riposo, nella regolazione del volume cellulare e nel controllo dell'eccitabilità dei neuroni e delle cellule muscolari. I canali del potassio sono coinvolti in vari processi fisiologici, tra cui la regolazione del ritmo cardiaco, la secrezione di insulina e il rilascio di neurotrasmettitori. La disfunzione dei canali del potassio è legata a condizioni come aritmie, epilessia e ipertensione. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei canali del potassio per supportare la tua ricerca in elettrofisiologia, salute cardiovascolare e neurobiologia.
Trovati 280 prodotti di "Canale del potassio"
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SCH-23390 hydrochloride
CAS:SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Formula:C17H19Cl2NOPurezza:98% - 99.83%Colore e forma:SolidPeso molecolare:324.24Ref: TM-T4369
1mg39,00€2mg50,00€5mg78,00€10mg97,00€25mg195,00€50mg369,00€100mg550,00€1mL*10mM (DMSO)78,00€ICA-105574
CAS:ICA-105574 activates hERG, enhancing peak current and shortening action potential, while modulating activation kinetics.Formula:C19H14N2O4Purezza:98.89%Colore e forma:SolidPeso molecolare:334.33Ref: TM-T9009
1mg43,00€5mg92,00€10mg144,00€25mg298,00€50mg469,00€100mg687,00€200mg938,00€1mL*10mM (DMSO)92,00€Branaplam
CAS:<p>Branaplam (LMI 070) is a highly potent, selective and orally active small molecule SMN2 splicing modulator.</p>Formula:C22H27N5O2Purezza:98.28% - 99.72%Colore e forma:SolidPeso molecolare:393.48Rosuvastatin
CAS:<p>Rosuvastatin (ZD4522) is an inhibitor of HMG-CoA reductase (HMGCR). Rosuvastatin has hypolipidemic and antiatherosclerotic effects. Cost-effective and quality-assured.</p>Formula:C22H28FN3O6SPurezza:95.24% - 99.8%Colore e forma:SolidPeso molecolare:481.54Levosimendan
CAS:<p>Levosimendan (OR1259) is a calcium sensitizer for acute heart failure, enhancing cardiac contractility without raising calcium levels.</p>Formula:C14H12N6OPurezza:99.37% - 99.91%Colore e forma:Yellow Crystalline PowderPeso molecolare:280.28H3B-120
CAS:H3B-120: selective, competitive CPS1 inhibitor with anti-cancer properties. IC50: 1.5 μM, Ki: 1.4 μM.Formula:C19H24N4O2SPurezza:99.03% - 99.2%Colore e forma:SolidPeso molecolare:372.48Ref: TM-T11529
1mg40,00€2mg52,00€5mg85,00€10mg125,00€25mg264,00€50mg425,00€100mg682,00€200mg944,00€1mL*10mM (DMSO)93,00€CLP290
CAS:CLP290 is an activator of the neuron-specific K+-Cl cotransporter KCC2 and displays potential for the treatment of a wide range of neurological and psychiatricFormula:C19H21FN4O3SPurezza:99.93% - >99.99%Colore e forma:SolidPeso molecolare:404.46Ref: TM-T5444
1mg37,00€5mg77,00€10mg123,00€25mg202,00€50mg303,00€100mg454,00€200mg663,00€1mL*10mM (DMSO)65,00€BMS-191011
CAS:<p>BMS-191011 (BMS-A) is an activator of large-conductance calcium-activated potassium (BKCa) channels ,effective in stroke models</p>Formula:C16H10ClF3N2O3Purezza:97.43%Colore e forma:SolidPeso molecolare:370.71Tetrandrine
CAS:Tetrandrine (Sinomenine A) is a naturally occurring biphenylisoquinoline alkaloid, a calcium channel inhibitor. Cost-effective and quality-assured.Formula:C38H42N2O6Purezza:99.61% - 99.94%Colore e forma:White SolidPeso molecolare:622.75Doxapram
CAS:Doxapram (Dopram) is a respiratory stimulant that inhibits TASK-1, TASK-3, and TASK-1/TASK-3 heterodimer channels.Formula:C24H30N2O2Purezza:99.42%Colore e forma:SolidPeso molecolare:378.51VU590
CAS:VU590 is an inhibitor of extrarenal medullary potassium ROMK.VU590 inhibits Kir7.1 and modulates uterine myometrial contractility and melanocortin signalling.Formula:C24H32N4O7Purezza:98.06%Colore e forma:SolidPeso molecolare:488.53BL-1249
CAS:BL-1249 is a selective and potent non-steroidal potassium channel activator with anti-inflammatory activity that activates K2P2.1 (TREK-1) and K2P10.1 (TREK-2).Formula:C17H17N5Purezza:98% - 98.25%Colore e forma:SolidPeso molecolare:291.35Ref: TM-T14666
1mg52,00€5mg111,00€10mg170,00€25mg259,00€50mg354,00€100mg620,00€500mg1.283,00€1mL*10mM (DMSO)155,00€HUP30
CAS:HUP30 is a potent vasodilating agent. HUP30 can stimulate soluble guanylyl cyclase, activate K+ channels, and block extracellular Ca2+ influx.Formula:C14H15N3O3SPurezza:99.96%Colore e forma:SolidPeso molecolare:305.35Ref: TM-TNU0864
5mg38,00€10mg56,00€25mg101,00€50mg164,00€100mg235,00€200mg328,00€1mL*10mM (DMSO)42,00€Eleclazine
CAS:Eleclazine (GS-6615) is a novel and selective voltage-gated sodium channel inhibitor with antiarrhythmic properties that reduces peak sodium current (INaP).Formula:C21H16F3N3O3Purezza:98.67%Colore e forma:SolidPeso molecolare:415.37Repaglinide D5
CAS:Repaglinide D5 is deuterium labeled Repaglinide. Repaglinide is an insulin secretagogue for treatment type-2 diabetes mellitus.Formula:C27H36N2O4Purezza:98%Colore e forma:SolidPeso molecolare:457.62Dofetilide D4
CAS:Dofetilide D4 (UK 68789 D4), a deuterium-labeled version of Dofetilide, is categorized as a Class III antiarrhythmic medication.Formula:C19H27N3O5S2Purezza:98%Colore e forma:SolidPeso molecolare:445.59Meclofenamic acid
CAS:Meclofenamic acid: non-selective gap-junction blocker, FTO inhibitor, anti-inflammatory.Formula:C14H11Cl2NO2Purezza:99.98%Colore e forma:SolidPeso molecolare:296.15Ref: TM-T11990
1mg88,00€5mg188,00€10mgPrezzo su richiesta25mg474,00€50mg658,00€1mL*10mM (DMSO)255,00€LY 303511
CAS:LY303511, an inactive analogue of LY294002, is a mTOR inhibitor and no inhibition for PI3-K.Formula:C19H18N2O2Purezza:98%Colore e forma:SolidPeso molecolare:306.36CPK20
CAS:CPK20 is a potent and selective inhibitor of the KCNT1 channel, useful for epilepsy research.Formula:C23H24F6N2O2SColore e forma:SolidPeso molecolare:506.50Nifekalant hydrochloride
CAS:Nifekalant hydrochloride is an IKr potassium channel blocker with an IC50 of 10 µM.Formula:C19H28ClN5O5Purezza:99.91%Colore e forma:SolidPeso molecolare:441.91
