
Ricettore GABA
I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.
Trovati 369 prodotti di "Ricettore GABA"
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Fipronil
CAS:Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.Formula:C12H4Cl2F6N4OSPurezza:97.21%Colore e forma:Solid PowderPeso molecolare:437.15Cholesterol myristate
CAS:Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.
Formula:C41H72O2Purezza:99.65%Colore e forma:SolidPeso molecolare:597.01Acetoxyvalerensre
CAS:Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.
Formula:C17H24O4Purezza:98.22%Colore e forma:SolidPeso molecolare:292.37Gabazine
CAS:Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)Formula:C15H18BrN3O3Purezza:98.51% - 99.24%Colore e forma:SolidPeso molecolare:368.23α-Asarone
CAS:alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.Formula:C12H16O3Purezza:99.64% - 99.64%Colore e forma:Monoclinic Needles From Water Monoclinic Needles From WaterPeso molecolare:208.254-Acetamidobutanoic acid
CAS:4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.Formula:C6H11NO3Purezza:98.51%Colore e forma:SolidPeso molecolare:145.16CGP52432
CAS:CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).Formula:C15H24Cl2NO4PPurezza:98.75%Colore e forma:SolidPeso molecolare:384.246-(4-Methoxyphenyl)-3-pyridazinamine
CAS:6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonistFormula:C11H11N3OPurezza:99.03%Colore e forma:SolidPeso molecolare:201.22AZD-6280
CAS:AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.Formula:C20H22N4O3Purezza:98.99%Colore e forma:SolidPeso molecolare:366.41Ref: TM-T7136
1mg227,00€5mg464,00€10mg677,00€25mg1.074,00€50mg1.501,00€100mg2.043,00€1mL*10mM (DMSO)510,00€Tiagabine
CAS:Tiagabine (NO050328) is an Anti-epileptic Agent.Formula:C20H25NO2S2Purezza:99.25% - 99.67%Colore e forma:White To Off-White Crystalline SolidPeso molecolare:375.55CL 218872
CAS:CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.Formula:C13H9F3N4Purezza:99.92%Colore e forma:SolidPeso molecolare:278.23Piperazine
CAS:Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.Formula:C4H10N2Colore e forma:SolidPeso molecolare:86.14Amentoflavone
CAS:Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.Formula:C30H18O10Purezza:98.21% - 99.22%Colore e forma:Odourless Whitish SolidPeso molecolare:538.46Ref: TM-T3417
2mg34,00€5mg50,00€10mg80,00€25mg126,00€50mg215,00€100mg349,00€200mg512,00€1mL*10mM (DMSO)59,00€Pikamilone
CAS:Pikamilone (Picamilon) is an intelligent medicine.Formula:C10H12N2O3Purezza:99.38%Colore e forma:White Crystalline PowderPeso molecolare:208.21Songorine
CAS:Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.Formula:C22H31NO3Purezza:98% - 99.92%Colore e forma:SolidPeso molecolare:357.49Aminooxyacetic acid hemihydrochloride
CAS:Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABAFormula:C2H5NO3·5HClPurezza:98.03%Colore e forma:Light Beige Crystalline PowderPeso molecolare:109.32'MeO6MF
CAS:2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functionalFormula:C17H14O3Purezza:99.28% - 99.63%Colore e forma:SolidPeso molecolare:266.29Ref: TM-T8887
1mg51,00€5mg107,00€10mg160,00€25mg255,00€50mg359,00€100mg485,00€200mg662,00€1mL*10mM (DMSO)101,00€Tiagabine hydrochloride hydrate
CAS:Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.Formula:C20H28ClNO3S2Colore e forma:SolidPeso molecolare:430.02AZD7325
CAS:AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.
Formula:C19H19FN4O2Purezza:99.83%Colore e forma:SolidPeso molecolare:354.38(-)-Securinine
CAS:(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.Formula:C13H15NO2Purezza:99.58% - 99.87%Colore e forma:SolidPeso molecolare:217.26
