
Canale del calcio
I canali del calcio sono proteine di membrana che regolano il flusso di ioni calcio dentro e fuori dalle cellule, essenziale per varie funzioni cellulari, tra cui la contrazione muscolare, il rilascio di neurotrasmettitori e l'espressione genica. La disfunzione dell'attività dei canali del calcio è associata a condizioni come ipertensione, aritmie cardiache e disturbi neurologici. Presso CymitQuimica, offriamo un'ampia selezione di modulatori dei canali del calcio per supportare la tua ricerca in salute cardiovascolare, neurobiologia e trasduzione del segnale.
Trovati 493 prodotti di "Canale del calcio"
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TTA-P2
CAS:<p>TTA-P2: potent CNS-penetrating T-type Ca2+ channel blocker; eliminates Cav3.1 window currents.</p>Formula:C21H29Cl2FN2O2Colore e forma:SolidPeso molecolare:431.37(R)-Amlodipine
CAS:<p>(R)-Amlodipine is the R-enantiomer of Amlodipine and functions as an orally active dihydropyridine calcium channel blocker with antianginal properties.</p>Formula:C20H25ClN2O5Purezza:99.977%Colore e forma:SolidPeso molecolare:408.88(R)-Lercanidipine hydrochloride
CAS:<p>(R)-Lercanidipine hydrochloride is the R-enantiomer of Lercanidipine. (R)-lercanidipine hydrochloride is a blocker of calcium channel.</p>Formula:C36H42ClN3O6Purezza:98%Colore e forma:SolidPeso molecolare:648.2Lercanidipine. (R)-
CAS:<p>(R)-Lercanidipine enantiomer: antihypertensive, blocks L-type Ca2+ channels, dilates blood vessels.</p>Formula:C36H41N3O6Colore e forma:SolidPeso molecolare:611.73Sadopine
CAS:<p>Sadopine is a high-affinity radioligand for DHP receptor in L-type Ca2+ channels, suitable for tissue and membrane labeling.</p>Formula:C30H40F3N3O7SColore e forma:SolidPeso molecolare:643.71TMB 8 (hydrochloride)
CAS:<p>TMB 8 blocks nAChRs (IC50: 390-480 nM), reduces Ca2+ in muscles, hinders rabbit aorta contraction at 50 μM, and inhibits PKC dose-dependently.</p>Formula:C22H38ClNO5Colore e forma:White SolidPeso molecolare:431.99YM 244769 hydrochloride
CAS:<p>inhibitor of the reverse mode of Na+/Ca2+ exchange (NCX)</p>Formula:C26H23ClFN3O3Purezza:98%Colore e forma:SolidPeso molecolare:479.93McN5691
CAS:<p>McN5691 is a voltage sensitive calcium channel blocker.</p>Formula:C30H35NO3Purezza:98.93% - 99.38%Colore e forma:SolidPeso molecolare:457.6TTA-Q6
CAS:<p>TTA-Q6 is a T-type Ca2+ channel antagonist that inhibits the uptake of extracellular calcium ions by tumour cells for the treatment of neurological diseases.</p>Formula:C20H15ClF3N3OPurezza:99.97%Colore e forma:SolidPeso molecolare:405.8piCRAC-1
CAS:<p>piCRAC-1 is a powerful inhibitor of the photoinducible Ca2+ release-activated Ca2+ (CRAC) channel.</p>Formula:C17H10F6N4Colore e forma:SolidPeso molecolare:384.28Ned-K
CAS:<p>Ned-K blocks NAADP, reduces heart ischemia-reperfusion calcium waves.</p>Formula:C31H31N5O3Colore e forma:SolidPeso molecolare:521.61Nemadipine-A
CAS:<p>Nemadipine A blocks L-type Ca2+ channels, alters C. elegans morphology, boosts TRAIL's cancer kill rate, and lowers Survivin in A549 cells.</p>Formula:C19H18F5NO4Colore e forma:SolidPeso molecolare:419.34TDN345
CAS:<p>TDN345 is a antagonist of Ca2+, for the treatment of vascular and senile dementia including Alzheimer's disease.</p>Formula:C28H34F2N2O2Purezza:98%Colore e forma:SolidPeso molecolare:468.58GSK-5503A
CAS:<p>GSK-5503A is a novel channel blocker of CRAC.</p>Formula:C23H17F2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:405.4Cavα2δ1&NET-IN-2
CAS:<p>Cavα2δ1&NET-IN-2 .</p>Formula:C22H26N6O2SColore e forma:SolidPeso molecolare:438.55AJG-049 HCl
CAS:<p>AJG-049 HCl is a calcium channel antagonist that inhibits L-type Ca2+ channels via diltiazem-binding site(s).</p>Formula:C27H31ClN2O2Colore e forma:SolidPeso molecolare:451.01PD-151307
CAS:<p>PD-151307 is used as an N-type calcium channel blocker.</p>Formula:C33H47N3O5Purezza:98%Colore e forma:SolidPeso molecolare:565.74(Rac)-MEM 1003
CAS:<p>MEM-1003, a calcium channel blocker, is used potentially for the treatment of bipolar disorders.</p>Formula:C22H25ClN2O5Colore e forma:SolidPeso molecolare:432.9BK 129
CAS:<p>BK 129 is a local anesthetic with relaxant properties. BK 129 inhibits Ca2+ entry into the smooth muscle cell and Ca2+ release from sarcoplasmic reticulum.</p>Formula:C22H36N2O4Purezza:98%Colore e forma:SolidPeso molecolare:392.53(2R/S)-6-PNG
CAS:<p>(2R/S)-6-PNG (6-Prenylnaringenin) from hops is a natural histone deacetylase inhibitor that blocks T-type calcium channels reducing neurogenicity in mice.</p>Formula:C20H20O5Purezza:98%Colore e forma:SolidPeso molecolare:340.37
