
Ricettore GABA
I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.
Trovati 369 prodotti di "Ricettore GABA"
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HIE-124
CAS:HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.Formula:C10H12N2O3SPurezza:98%Colore e forma:SolidPeso molecolare:240.28Suclofenide
CAS:Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.Formula:C16H13ClN2O4SPurezza:98%Colore e forma:SolidPeso molecolare:364.8(S)-Baclofen
CAS:(S)-Baclofen may treat hyperacusis and tinnitus by reducing auditory pathway excitation.Formula:C10H12ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:213.66ABP-700
CAS:ABP-700 is a positive allosteric modulator of the GABAA receptor.Formula:C17H18N2O4Purezza:98%Colore e forma:SolidPeso molecolare:314.34Nerisopam
CAS:Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.Formula:C18H19N3O2Purezza:98.52%Colore e forma:SolidPeso molecolare:309.36Ref: TM-T28159
1mg88,00€5mg190,00€10mg286,00€25mg464,00€50mg672,00€100mg945,00€200mg1.279,00€1mL*10mM (DMSO)256,00€BPDBA
CAS:BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 andFormula:C19H20Cl2N2OPurezza:99.43% - 99.95%Colore e forma:SolidPeso molecolare:363.28RWJ-51204
CAS:RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.
Formula:C21H19F2N3O3Purezza:99.57% - 99.95%Colore e forma:SolidPeso molecolare:399.39Ref: TM-T16811
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€Alpidem
CAS:Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.Formula:C21H23Cl2N3OPurezza:99.56% - 99.97%Colore e forma:White To Off-White SolidPeso molecolare:404.33Ref: TM-T26600
1mg62,00€5mg144,00€10mg219,00€25mg393,00€50mg550,00€100mg787,00€500mg1.596,00€1mL*10mM (DMSO)129,00€NNC 05-711
CAS:NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.Formula:C21H23ClN2O3Purezza:99.92%Colore e forma:SolidPeso molecolare:386.87Divaplon
CAS:Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.Formula:C17H17N3O2Purezza:97.44% - 98.25%Colore e forma:SolidPeso molecolare:295.34DSP-0565
CAS:DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.Formula:C14H12FNOPurezza:99.51% - 99.56%Colore e forma:SolidPeso molecolare:229.25Ref: TM-T11106
1mg109,00€2mg163,00€5mg241,00€10mg354,00€25mg532,00€50mg745,00€100mg1.018,00€500mg2.035,00€1mL*10mM (DMSO)208,00€Sarmazenil
CAS:Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.Formula:C15H14ClN3O3Purezza:99.46%Colore e forma:SolidPeso molecolare:319.74DMCM hydrochloride
CAS:DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.Formula:C17H19ClN2O4Purezza:99.56%Colore e forma:SolidPeso molecolare:350.8Ref: TM-T11061
1mg34,00€2mg50,00€5mg80,00€10mg105,00€25mg236,00€50mg439,00€100mg620,00€1mL*10mM (DMSO)88,00€Ru-32514
CAS:Ru-32514 is a benzodiazepine receptor agonist.Formula:C18H17N3O2Purezza:99.21%Colore e forma:SolidPeso molecolare:307.35ELB-139
CAS:ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.Formula:C14H16ClN3OPurezza:>99.99%Colore e forma:SolidPeso molecolare:277.75L-838417
CAS:L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disordersFormula:C19H19F2N7OPurezza:98.12% - 99.70%Colore e forma:SolidPeso molecolare:399.4Saripidem
CAS:Saripidem (SL-85.0274) is a compound with anxiolytic activity.Formula:C19H20ClN3OPurezza:98.42%Colore e forma:SolidPeso molecolare:341.83Lirequinil
CAS:Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.Formula:C26H25ClN2O3Purezza:98.54%Colore e forma:SolidPeso molecolare:448.94Riluzole hydrochloride
CAS:Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).Formula:C8H6ClF3N2OSPurezza:99.76%Colore e forma:SolidPeso molecolare:270.66Golexanolone
CAS:Golexanolone can be used to study neurological diseases.Formula:C21H31NO2Purezza:99.90% - 99.99%Colore e forma:SolidPeso molecolare:329.48
