
Ricettore GABA
I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.
Trovati 366 prodotti di "Ricettore GABA"
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rac-BHFF
CAS:rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.Formula:C17H21F3O3Purezza:99.69% - >99.99%Colore e forma:SolidPeso molecolare:330.34Ref: TM-T4176
2mg43,00€5mg60,00€10mg96,00€25mg187,00€50mg311,00€100mg472,00€200mg657,00€1mL*10mM (DMSO)71,00€Loreclezole hydrochloride
CAS:Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.Formula:C10H7Cl4N3Colore e forma:SolidPeso molecolare:310.996-Aminonicotinic acid
CAS:<p>6-Aminonicotinic acid is a natural product.</p>Formula:C6H6N2O2Purezza:99.94%Colore e forma:SoildPeso molecolare:138.1238Tiagabine
CAS:Tiagabine (NO050328) is an Anti-epileptic Agent.Formula:C20H25NO2S2Purezza:99.25% - 99.67%Colore e forma:White To Off-White Crystalline SolidPeso molecolare:375.55Guvacine hydrochloride
CAS:Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)Formula:C6H10ClNO2Purezza:98.42%Colore e forma:SolidPeso molecolare:163.602L-DABA
CAS:L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).Formula:C4H10N2O2Purezza:99.32%Colore e forma:SolidPeso molecolare:118.13Amentoflavone
CAS:Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.Formula:C30H18O10Purezza:98.21% - 99.22%Colore e forma:Odourless Whitish SolidPeso molecolare:538.46Ref: TM-T3417
2mg35,00€5mg52,00€10mg85,00€25mg133,00€50mg227,00€100mg369,00€200mg540,00€1mL*10mM (DMSO)63,00€CGP52432
CAS:CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).Formula:C15H24Cl2NO4PPurezza:98.75%Colore e forma:SolidPeso molecolare:384.24Aminooxyacetic acid hemihydrochloride
CAS:Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABAFormula:C2H5NO3·5HClPurezza:98.03%Colore e forma:Light Beige Crystalline PowderPeso molecolare:109.3Cyclothiazide
CAS:Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).Formula:C14H16ClN3O4S2Purezza:98.23% - 99.49%Colore e forma:Crystals From Dilute Alcohol SolidPeso molecolare:389.88Acamprosate calcium
CAS:Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.Formula:C10H20CaN2O8S2Purezza:98% - 99.93%Colore e forma:White Odorless Or Nearly Odorless PowderPeso molecolare:400.48SSD114 HCl
CAS:SSD114 is a novel GABAB receptor positive allosteric modulator.Formula:C18H21ClF3N3OPurezza:99.03% - 99.95%Colore e forma:SolidPeso molecolare:387.83Ref: TM-T4522
2mg34,00€5mg50,00€10mg75,00€25mg111,00€50mg172,00€100mg290,00€200mg419,00€1mL*10mM (DMSO)46,00€p-Hydroxybenzaldehyde
CAS:1.Formula:C7H6O2Purezza:99.05% - 99.86%Colore e forma:SolidPeso molecolare:122.122'-O-Methylisoliquiritigenin
CAS:2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-Formula:C16H14O4Purezza:98.75%Colore e forma:SolidPeso molecolare:270.28Ref: TM-TN1217
1mg115,00€5mg274,00€10mg455,00€25mg730,00€50mgPrezzo su richiesta1mL*10mM (DMSO)378,00€Ginsenoside Rc
CAS:<p>Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.</p>Formula:C53H90O22Purezza:98.83% - 99.56%Colore e forma:White PowderPeso molecolare:1079.27Darigabat
CAS:Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.Formula:C22H21FN4O3SPurezza:98.42% - 99.29%Colore e forma:SolidPeso molecolare:440.49Riluzole
CAS:<p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>Formula:C8H5F3N2OSPurezza:99.71% - 99.88%Colore e forma:PowderPeso molecolare:234.2CGP 36216 hydrochloride
CAS:CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).Formula:C5H14NO2PPurezza:98%Colore e forma:SolidPeso molecolare:151.14MK-0343
CAS:MK0343 is an orally bioavailable GABAA receptor subtype-selective partial agonist and is a non-sedating anxiolytic.Formula:C19H17F2N7OPurezza:98%Colore e forma:SolidPeso molecolare:397.38GABA-AT-IN-1
CAS:GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.Formula:C23H18N2O6Colore e forma:SolidPeso molecolare:418.4
