
Canale del calcio
I canali del calcio sono proteine di membrana che regolano il flusso di ioni calcio dentro e fuori dalle cellule, essenziale per varie funzioni cellulari, tra cui la contrazione muscolare, il rilascio di neurotrasmettitori e l'espressione genica. La disfunzione dell'attività dei canali del calcio è associata a condizioni come ipertensione, aritmie cardiache e disturbi neurologici. Presso CymitQuimica, offriamo un'ampia selezione di modulatori dei canali del calcio per supportare la tua ricerca in salute cardiovascolare, neurobiologia e trasduzione del segnale.
Trovati 493 prodotti di "Canale del calcio"
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3',4'-Dichlorobenzamil HCl
CAS:<p>3',4'-Dichlorobenzamil HCl is an inhibitor of Na+ transport, Na+/Ca2+ exchanger, sarcoplasmic reticulum Ca2+ release channels.</p>Formula:C13H12Cl3N7OPurezza:98%Colore e forma:Yellow SolidPeso molecolare:388.64BAY-Y-5959
CAS:<p>BAY-Y-5959, a calcium channel agonist, is used potentially for the treatment of arrhythmia, heart failure and myocardial.</p>Formula:C26H24N4O2Colore e forma:SolidPeso molecolare:424.49Aprindine hydrochloride
CAS:<p>Aprindine HCl, a Class 1b antiarrhythmic, treats heart arrhythmias, outperforming digoxin in delaying atrial fibrillation. It's effective orally.</p>Formula:C22H31ClN2Colore e forma:SolidPeso molecolare:358.95Levamlodipine gentisate
CAS:<p>Levamlodipine gentisate, an active amlodipine enantiomer, is a dihydropyridine calcium channel blocker for treating hypertension and angina.</p>Formula:C27H31ClN2O9Purezza:98%Colore e forma:SolidPeso molecolare:563Flordipine
CAS:<p>Flordipine is used as a calcium channel blocker.</p>Formula:C26H33F3N2O5Purezza:98%Colore e forma:SolidPeso molecolare:510.55S-312-d
CAS:<p>S-312d is a calcium channel antagonist. S-312-d can offer marked neuronal protective effects against ischemic injury.</p>Formula:C20H22N2O4SPurezza:98%Colore e forma:SolidPeso molecolare:386.46Niguldipine Free Base
CAS:<p>Niguldipine Free Base is a calcium channel blocker and a₁-adrenergic receptor antagonist and a clinical modulator of multidrug resistance.</p>Formula:C36H39N3O6Purezza:98.97%Colore e forma:SolidPeso molecolare:609.71CGP 28392
CAS:<p>CGP 28392 is used as a partial calcium channel agonist.</p>Formula:C18H17F2NO5Purezza:98%Colore e forma:SolidPeso molecolare:365.33ML218
CAS:<p>ML218 is an inhibitor of T-type Ca2+ channels (Cav3.1, Cav3.2, Cav3.3).ML218 inhibits the synaptic activity of subthalamic nucleus (STN) neurons.</p>Formula:C19H26Cl2N2OPurezza:99.2% - 99.45%Colore e forma:SolidPeso molecolare:369.33Aladorian
CAS:<p>Aladorian (ARM036), a benzothiazepine, has anti-arrhythmic properties for heart failure and CPVT research.</p>Formula:C12H13NO4SPurezza:98%Colore e forma:SolidPeso molecolare:267.3Carboxyamidotriazole
CAS:<p>Carboxyamidotriazole is a cytostatic inhibitor of non-voltage-operated calcium channels and calcium channel-mediated signaling pathways.</p>Formula:C17H12Cl3N5O2Purezza:98%Colore e forma:SolidPeso molecolare:424.67Topiramate lithium
CAS:<p>Topiramate lithium: antiepileptic, GluR5 antagonist, enhances GABA, inhibits kainate/AMPA, Na+/Ca2+ channels; ↑ K+ conductance; ↓ carbonic anhydrase.</p>Formula:C12H20LiNO8SColore e forma:SolidPeso molecolare:345.29YS-201
CAS:<p>YS-201 is an antagonist of dihydropyridine-type calcium channel.</p>Formula:C24H31N3O6Purezza:98%Colore e forma:SolidPeso molecolare:457.52JTV-519
CAS:<p>K201 (JTV-519) is a Ca2+-dependent blocker and prevents abnormal Ca(2+) leak from the sarcoplasmic reticulum in the ischemic heart and skeletal muscle (SkM) by</p>Formula:C25H33ClN2O2SPurezza:99.88%Colore e forma:SolidPeso molecolare:461.06JTV-519 fumarate
CAS:<p>Ryanodine receptor (RyR) inhibitor; stabilizes RyR2 in a closed conformation. Exhibits antiarrhythmic and cardioprotective properties in vivo.</p>Formula:C29H36N2O6SColore e forma:SolidPeso molecolare:540.67Halofuginone hydrobromide
CAS:<p>Halofuginone specifically inhibits collagen type I and MMP-2 gene expression, which may result in the suppression of angiogenesis and tumor cell growth.</p>Formula:C16H17BrClN3O3·HBrPurezza:97.01% - 99.73%Colore e forma:SolidPeso molecolare:495.59Gallopamil hydrochloride
CAS:<p>Gallopamil hydrochloride (Methoxyverapamil hydrochloride) is an antagonist of phenylalkylamine calcium.</p>Formula:C28H41ClN2O5Purezza:99.86%Colore e forma:SolidPeso molecolare:521.0918:0 LYSO-PE
CAS:<p>18:0 LYSO-PE is a compound that induces an increase in [Ca2+]i and can be used as a phospholipid (PL) standard for lipid analysis by electrospray mass spectrometry (ESI-MS)/MS.</p>Formula:C23H48NO7PPurezza:98%Colore e forma:SolidPeso molecolare:481.6Norverapamil
CAS:<p>Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .</p>Formula:C26H36N2O4Purezza:98%Colore e forma:SolidPeso molecolare:440.58DHP-218
CAS:<p>DHP-218, a calcium channel blocker, inhibits rat aorta contractions; pA2: 9.11, IC50: 6.3 nmol/L (high K+) & 66 nmol/L (phenylephrine).</p>Formula:C18H21N2O7PPurezza:98%Colore e forma:SolidPeso molecolare:408.34
