Canale del calcio
I canali del calcio sono proteine di membrana che regolano il flusso di ioni calcio dentro e fuori dalle cellule, essenziale per varie funzioni cellulari, tra cui la contrazione muscolare, il rilascio di neurotrasmettitori e l'espressione genica. La disfunzione dell'attività dei canali del calcio è associata a condizioni come ipertensione, aritmie cardiache e disturbi neurologici. Presso CymitQuimica, offriamo un'ampia selezione di modulatori dei canali del calcio per supportare la tua ricerca in salute cardiovascolare, neurobiologia e trasduzione del segnale.
Trovati 493 prodotti di "Canale del calcio"
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Gallopamil, (-)-
CAS:<p>Gallopamil, (-)- is an L-type calcium channel blocker. It is used in the treatment of abnormal heart rhythms.</p>Formula:C28H40N2O5Purezza:98%Colore e forma:SolidPeso molecolare:484.63AK-2-38
CAS:<p>AK-2-38 is a nifedipine analogue with potent smooth muscle calcium antagonist action and partial agonist effects on isolated guinea pig left atrium.</p>Formula:C26H30N2O4Purezza:98%Colore e forma:SolidPeso molecolare:434.53Falipamil
CAS:<p>Falipamil, a verapamil derivative, is a calcium channel blocker with antitachycardic and potential antianginal effects.</p>Formula:C24H32N2O5Purezza:98%Colore e forma:SolidPeso molecolare:428.52Tiropramide
CAS:<p>Tiropramide is an antispasmodic drug. It also useful to inhibit the contractile response of the urinary bladder and in managing abdominal pain in IBS.</p>Formula:C28H41N3O3Purezza:98%Colore e forma:SolidPeso molecolare:467.64Bms 188107
CAS:<p>Bms 188107 is a calcium antagonist, it has cardioprotective effects.</p>Formula:C25H26N2O4Purezza:98%Colore e forma:SolidPeso molecolare:418.48AZD 2066
CAS:<p>AZD 2066 is a selective, orally active, and brain-penetrant mGluR5 antagonist with analgesic activity.</p>Formula:C19H16ClN5O2Purezza:98%Colore e forma:SolidPeso molecolare:381.82BBR 2160
CAS:<p>BBR 2160: a calcium-antagonist dihydropyridine derivative, reduces heart tissue contractility and shortens action potentials.</p>Formula:C21H25N3O7SColore e forma:SolidPeso molecolare:463.5DS16570511
CAS:<p>DS16570511 is a novel, cell-permeable inhibitor targeting the mitochondrial calcium uniporter.</p>Formula:C30H25Cl2N3O4Purezza:98.34% - 98.45%Colore e forma:SolidPeso molecolare:562.44Tamolarizine
CAS:<p>Tamolarizine (Tamolarizine free base) free base is a novel calcium antagonist.</p>Formula:C27H32N2O3Purezza:98.17%Colore e forma:SoildPeso molecolare:432.55Tiapamil hydrochloride
CAS:<p>Tiapamil hydrochloride (Ro 11-1781 hydrochloride) is a calcium channel blocker with antihypertensive activity used in the study of angina pectoris.</p>Formula:C26H38ClNO8S2Purezza:99.17%Colore e forma:SolidPeso molecolare:592.16R 56865
CAS:<p>R 56865 is a weak potential-operated channel inhibitor that inhibits the late sodium current in human isolated cardiomyocytes.</p>Formula:C23H28FN3OSPurezza:99.52%Colore e forma:SolidPeso molecolare:413.55Enecadin
CAS:<p>Enecadin is a neuroprotective agent.</p>Formula:C21H28FN3OPurezza:98.53%Colore e forma:SolidPeso molecolare:357.46Clopimozide
CAS:<p>Clopimozide (R-29764), a long-acting oral antischizophrenic, blocks calcium channels and [3H] nilandipine binding.</p>Formula:C28H28ClF2N3OPurezza:98.19% - >99.99%Colore e forma:SolidPeso molecolare:495.99GSK205
CAS:<p>GSK205 is a selective TRPV4 antagonist (IC50: 4.19 μM) for inhibiting TRPV4-mediated Ca2+ influx.</p>Formula:C24H25BrN4SPurezza:99.46%Colore e forma:SolidPeso molecolare:481.45SAK3
CAS:<p>SAK3 is a modulator of nAChR activity and is used to study memory deficits and Alzheimer's disease.</p>Formula:C20H23N3O4Purezza:98.37% - 99.43%Colore e forma:SolidPeso molecolare:369.418-Bromo-cGMP sodium
