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Canale del calcio

Canale del calcio

I canali del calcio sono proteine di membrana che regolano il flusso di ioni calcio dentro e fuori dalle cellule, essenziale per varie funzioni cellulari, tra cui la contrazione muscolare, il rilascio di neurotrasmettitori e l'espressione genica. La disfunzione dell'attività dei canali del calcio è associata a condizioni come ipertensione, aritmie cardiache e disturbi neurologici. Presso CymitQuimica, offriamo un'ampia selezione di modulatori dei canali del calcio per supportare la tua ricerca in salute cardiovascolare, neurobiologia e trasduzione del segnale.

Trovati 541 prodotti di "Canale del calcio"

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  • Mipsagargin

    CAS:
    Mipsagargin (G-202) is a new antibiotic that inhibits DNA biosynthesis.
    Formula:C66H100N6O27
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1409.52
  • Cavα2δ-IN-1

    CAS:
    Cavα2δ-IN-1 demonstrates exceptional specificity for voltage-gated calcium channels Cavα2δ-1 (with a Ki value of 6 nM), in comparison to Cavα2δ-2 (with a Ki
    Formula:C18H27N5O
    Colore e forma:Solid
    Peso molecolare:329.448
  • MMK 1

    CAS:
    Potent hFPR2 agonist; EC50: 1 nM (mFPR2), 2 nM (hFPR2), >10,000 nM (hFPR1). Induces monocyte/neutrophil migration, boosts IL-1β/IL-6, activates NADPH-oxidase.
    Formula:C75H123N19O18S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1610.97
  • Flosatidil

    CAS:
    Flosatidil is a small molecule voltage-gated calcium channel complex (VDCCs) blocker for the treatment of neurological disorders and cardiovascular diseases,
    Formula:C26H34F3N3O3S
    Purezza:99.87% - 99.99%
    Colore e forma:Solid
    Peso molecolare:525.63
  • ProTx-I

    CAS:
    <p>Selective blocker for CaV3.1 (IC50 = 0.2 μM), CaV3.2 (31.8 μM), also inhibits NaV1.8 and blocks KV2.1 channels.</p>
    Formula:C171H245N53O47S6
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3987.51
  • Lyso-Globotriaosylceramide (d18:1)

    CAS:
    Lyso-Gb3, lacking fatty acyl, binds Stx1 with cholesterol and phosphatidylcholine, not Stx2; lowers neutrophil viability; accumulates in Fabry disease.
    Formula:C36H67NO17
    Colore e forma:Solid
    Peso molecolare:785.922
  • Sulcardine 2HCl

    CAS:
    Sulcardine 2HCl is a multi-ion channel blocker that blocks the properties of hERG and hNav1.5 channels and can be used to study atrial fibrillation.
    Formula:C24H35Cl2N3O4S
    Purezza:99.33% - 99.76%
    Colore e forma:Soild
    Peso molecolare:532.523
  • ω-Conotoxin MVIIC

    CAS:
    Peptide neurotoxin; wide spectrum blocker of N, P and Q type calcium channels.
    Formula:C106H178N40O32S7
    Purezza:98%
    Colore e forma:White Lyophilised Solid
    Peso molecolare:2749
  • NAADP tetrasodium salt

    CAS:
    Ca2+ mobilizing agent
    Formula:C21H27N6O18P3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:744.39
  • Triphenylethylene

    CAS:
    <p>Compound PDK0283, with CAS No. 58-72-0, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0283 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>
    Formula:C20H16
    Colore e forma:White Powder
    Peso molecolare:256.34
  • DMNPE-4 AM-caged-calcium

    CAS:
    DMNPE-4 AM is an EGTA analogue, Ca2+-selective, with Kd 48 nM (pH 7.2) and 19 nM (pH 7.4). Photolysis reduces its Ca2+ affinity to ~2 nM.
    Formula:C34H47N3O22
    Colore e forma:Solid
    Peso molecolare:849.749
  • OPC 8490 free base

    CAS:
    OPC 8490 free base is a positive inotropic vasodilator and a cardiotonic agent that can be used to study cardiovascular diseases.
    Formula:C24H27N3O3
    Purezza:99.53%
    Colore e forma:Soild
    Peso molecolare:405.49
  • PACAP-38 (31-38), human, mouse, rat TFA


    PACAP-38 (31-38), human, mouse, rat (TFA) demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal.
    Formula:C49H84F3N17O13
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1176.29
  • Nesiritide acetate

    CAS:
    Nesiritide, a 32-amino acid natriuretic peptide and recombinant form of human brain natriuretic peptide, enhances vasorelaxation ex vivo in porcine hearts from an acute coronary occlusion model when given as a 2 µg/kg bolus dose followed by a 0.01 µg/kg per minute infusion, facilitated by the calcium ionophore A23187. Formulations containing nesiritide have been utilized in managing congestive heart failure.
    Formula:C143H244N50O42S4C2H4O2
    Colore e forma:Solid
    Peso molecolare:3524.1
  • LY393615


    LY393615 (NCC1048) is a novel blocker of both neuronal Ca²⁺ (calcium) and Na⁺ (sodium) channels, exhibiting half-maximal inhibitory concentrations (IC₅₀) of 1.9
    Purezza:98%
    Colore e forma:Odour Solid
  • sFTX-3.3

    CAS:
    sFTX-3.3 is a calcium ion channel antagonist, exhibiting IC50 values of approximately 0.24 mM and 0.70 mM against P-type and N-type channels respectively.
    Formula:C12H29N7O
    Colore e forma:Solid
    Peso molecolare:287.412
  • β-Cyfluthrin

    CAS:
    β-Cyfluthrin is a type II synthetic pyrethroid compound commonly utilized as an active ingredient in agricultural insecticide products.
    Formula:C22H18Cl2FNO3
    Colore e forma:Solid
    Peso molecolare:434.29
  • (S)-Lercanidipine D3 hydrochloride

    CAS:
    (S)-Lercanidipine D3 hydrochloride is a deuterium labeled Lercanidipine D3 hydrochloride. (S)-Lercanidipine hydrochloride is an agent of antihypertensive.
    Formula:C36H42ClN3O6
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:651.21
  • Magnesium sulfate

    CAS:
    Magnesium sulfate: anticonvulsant for eclampsia, tocolytic agent.
    Formula:MgSO4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:120.37
  • (R)-Nicardipine

    CAS:
    (R)-Nicardipine is the less active R enantiomer of Nicardipine. Nicardipine is a blocker of calcium channel(IC50 of 1 μM for blocking cardiac calcium channels).
    Formula:C26H29N3O6
    Colore e forma:Solid
    Peso molecolare:479.53