Canale del calcio
I canali del calcio sono proteine di membrana che regolano il flusso di ioni calcio dentro e fuori dalle cellule, essenziale per varie funzioni cellulari, tra cui la contrazione muscolare, il rilascio di neurotrasmettitori e l'espressione genica. La disfunzione dell'attività dei canali del calcio è associata a condizioni come ipertensione, aritmie cardiache e disturbi neurologici. Presso CymitQuimica, offriamo un'ampia selezione di modulatori dei canali del calcio per supportare la tua ricerca in salute cardiovascolare, neurobiologia e trasduzione del segnale.
Trovati 493 prodotti di "Canale del calcio"
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Nicardipine-d3 hydrochloride
CAS:<p>Nicardipine D3 hydrochloride is the deuterium labeled Nicardipine hydrochloride.</p>Formula:C26H30ClN3O6Purezza:98%Colore e forma:SolidPeso molecolare:519YM-244769 dihydrochloride
CAS:<p>YM-244769 dihydrochloride is an effective inhibitor of Na+/Ca2+ exchange 3 (NCX3) with an IC50 of 18 nM.</p>Formula:C26H24Cl2FN3O3Purezza:98%Colore e forma:SolidPeso molecolare:516.39HSK16149
CAS:<p>HSK16149 is a novel ligand of voltage-gated calcium channel (VGCC) α 2 δ subunit with analgesic activity.</p>Formula:C12H19NO2Colore e forma:SolidPeso molecolare:209.28MRS1845
CAS:<p>MRS1845 is a selective inhibitor of store-operated calcium (SOC) channel (IC50 of 1.7 μM).</p>Formula:C21H22N2O6Purezza:99.69%Colore e forma:SolidPeso molecolare:398.41(S)-Nicardipine
CAS:<p>(S)-Nicardipine is the less active S enantiomer of Nicardipine. Nicardipine is a blocker of calcium channel(IC50 of 1 μM for blocking cardiac calcium channels).</p>Formula:C26H29N3O6Colore e forma:SolidPeso molecolare:479.53Almorexant hydrochloride
CAS:<p>Almorexant hydrochloride (ACT 078573 hydrochloride) is a dual orexin receptor antagonist that induces apoptosis and can be used to study sleep disorders.</p>Formula:C29H32ClF3N2O3Purezza:99.85%Colore e forma:SolidPeso molecolare:549.02Norverapamil-d7
CAS:<p>Norverapamil D7 is a deuterium labeled Norverapamil . Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .</p>Formula:C26H36N2O4Purezza:98%Colore e forma:SolidPeso molecolare:447.62Hexadecylphosphoserine TFA
<p>Hexadecylphosphoserine is a type of phospholipid molecule that incorporates a long-chain alkyl group (hexadecyl) and a phosphatidylserine group, granting it high affinity for cell membranes. This compound exhibits antitumor activity by modulating [Ca++]i and related signaling pathways, making it useful for breast cancer research.</p>Formula:C21H41F3NO8PColore e forma:SolidPeso molecolare:523.52Dronedarone
CAS:<p>Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.</p>Formula:C31H44N2O5SPurezza:98.85% - 99.58%Colore e forma:SolidPeso molecolare:556.76Azumolene
CAS:<p>Azumolene (EU4093 free base)</p>Formula:C13H9BrN4O3Purezza:98.1% - 98.35%Colore e forma:SolidPeso molecolare:349.14Ginsenoside Rd
CAS:<p>Ginsenoside Rd (Gypenoside VIII) may have properties that inhibit or prevent the growth of tumors.</p>Formula:C48H82O18Purezza:99.13% - 99.92%Colore e forma:SolidPeso molecolare:947.15JNJ-26990990
CAS:<p>"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."</p>Formula:C9H10N2O2S2Purezza:97.37%Colore e forma:SolidPeso molecolare:242.32Efonidipine
CAS:Efonidipine (NZ-105)(NZ-105) is a dihydropyridine calcium channel blocker, blocking both T-type and L-type calcium channels.Formula:C34H38N3O7PPurezza:98.35% - 99.47%Colore e forma:SolidPeso molecolare:631.66Bepridil hydrochloride
CAS:<p>Bepridil hydrochloride (CERM 1978) is a calcium channel blocker and also inhibits Na+/Ca2+ exchange (NCX), sodium channels and cardiac sarcolemmal KATP channels</p>Formula:C24H35ClN2OPurezza:99.45% - 99.68%Colore e forma:SolidPeso molecolare:4032,5-Di-tert-butylhydroquinone
