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Ricettore GABA

Ricettore GABA

I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.

Trovati 366 prodotti di "Ricettore GABA"

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  • rac-BHFF

    CAS:
    rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.
    Formula:C17H21F3O3
    Purezza:99.69% - >99.99%
    Colore e forma:Solid
    Peso molecolare:330.34

    Ref: TM-T4176

    2mg
    43,00€
    5mg
    60,00€
    10mg
    96,00€
    25mg
    187,00€
    50mg
    311,00€
    100mg
    472,00€
    200mg
    657,00€
    1mL*10mM (DMSO)
    71,00€
  • Loreclezole hydrochloride

    CAS:
    Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.
    Formula:C10H7Cl4N3
    Colore e forma:Solid
    Peso molecolare:310.99

    Ref: TM-T39708

    10mg
    919,00€
    50mg
    3.771,00€
  • 6-Aminonicotinic acid

    CAS:
    <p>6-Aminonicotinic acid is a natural product.</p>
    Formula:C6H6N2O2
    Purezza:99.94%
    Colore e forma:Soild
    Peso molecolare:138.1238

    Ref: TM-T7919

    1g
    34,00€
  • Tiagabine

    CAS:
    Tiagabine (NO050328) is an Anti-epileptic Agent.
    Formula:C20H25NO2S2
    Purezza:99.25% - 99.67%
    Colore e forma:White To Off-White Crystalline Solid
    Peso molecolare:375.55

    Ref: TM-T2407

    5mg
    44,00€
    10mg
    55,00€
    25mg
    86,00€
    50mg
    131,00€
    1mL*10mM (DMSO)
    56,00€
  • Guvacine hydrochloride

    CAS:
    Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)
    Formula:C6H10ClNO2
    Purezza:98.42%
    Colore e forma:Solid
    Peso molecolare:163.602

    Ref: TM-T7557

    10mg
    39,00€
    25mg
    60,00€
    50mg
    88,00€
    100mg
    101,00€
  • L-DABA

    CAS:
    L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).
    Formula:C4H10N2O2
    Purezza:99.32%
    Colore e forma:Solid
    Peso molecolare:118.13

    Ref: TM-T7595

    25mg
    34,00€
  • Amentoflavone

    CAS:
    Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.
    Formula:C30H18O10
    Purezza:98.21% - 99.22%
    Colore e forma:Odourless Whitish Solid
    Peso molecolare:538.46

    Ref: TM-T3417

    2mg
    35,00€
    5mg
    52,00€
    10mg
    85,00€
    25mg
    133,00€
    50mg
    227,00€
    100mg
    369,00€
    200mg
    540,00€
    1mL*10mM (DMSO)
    63,00€
  • CGP52432

    CAS:
    CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).
    Formula:C15H24Cl2NO4P
    Purezza:98.75%
    Colore e forma:Solid
    Peso molecolare:384.24

    Ref: TM-T4363

    1mg
    40,00€
    5mg
    87,00€
    10mg
    140,00€
    25mg
    255,00€
    50mg
    374,00€
    1mL*10mM (DMSO)
    96,00€
  • Aminooxyacetic acid hemihydrochloride

    CAS:
    Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA
    Formula:C2H5NO3·5HCl
    Purezza:98.03%
    Colore e forma:Light Beige Crystalline Powder
    Peso molecolare:109.3

    Ref: TM-T5880

    1g
    74,00€
    2g
    96,00€
    5g
    157,00€
    200mg
    35,00€
    500mg
    48,00€
    1mL*10mM (DMSO)
    49,00€
  • Cyclothiazide

    CAS:
    Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).
    Formula:C14H16ClN3O4S2
    Purezza:98.23% - 99.49%
    Colore e forma:Crystals From Dilute Alcohol Solid
    Peso molecolare:389.88

    Ref: TM-T4573

    5mg
    52,00€
    10mg
    80,00€
    25mg
    144,00€
    50mg
    235,00€
    100mg
    349,00€
    200mg
    515,00€
    1mL*10mM (DMSO)
    58,00€
  • Acamprosate calcium

    CAS:
    Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.
    Formula:C10H20CaN2O8S2
    Purezza:98% - 99.93%
    Colore e forma:White Odorless Or Nearly Odorless Powder
    Peso molecolare:400.48

    Ref: TM-T1673

    1ml
    47,00€
    50mg
    48,00€
  • SSD114 HCl

    CAS:
    SSD114 is a novel GABAB receptor positive allosteric modulator.
    Formula:C18H21ClF3N3O
    Purezza:99.03% - 99.95%
    Colore e forma:Solid
    Peso molecolare:387.83

    Ref: TM-T4522

    2mg
    34,00€
    5mg
    50,00€
    10mg
    75,00€
    25mg
    111,00€
    50mg
    172,00€
    100mg
    290,00€
    200mg
    419,00€
    1mL*10mM (DMSO)
    46,00€
  • p-Hydroxybenzaldehyde

    CAS:
    1.
    Formula:C7H6O2
    Purezza:99.05% - 99.86%
    Colore e forma:Solid
    Peso molecolare:122.12

    Ref: TM-T2S1814

    10g
    37,00€
    25g
    48,00€
    1mL*10mM (DMSO)
    33,00€
  • 2'-O-Methylisoliquiritigenin

    CAS:
    2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-
    Formula:C16H14O4
    Purezza:98.75%
    Colore e forma:Solid
    Peso molecolare:270.28

    Ref: TM-TN1217

    1mg
    115,00€
    5mg
    274,00€
    10mg
    455,00€
    25mg
    730,00€
    50mg
    Prezzo su richiesta
    1mL*10mM (DMSO)
    378,00€
  • Ginsenoside Rc

    CAS:
    <p>Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.</p>
    Formula:C53H90O22
    Purezza:98.83% - 99.56%
    Colore e forma:White Powder
    Peso molecolare:1079.27

    Ref: TM-T2720

    5mg
    48,00€
    10mg
    70,00€
    25mg
    120,00€
    50mg
    170,00€
    100mg
    255,00€
    200mg
    379,00€
  • Darigabat

    CAS:
    Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.
    Formula:C22H21FN4O3S
    Purezza:98.42% - 99.29%
    Colore e forma:Solid
    Peso molecolare:440.49

    Ref: TM-T16489

    1mg
    54,00€
  • Riluzole

    CAS:
    <p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>
    Formula:C8H5F3N2OS
    Purezza:99.71% - 99.88%
    Colore e forma:Powder
    Peso molecolare:234.2

    Ref: TM-T0349

    1g
    155,00€
    25mg
    39,00€
    50mg
    49,00€
    100mg
    64,00€
    500mg
    115,00€
  • CGP 36216 hydrochloride

    CAS:
    CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).
    Formula:C5H14NO2P
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:151.14

    Ref: TM-T22647

    25mg
    Prezzo su richiesta
    50mg
    Prezzo su richiesta
    100mg
    Prezzo su richiesta
  • MK-0343

    CAS:
    MK0343 is an orally bioavailable GABAA receptor subtype-selective partial agonist and is a non-sedating anxiolytic.
    Formula:C19H17F2N7O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:397.38

    Ref: TM-T16084

    2mg
    187,00€
    25mg
    1.045,00€
    50mg
    1.369,00€
    100mg
    2.072,00€
  • GABA-AT-IN-1

    CAS:
    GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.
    Formula:C23H18N2O6
    Colore e forma:Solid
    Peso molecolare:418.4

    Ref: TM-T62185

    25mg
    2.033,00€
    50mg
    2.645,00€
    100mg
    3.345,00€