
Canale del calcio
I canali del calcio sono proteine di membrana che regolano il flusso di ioni calcio dentro e fuori dalle cellule, essenziale per varie funzioni cellulari, tra cui la contrazione muscolare, il rilascio di neurotrasmettitori e l'espressione genica. La disfunzione dell'attività dei canali del calcio è associata a condizioni come ipertensione, aritmie cardiache e disturbi neurologici. Presso CymitQuimica, offriamo un'ampia selezione di modulatori dei canali del calcio per supportare la tua ricerca in salute cardiovascolare, neurobiologia e trasduzione del segnale.
Trovati 493 prodotti di "Canale del calcio"
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JNJ-26990990
CAS:<p>"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."</p>Formula:C9H10N2O2S2Purezza:97.37%Colore e forma:SolidPeso molecolare:242.32Efonidipine
CAS:Efonidipine (NZ-105)(NZ-105) is a dihydropyridine calcium channel blocker, blocking both T-type and L-type calcium channels.Formula:C34H38N3O7PPurezza:98.35% - 99.47%Colore e forma:SolidPeso molecolare:631.66Bepridil hydrochloride
CAS:<p>Bepridil hydrochloride (CERM 1978) is a calcium channel blocker and also inhibits Na+/Ca2+ exchange (NCX), sodium channels and cardiac sarcolemmal KATP channels</p>Formula:C24H35ClN2OPurezza:99.45% - 99.68%Colore e forma:SolidPeso molecolare:4032,5-Di-tert-butylhydroquinone
CAS:<p>2,5-Di-tert-butylhydroquinone (BHQ) is an effective and selective endoplasmic reticulum Ca2+-ATPase inhibitor.</p>Formula:C14H22O2Purezza:97.11%Colore e forma:PelletslargecrystalsPeso molecolare:222.32Quadrol
CAS:<p>Quadrol (EDTP) is an immunostimulant, accelerated wound healing.</p>Formula:C14H32N2O4Purezza:99.91% - 99.92%Colore e forma:Viscous Liquid Liquid ViscousPeso molecolare:292.41DHBP dibromide
CAS:<p>DHBP dibromide (1,1'-DI-N-HEPTYL-4,4'-BIPYRIDINIUM DIBRO) is calcium release and a muscle relaxant inhibitor.</p>Formula:C24H38Br2N2Purezza:99.73%Colore e forma:Yellow To Yellow-Green Powder Or FlakesPeso molecolare:514.38GSK1016790A
CAS:<p>GSK1016790A (GSK101) (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial</p>Formula:C28H32Cl2N4O6S2Purezza:97.37% - 99.38%Colore e forma:SolidPeso molecolare:655.61Propiverine hydrochloride
CAS:<p>Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB).</p>Formula:C23H30ClNO3Purezza:99.93%Colore e forma:White Crystalling PowerPeso molecolare:403.94S107
CAS:<p>S107 stabilizes RyR2 by improving calstabin2 binding to mutant/PKA-phosphorylated channels.</p>Formula:C11H15NOSPurezza:99.90%Colore e forma:SolidPeso molecolare:209.31Praeruptorin E
CAS:<p>Praeruptorin C/E relaxes arteries, reduces heart contractility, acting like calcium blockers. D/E protect mice from acid lung injury by halting PMNs and IL-6.</p>Formula:C24H28O7Purezza:98.04% - 99.95%Colore e forma:SolidPeso molecolare:428.47(±)-Praeruptorin A
CAS:<p>(±)-Praeruptorin A could exhibit its anti-osteoclastogenic activity by inhibiting p38/Akt-c-Fos-NFATc1 signaling and PLCγ-independent Ca(2+) oscillation.</p>Formula:C21H22O7Purezza:98.9% - 99.73%Colore e forma:SolidPeso molecolare:386.4(+)-Kavain
CAS:<p>(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.</p>Formula:C14H14O3Purezza:97% - ≥95%Colore e forma:White Fine PowderPeso molecolare:230.26Suvecaltamide
CAS:<p>Suvecaltamide (MK-8998) as potent inhibitors of T-type calcium channels.</p>Formula:C20H23F3N2O2Purezza:99.29% - 99.70%Colore e forma:SolidPeso molecolare:380.4NP118809
CAS:<p>NP118809 (39-1B4) is a potent N-type calcium channel blocker(IC50 : 0.11 μM).</p>Formula:C32H32N2OPurezza:97.74% - 98.68%Colore e forma:SolidPeso molecolare:460.61NS-638
CAS:<p>NS-638 is a Ca2+-channel blocker. It can block K+-stimulated intracellular Ca2+-elevation (IC50: 3.4 μM).</p>Formula:C15H11ClF3N3Purezza:98.44%Colore e forma:SolidPeso molecolare:325.72Pyr6
CAS:<p>Pyr6 (N-[4-[3,5-Bis(trifluoromethyl)-1H-pyrazol-1-yl]phenyl]-3-fluoro-4-pyridinecarboxamide) is a selective TRPC3 inhibitor with IC50 of 0.49 uM(Ca2+ influx</p>Formula:C17H9F7N4OPurezza:98.89%Colore e forma:SolidPeso molecolare:418.27HC-056456
CAS:<p>HC-056456 (3,4-Bis(2-thienoyl)-1,2,5-oxadiazole-N-oxide) is a CatSper channel modulator.</p>Formula:C12H6N2O4S2Purezza:99.62% - 99.65%Colore e forma:SolidPeso molecolare:306.32Efonidipine hydrochloride monoethanolate
CAS:<p>Efonidipine HCl monoethanolate is a calcium blocker, boosts dehydroepiandrosterone sulfate in NCI-H295R cells.</p>Formula:C36H45ClN3O8PPurezza:>99.99%Colore e forma:SolidPeso molecolare:714.18Mirogabalin
CAS:<p>Mirogabalin (DS5565) is a calcium channel blocker with analgesic effects.</p>Formula:C12H19NO2Purezza:98.57%Colore e forma:SolidPeso molecolare:209.28Ibutilide Fumarate
CAS:<p>Ibutilide Fumarate is a class III antiarrhythmic, prolonging action potentials by enhancing sodium influx, and can extend QT interval.</p>Formula:(C20H36N2O3S)2·C4H4O4Purezza:99.68% - 99.74%Colore e forma:SolidPeso molecolare:885.23