CAS:<p>2,5-Di-tert-butylhydroquinone (BHQ) is an effective and selective endoplasmic reticulum Ca2+-ATPase inhibitor.</p>Formula:C14H22O2Purezza:97.11%Colore e forma:PelletslargecrystalsPeso molecolare:222.32DHBP dibromide
CAS:<p>DHBP dibromide (1,1'-DI-N-HEPTYL-4,4'-BIPYRIDINIUM DIBRO) is calcium release and a muscle relaxant inhibitor.</p>Formula:C24H38Br2N2Purezza:99.73%Colore e forma:Yellow To Yellow-Green Powder Or FlakesPeso molecolare:514.38L-Phenylalanine
CAS:<p>L-Phenylalanine (3-Phenyl-L-alanine) is an essential amino acid and the precursor of the amino acid tyrosine, acts as an antagonist at α2δ calcium channels.</p>Formula:C9H11NO2Purezza:99.37% - 99.87%Colore e forma:Solid CrystallinePeso molecolare:165.19GSK1016790A
CAS:<p>GSK1016790A (GSK101) (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial</p>Formula:C28H32Cl2N4O6S2Purezza:97.37% - 99.38%Colore e forma:SolidPeso molecolare:655.61Propiverine hydrochloride
CAS:<p>Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB).</p>Formula:C23H30ClNO3Purezza:99.93%Colore e forma:White Crystalling PowerPeso molecolare:403.94Dantrolene sodium hemiheptahydrate
CAS:<p>Dantrolene depresses excitation-contraction coupling in skeletal muscle by binding to the ryanodine receptor 1 and decreasing intracellular calcium</p>Formula:C14H9N4NaO5·5H2OPurezza:99.72%Colore e forma:Orange PowderPeso molecolare:399.29Pranidipine
CAS:<p>Pranidipine (OPC-13340) is a novel, long-acting 1,4-dihydropyridine calcium channel blocker.</p>Formula:C25H24N2O6Purezza:99.95%Colore e forma:Yellow SolidPeso molecolare:448.47Aranidipine
CAS:<p>Aranidipine (MPC1304) (MPC1304) is a calcium channel antagonist with potent and long-lasting antihypertensive effects.</p>Formula:C19H20N2O7Purezza:99.15%Colore e forma:SolidPeso molecolare:388.37(±)-Praeruptorin A
CAS:<p>(±)-Praeruptorin A could exhibit its anti-osteoclastogenic activity by inhibiting p38/Akt-c-Fos-NFATc1 signaling and PLCγ-independent Ca(2+) oscillation.</p>Formula:C21H22O7Purezza:98.9% - 99.73%Colore e forma:SolidPeso molecolare:386.4(+)-Kavain
CAS:<p>(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.</p>Formula:C14H14O3Purezza:97% - ≥95%Colore e forma:White Fine PowderPeso molecolare:230.26Suvecaltamide
CAS:<p>Suvecaltamide (MK-8998) as potent inhibitors of T-type calcium channels.</p>Formula:C20H23F3N2O2Purezza:99.29% - 99.70%Colore e forma:SolidPeso molecolare:380.4NS-638
CAS:<p>NS-638 is a Ca2+-channel blocker. It can block K+-stimulated intracellular Ca2+-elevation (IC50: 3.4 μM).</p>Formula:C15H11ClF3N3Purezza:98.44%Colore e forma:SolidPeso molecolare:325.72NFAT Inhibitor-2
CAS:<p>NFAT Inhibitor-2 is a compound used as a molecular building block.</p>Formula:C22H20F2N2O4SPurezza:97.37%Colore e forma:SolidPeso molecolare:446.47Efonidipine hydrochloride monoethanolate
CAS:<p>Efonidipine HCl monoethanolate is a calcium blocker, boosts dehydroepiandrosterone sulfate in NCI-H295R cells.</p>Formula:C36H45ClN3O8PPurezza:>99.99%Colore e forma:SolidPeso molecolare:714.18Praeruptorin E
CAS:<p>Praeruptorin C/E relaxes arteries, reduces heart contractility, acting like calcium blockers. D/E protect mice from acid lung injury by halting PMNs and IL-6.</p>Formula:C24H28O7Purezza:98.04% - 99.95%Colore e forma:SolidPeso molecolare:428.47SR33805
CAS:<p>SR33805 is a potent antagonist of Ca2+ channel(EC50s of 4.1 nM and 33 nM in depolarized and polarized conditions, respectively)</p>Formula:C32H40N2O5SPurezza:99.15%Colore e forma:SolidPeso molecolare:564.74Ibutilide Fumarate
CAS:<p>Ibutilide Fumarate is a class III antiarrhythmic, prolonging action potentials by enhancing sodium influx, and can extend QT interval.</p>Formula:(C20H36N2O3S)2·C4H4O4Purezza:99.68% - 99.74%Colore e forma:SolidPeso molecolare:885.23Azumolene sodium anhydrous
