
Canale del calcio
I canali del calcio sono proteine di membrana che regolano il flusso di ioni calcio dentro e fuori dalle cellule, essenziale per varie funzioni cellulari, tra cui la contrazione muscolare, il rilascio di neurotrasmettitori e l'espressione genica. La disfunzione dell'attività dei canali del calcio è associata a condizioni come ipertensione, aritmie cardiache e disturbi neurologici. Presso CymitQuimica, offriamo un'ampia selezione di modulatori dei canali del calcio per supportare la tua ricerca in salute cardiovascolare, neurobiologia e trasduzione del segnale.
Trovati 493 prodotti di "Canale del calcio"
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Sulcardine sulfate
CAS:<p>Sulcardine sulfate (B-87823) is a multi-ion channel blocker with antiarrhythmic activity that inhibits Na+, K+, and Ca2+ channels.</p>Formula:C24H35N3O8S2Purezza:98.74%Colore e forma:SolidPeso molecolare:557.68O-1602
CAS:<p>O-1602 is a novel GPR55 agonist, an atypical cannabinoid associated with the central nervous system and obesity, and is a candidate compound for the treatment</p>Formula:C17H22O2Purezza:99.85%Colore e forma:SolidPeso molecolare:258.36VU 0240551
CAS:<p>VU 0240551 is a selective antagonist of neuronal K-Cl cotransporter KCC2 inhibitor with an IC50 of 560 nM. VU 0240551 inhibits L-type calcium channels and hERG.</p>Formula:C16H14N4OS2Purezza:99.9%Colore e forma:SolidPeso molecolare:342.44SERCA2a activator 1
CAS:<p>SERCA2a activator 1 boosts heart function by reducing phospholamban restraint and enhancing cardiac contraction-relaxation cycles.</p>Formula:C32H29N3O4SPurezza:99.75%Colore e forma:SolidPeso molecolare:551.66CERM-11956
CAS:<p>Pelretin (BASF 43915) is a potential protein inhibitor for the study of dermatologic diseases.</p>Formula:C29H38N2O7Purezza:99.38%Colore e forma:SolidPeso molecolare:526.62Ticolubant
CAS:<p>Ticolubant: Oral LTB4 antagonist, Ki=0.78 nM; blocks Ca2+ migration, IC50=6.6 nM; anti-inflammatory in mice.</p>Formula:C23H19Cl2NO3SPurezza:99.59%Colore e forma:SolidPeso molecolare:460.37CP-060
CAS:<p>CP-060 is a potent Ca2+ antagonist and inhibits Ca2+ overload with antioxidant and cardioprotective activities.</p>Formula:C30H42N2O5SPurezza:99.54%Colore e forma:SolidPeso molecolare:542.73PD173212
CAS:<p>PD 173212 is a blocker that blocks N-type voltage sensitive calcium channel (Cav2.2).</p>Formula:C38H53N3O3Purezza:99.84%Colore e forma:SolidPeso molecolare:599.85Terflavoxate
CAS:<p>Terflavoxate is a novel, orally active, semisynthetic statin microtubule inhibitor commonly used in combination with capecitabine.</p>Formula:C26H29NO4Purezza:98%Colore e forma:SolidPeso molecolare:419.51Cerebrocrast
CAS:<p>Cerebrocrast (IOS-11212) has anti-inflammatory and hypoglycemic activity, blocks human platelet activation, and is used in the study of diabetes.</p>Formula:C26H35F2NO7Purezza:99.71%Colore e forma:SolidPeso molecolare:511.56Fenoverine
CAS:<p>Fenoverine (Spasmopriv) has antispasmodic activity and can be used to study gastrointestinal spasms.</p>Formula:C26H25N3O3SPurezza:98.34%Colore e forma:SolidPeso molecolare:459.56NecroX-5
CAS:<p>NecroX-5, a derivative of NecroX, exhibits anti-inflammatory and anti-cancer activities. NecroX-5 reduces intracellular calcium concentration.</p>Formula:C27H39N3O9S3Purezza:99.944%Colore e forma:SolidPeso molecolare:645.81Diproteverine HCl
CAS:<p>Diproteverine HCl is a novel calcium antagonist with antianginal properties, antispasmodic and vasoactive.</p>Formula:C26H36ClNO4Purezza:98.55% - 99.84%Colore e forma:SolidPeso molecolare:462.02Opc 8490
CAS:<p>Opc 8490 is a cardiotonic agent and a positive inotropic vasodilator, which prolongs the atrial action potential in a concentration-dependent manner.</p>Formula:C30H35N3O10Purezza:98.88%Colore e forma:SolidPeso molecolare:597.61Lifarizine
CAS:<p>Lifarizine (RS-87476), a calcium-sodium channel antagonist, shows neuroprotective activity in a simplified rat survival model of double vessel occlusion.</p>Formula:C29H32N4Purezza:99.88%Colore e forma:SolidPeso molecolare:436.59AZD-1305
CAS:<p>AZD-1305: novel anti-arrhythmic blocking IKr, Ca, Na currents; useful in arrhythmia research.</p>Formula:C22H31FN4O4Purezza:99.31% - 99.86%Colore e forma:SolidPeso molecolare:434.5N106
CAS:<p>N106 is an activator of the SUMO-activating enzyme, E1 ligase, and triggers intrinsic sumoylation of SERCA2a. N106 can be used in studies about heart failure.</p>Formula:C17H14N4O3SPurezza:99.69%Colore e forma:SolidPeso molecolare:354.38Crobenetine
CAS:<p>Crobenetine (BIII 890 CL) Free Base is a selective NaV channel blocker that eliminates VTD-induced [Ca2+] elevation.</p>Formula:C25H33NO2Purezza:98.99%Colore e forma:SolidPeso molecolare:379.54Mioflazine
CAS:<p>Mioflazine suppresses nucleoside uptake. Mioflazine is an orally active nucleoside transport inhibitor. It has the potential for sleep disorders treatment.</p>Formula:C29H30Cl2F2N4O2Purezza:98%Colore e forma:SolidPeso molecolare:575.48Iganidipine
CAS:<p>Iganidipine(NKY 722) is a new water-soluble Ca2+ antagonist with antihypertensive activity for research and neurological related diseases.</p>Formula:C28H38N4O6Purezza:96.3%Colore e forma:SolidPeso molecolare:526.62