CAS:<p>8-Bromo-cGMP sodium: PKG activator, eases pain, dilates vessels, reduces Ca2+ currents & insulin release.</p>Formula:C10H10BrN5NaO7PPurezza:99.45%Colore e forma:SolidPeso molecolare:446.09Gallopamil
CAS:<p>Gallopamil blocks acid secretion (IC50: 10.9 μM), acts as antiarrhythmic, vasodilator, and is a methoxy Verapamil derivative.</p>Formula:C28H40N2O5Purezza:99.85%Colore e forma:SolidPeso molecolare:484.63Cronidipine
CAS:<p>Cronidipine (LF 20254), a calcium channel antagonist, is used potentially for the treatment of hypertension and myocardia ischemia.</p>Formula:C30H32ClN3O8Purezza:99.47%Colore e forma:SolidPeso molecolare:598.04Upacicalcet
CAS:<p>Upacicalcet (AJT-240) is a calcium mimetic for SHPT in dialysis, reducing PTH by targeting parathyroid receptors.</p>Formula:C11H14ClN3O6SPurezza:99.83%Colore e forma:SolidPeso molecolare:351.76Vatanidipine
CAS:<p>Vatanidipine (AE0047) is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.A slow-onset and long-lasting</p>Formula:C41H42N4O6Purezza:99.95%Colore e forma:SolidPeso molecolare:686.8Sulcardine sulfate
CAS:<p>Sulcardine sulfate (B-87823) is a multi-ion channel blocker with antiarrhythmic activity that inhibits Na+, K+, and Ca2+ channels.</p>Formula:C24H35N3O8S2Purezza:98.74%Colore e forma:SolidPeso molecolare:557.68O-1602
CAS:<p>O-1602 is a novel GPR55 agonist, an atypical cannabinoid associated with the central nervous system and obesity, and is a candidate compound for the treatment</p>Formula:C17H22O2Purezza:99.85%Colore e forma:SolidPeso molecolare:258.36VU 0240551
CAS:<p>VU 0240551 is a selective antagonist of neuronal K-Cl cotransporter KCC2 inhibitor with an IC50 of 560 nM. VU 0240551 inhibits L-type calcium channels and hERG.</p>Formula:C16H14N4OS2Purezza:99.9%Colore e forma:SolidPeso molecolare:342.44SERCA2a activator 1
CAS:<p>SERCA2a activator 1 boosts heart function by reducing phospholamban restraint and enhancing cardiac contraction-relaxation cycles.</p>Formula:C32H29N3O4SPurezza:99.75%Colore e forma:SolidPeso molecolare:551.66CERM-11956
CAS:<p>Pelretin (BASF 43915) is a potential protein inhibitor for the study of dermatologic diseases.</p>Formula:C29H38N2O7Purezza:99.38%Colore e forma:SolidPeso molecolare:526.62Ticolubant
CAS:<p>Ticolubant: Oral LTB4 antagonist, Ki=0.78 nM; blocks Ca2+ migration, IC50=6.6 nM; anti-inflammatory in mice.</p>Formula:C23H19Cl2NO3SPurezza:99.59%Colore e forma:SolidPeso molecolare:460.37CP-060
CAS:<p>CP-060 is a potent Ca2+ antagonist and inhibits Ca2+ overload with antioxidant and cardioprotective activities.</p>Formula:C30H42N2O5SPurezza:99.54%Colore e forma:SolidPeso molecolare:542.73PD173212
CAS:<p>PD 173212 is a blocker that blocks N-type voltage sensitive calcium channel (Cav2.2).</p>Formula:C38H53N3O3Purezza:99.84%Colore e forma:SolidPeso molecolare:599.85Terflavoxate
CAS:<p>Terflavoxate is a novel, orally active, semisynthetic statin microtubule inhibitor commonly used in combination with capecitabine.</p>Formula:C26H29NO4Purezza:98%Colore e forma:SolidPeso molecolare:419.51Cerebrocrast
CAS:<p>Cerebrocrast (IOS-11212) has anti-inflammatory and hypoglycemic activity, blocks human platelet activation, and is used in the study of diabetes.</p>Formula:C26H35F2NO7Purezza:99.71%Colore e forma:SolidPeso molecolare:511.56Fenoverine
CAS:<p>Fenoverine (Spasmopriv) has antispasmodic activity and can be used to study gastrointestinal spasms.</p>Formula:C26H25N3O3SPurezza:98.34%Colore e forma:SolidPeso molecolare:459.56NecroX-5
CAS:<p>NecroX-5, a derivative of NecroX, exhibits anti-inflammatory and anti-cancer activities. NecroX-5 reduces intracellular calcium concentration.</p>Formula:C27H39N3O9S3Purezza:99.944%Colore e forma:SolidPeso molecolare:645.81Diproteverine HCl