CAS:<p>Azumolene sodium, a muscle relaxant, blocks calcium release from muscles and halts SOCE linked to RyR1 except when induced by thapsigargin.</p>Formula:C13H8BrN4NaO3Colore e forma:SolidPeso molecolare:371.13Argireline
CAS:<p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>Formula:C34H60N14O12SPurezza:96.79% - 99.65%Colore e forma:White PowderPeso molecolare:888.99TGR5 Receptor Agonist
CAS:TGR5 is a potent TGR5(GPCR19) agonist.Formula:C18H14Cl2N2O2Purezza:99.77% - ≥95%Colore e forma:SolidPeso molecolare:361.22Ethacrynic acid
CAS:<p>Ethacrynic acid (Edecrin) 是谷胱甘肽 S-转移酶抑制剂，也是NF-κB 信号传导途径的有效抑制剂，并且还调节白三烯的形成。它还可抑制 L 型电压依赖性和储存操作的钙通道，从而导致气道平滑肌细胞松弛。它是利尿剂，具有抗炎特性，可减轻类维生素 A 诱导的小鼠耳部水肿。</p>Formula:C13H12Cl2O4Purezza:98.61% - 99.85%Colore e forma:Crystals Physical Description White Solid (Ntp 1992)Peso molecolare:303.14Glaucine
CAS:<p>Glaucine: antitussive, antioxidative, antiviral, may fight arthritis, boosts IL-10, hinders breast cancer cell spread by inhibiting MMP-9 and NF-κB.</p>Formula:C21H25NO4Purezza:99.42% - 99.56%Colore e forma:SolidPeso molecolare:355.43HC-056456
CAS:<p>HC-056456 (3,4-Bis(2-thienoyl)-1,2,5-oxadiazole-N-oxide) is a CatSper channel modulator.</p>Formula:C12H6N2O4S2Purezza:99.62% - 99.65%Colore e forma:SolidPeso molecolare:306.32Psoralenoside
CAS:<p>Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.</p>Formula:C17H18O9Purezza:99.03% - 99.49%Colore e forma:SolidPeso molecolare:366.32Quadrol
CAS:<p>Quadrol (EDTP) is an immunostimulant, accelerated wound healing.</p>Formula:C14H32N2O4Purezza:99.91% - 99.92%Colore e forma:Viscous Liquid Liquid ViscousPeso molecolare:292.41Mirogabalin
CAS:<p>Mirogabalin (DS5565) is a calcium channel blocker with analgesic effects.</p>Formula:C12H19NO2Purezza:98.57%Colore e forma:SolidPeso molecolare:209.28Efonidipine hydrochloride
CAS:<p>Efonidipine HCl (NZ-105) blocks T-type/L-type calcium channels; used in hypertension treatment.</p>Formula:C34H39ClN3O7PColore e forma:SolidPeso molecolare:668.12NP118809
CAS:<p>NP118809 (39-1B4) is a potent N-type calcium channel blocker(IC50 : 0.11 μM).</p>Formula:C32H32N2OPurezza:97.74% - 98.68%Colore e forma:SolidPeso molecolare:460.61Praeruptorin C
CAS:<p>Praeruptorin C: an antioxidant, calcium antagonist, protects neurons, reduces vascular hypertrophy, affects cellular signals.</p>Formula:C24H28O7Purezza:99.6% - 99.92%Colore e forma:SolidPeso molecolare:428.47CDN1163
CAS:<p>CDN1163 is a small molecule activator of sarco/endoplasmic reticulum Ca2+-ATPase (SERCA).</p>Formula:C20H20N2O2Purezza:99.83% - ≥95%Colore e forma:SolidPeso molecolare:320.39ABT-639 hydrochloride
CAS:<p>ABT-639 hydrochloride is a selective, novel T-type Ca2+ channel blocker.</p>Formula:C20H21Cl2F2N3O3SColore e forma:SolidPeso molecolare:492.36Pyr6
CAS:<p>Pyr6 (N-[4-[3,5-Bis(trifluoromethyl)-1H-pyrazol-1-yl]phenyl]-3-fluoro-4-pyridinecarboxamide) is a selective TRPC3 inhibitor with IC50 of 0.49 uM(Ca2+ influx</p>Formula:C17H9F7N4OPurezza:98.89%Colore e forma:SolidPeso molecolare:418.27Gabapentin hydrochloride
CAS:<p>Gabapentin hydrochloride (Neurontin HCl) is a GABA analogue, used to treat seizures and neuropathic pain.</p>Formula:C9H17NO2·HClPurezza:99.71%Colore e forma:Off-White SolidPeso molecolare:207.7Pinaverium bromide
CAS:<p>Pinaverium bromide is an calcium channel blocker with Antispasmodic and effectively relieves pain, diarrhea and intestinal discomfort.</p>Formula:C26H41Br2NO4Purezza:99.52%Colore e forma:White Crystalline PowderPeso molecolare:591.42Taurolithocholic acid sodium salt
CAS:<p>Taurolithocholic acid sodium salt (Sodium taurolithocholate) is the major human metabolite, a bile acid which inhibits radioligand binding to muscarinic M1, but</p>Formula:C26H44NNaO5SPurezza:99.79% - 99.93%Colore e forma:SolidPeso molecolare:505.69FPL64176
CAS:<p>FPL64176 is a L-type calcium channels activator.</p>Formula:C22H21NO3Purezza:98.68%Colore e forma:SolidPeso molecolare:347.41
