
Canale del calcio
I canali del calcio sono proteine di membrana che regolano il flusso di ioni calcio dentro e fuori dalle cellule, essenziale per varie funzioni cellulari, tra cui la contrazione muscolare, il rilascio di neurotrasmettitori e l'espressione genica. La disfunzione dell'attività dei canali del calcio è associata a condizioni come ipertensione, aritmie cardiache e disturbi neurologici. Presso CymitQuimica, offriamo un'ampia selezione di modulatori dei canali del calcio per supportare la tua ricerca in salute cardiovascolare, neurobiologia e trasduzione del segnale.
Trovati 493 prodotti di "Canale del calcio"
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RyRs activator 3
CAS:<p>RyRs activator 3 (compound A4) serves as an insecticide highly effective against both the diamondback moths, M.</p>Formula:C23H19BrCl2N6O3Purezza:98%Colore e forma:SolidPeso molecolare:578.25AMG-1
CAS:<p>AMG-1 inhibits CRAC channels, blocks effector T cells, not regulatory ones, and reduces EAE progression.</p>Formula:C18H9ClF5N3OColore e forma:SolidPeso molecolare:413.73RQ-00311651
CAS:<p>RQ-00311651 is a novel T-type Ca2+ channel blocker. RQ-00311651 also inhibited high K-induced Ca signaling in those cells.</p>Formula:C19H18F3N5O2Colore e forma:SolidPeso molecolare:405.37β-Amino Acid Imagabalin Hydrochloride
CAS:<p>β-Amino Acid Imagabalin Hydrochloride is the voltage-dependent calcium channel ligand for the α2δ subunit.</p>Formula:C9H20ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:209.71Lidoflazine
CAS:<p>Lidoflazine: antianginal, blocks HERG K+ & Ca channels, risks QT prolongation & arrhythmia.</p>Formula:C30H35F2N3OPurezza:98%Colore e forma:SolidPeso molecolare:491.62Semotiadil recemate fumarate
CAS:<p>Semotiadil recemate fumarate is the recemate of Semotiadil fumarate. Semotiadil fumarate is a novel antagonist of vasoselective Ca2+ channel.</p>Formula:C33H36N2O10SPurezza:98%Colore e forma:SolidPeso molecolare:652.71PD 122860
CAS:<p>PD 122860 is a dihydropyridine enhancing heart contractility, altering ECG, and relaxing aortic rings.</p>Formula:C23H20F3N3O4SPurezza:98%Colore e forma:SolidPeso molecolare:491.48GSK205
CAS:<p>GSK205 is a selective TRPV4 antagonist (IC50: 4.19 μM) for inhibiting TRPV4-mediated Ca2+ influx.</p>Formula:C24H25BrN4SPurezza:99.46%Colore e forma:SolidPeso molecolare:481.45SAK3
CAS:<p>SAK3 is a modulator of nAChR activity and is used to study memory deficits and Alzheimer's disease.</p>Formula:C20H23N3O4Purezza:98.37% - 99.43%Colore e forma:SolidPeso molecolare:369.41Tamolarizine
CAS:<p>Tamolarizine (Tamolarizine free base) free base is a novel calcium antagonist.</p>Formula:C27H32N2O3Purezza:98.17%Colore e forma:SoildPeso molecolare:432.55O-1602
CAS:<p>O-1602 is a novel GPR55 agonist, an atypical cannabinoid associated with the central nervous system and obesity, and is a candidate compound for the treatment</p>Formula:C17H22O2Purezza:99.85%Colore e forma:SolidPeso molecolare:258.36Sulcardine sulfate
CAS:<p>Sulcardine sulfate (B-87823) is a multi-ion channel blocker with antiarrhythmic activity that inhibits Na+, K+, and Ca2+ channels.</p>Formula:C24H35N3O8S2Purezza:98.74%Colore e forma:SolidPeso molecolare:557.68Crobenetine
CAS:<p>Crobenetine (BIII 890 CL) Free Base is a selective NaV channel blocker that eliminates VTD-induced [Ca2+] elevation.</p>Formula:C25H33NO2Purezza:98.99%Colore e forma:SolidPeso molecolare:379.54Clopimozide
CAS:<p>Clopimozide (R-29764), a long-acting oral antischizophrenic, blocks calcium channels and [3H] nilandipine binding.</p>Formula:C28H28ClF2N3OPurezza:98.19% - >99.99%Colore e forma:SolidPeso molecolare:495.99CP-060
CAS:<p>CP-060 is a potent Ca2+ antagonist and inhibits Ca2+ overload with antioxidant and cardioprotective activities.</p>Formula:C30H42N2O5SPurezza:99.54%Colore e forma:SolidPeso molecolare:542.73Opc 8490
CAS:<p>Opc 8490 is a cardiotonic agent and a positive inotropic vasodilator, which prolongs the atrial action potential in a concentration-dependent manner.</p>Formula:C30H35N3O10Purezza:98.88%Colore e forma:SolidPeso molecolare:597.61Vatanidipine
CAS:<p>Vatanidipine (AE0047) is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.A slow-onset and long-lasting</p>Formula:C41H42N4O6Purezza:99.95%Colore e forma:SolidPeso molecolare:686.8Enecadin
CAS:<p>Enecadin is a neuroprotective agent.</p>Formula:C21H28FN3OPurezza:98.53%Colore e forma:SolidPeso molecolare:357.46Tiapamil hydrochloride
CAS:<p>Tiapamil hydrochloride (Ro 11-1781 hydrochloride) is a calcium channel blocker with antihypertensive activity used in the study of angina pectoris.</p>Formula:C26H38ClNO8S2Purezza:99.17%Colore e forma:SolidPeso molecolare:592.16Diproteverine HCl
CAS:<p>Diproteverine HCl is a novel calcium antagonist with antianginal properties, antispasmodic and vasoactive.</p>Formula:C26H36ClNO4Purezza:98.55% - 99.84%Colore e forma:SolidPeso molecolare:462.02