CAS:<p>Diproteverine HCl is a novel calcium antagonist with antianginal properties, antispasmodic and vasoactive.</p>Formula:C26H36ClNO4Purezza:98.55% - 99.84%Colore e forma:SolidPeso molecolare:462.02Opc 8490
CAS:<p>Opc 8490 is a cardiotonic agent and a positive inotropic vasodilator, which prolongs the atrial action potential in a concentration-dependent manner.</p>Formula:C30H35N3O10Purezza:98.88%Colore e forma:SolidPeso molecolare:597.61Lifarizine
CAS:<p>Lifarizine (RS-87476), a calcium-sodium channel antagonist, shows neuroprotective activity in a simplified rat survival model of double vessel occlusion.</p>Formula:C29H32N4Purezza:99.88%Colore e forma:SolidPeso molecolare:436.59AZD-1305
CAS:<p>AZD-1305: novel anti-arrhythmic blocking IKr, Ca, Na currents; useful in arrhythmia research.</p>Formula:C22H31FN4O4Purezza:99.31% - 99.86%Colore e forma:SolidPeso molecolare:434.5N106
CAS:<p>N106 is an activator of the SUMO-activating enzyme, E1 ligase, and triggers intrinsic sumoylation of SERCA2a. N106 can be used in studies about heart failure.</p>Formula:C17H14N4O3SPurezza:99.69%Colore e forma:SolidPeso molecolare:354.38Crobenetine
CAS:<p>Crobenetine (BIII 890 CL) Free Base is a selective NaV channel blocker that eliminates VTD-induced [Ca2+] elevation.</p>Formula:C25H33NO2Purezza:98.99%Colore e forma:SolidPeso molecolare:379.54Mioflazine
CAS:<p>Mioflazine suppresses nucleoside uptake. Mioflazine is an orally active nucleoside transport inhibitor. It has the potential for sleep disorders treatment.</p>Formula:C29H30Cl2F2N4O2Purezza:98%Colore e forma:SolidPeso molecolare:575.48Iganidipine
CAS:<p>Iganidipine（NKY 722） is a new water-soluble Ca2+ antagonist with antihypertensive activity for research and neurological related diseases.</p>Formula:C28H38N4O6Purezza:96.3%Colore e forma:SolidPeso molecolare:526.62RS 5773
CAS:<p>RS 5773 is a benzothiazepine derivative with antianginal effects.</p>Formula:C29H33ClN2O4SPurezza:98%Colore e forma:SolidPeso molecolare:541.1Budiodarone
CAS:<p>Budiodarone (ATI-2042) resembles amiodarone, potentially preventing atrial fibrillation.</p>Formula:C27H31I2NO5Colore e forma:SolidPeso molecolare:703.35Coelenterazine h
CAS:<p>Coelenterazine H, a Ca2+ sensitive synthetic derivative, is a luminescent biomolecule used to measure Ca2+ changes.</p>Formula:C26H21N3O2Purezza:99.49%Colore e forma:Yellow To Brownish PowderPeso molecolare:407.46TROX-1
CAS:<p>TROX-1 is the activation state-dependent Cav2 channel antagonist.</p>Formula:C22H16ClFN6OPurezza:98%Colore e forma:SolidPeso molecolare:434.85Piprofurol
CAS:<p>Piprofurol is used as a Calcium channel blocker.</p>Formula:C26H33NO6Purezza:98%Colore e forma:SolidPeso molecolare:455.54A 425619
CAS:<p>A 425619 (1-(4-(TRIFLUOROMETHYL)BENZYL)-3-(ISOQUINOLIN-5-YL)UREA) is a potent TRPV1 antagonist</p>Formula:C18H14F3N3OPurezza:99.75%Colore e forma:SolidPeso molecolare:345.32Cavα2δ1&NET-IN-3
CAS:<p>Cavα2δ1&NET-IN-3 (example 216) is an inhibitor targeting both the α2δ subunit of voltage-gated calcium channels (VGCC) and the noradrenaline transporter (NET).</p>Formula:C24H30N6O2SColore e forma:SolidPeso molecolare:466.6N-type calcium channel blocker-1
CAS:<p>N-type calcium channel blocker-1 is an orally active analgesic agent,shows high affinity to functionally block N-type calcium channels.</p>Formula:C31H47N3Purezza:98%Colore e forma:SolidPeso molecolare:461.73(S)-(-)-Bay-K-8644
CAS:<p>(S)-(-)-Bay-K-8644 ((S)-(-)-Bay K 8644) is an agonist of L-type Ca2+ channel and activates Ba2+ currents with an EC50 of 32 nM.</p>Formula:C16H15F3N2O4Purezza:98.28% - 99.37%Colore e forma:SolidPeso molecolare:356.3KCa1.1 channel activator-1
<p>A selective vascular KCa1.1 channel stimulator with CaV1.2 blocking ability and mild myorelaxant effects.</p>Formula:C25H16O10Colore e forma:SolidPeso molecolare:476.39
