Ricettore GABA
I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.
Trovati 369 prodotti di "Ricettore GABA"
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TP003
CAS:TP003 is a novel non-selective GABAA receptor benzodiazepine site agonist with affinity for α1β2gam2, α2β3gam2, α3β3gam2, α5β2gam2, EC50 of 20.3, 10.6, 3.24, 5.
Formula:C23H16F3N3OPurezza:99.17%Colore e forma:SolidPeso molecolare:407.39β-CCM
CAS:β-CCM is a benzodiazepine receptor inverse agonist with anxiogenic and convulsant effects. It enhances emotional reactivity and reduces interference sensitivity in spatial working memory tasks. β-CCM is applicable in research related to anxiety disorders.Formula:C13H10N2O2Colore e forma:SolidPeso molecolare:226.231Gabaculine HCl
CAS:Gabaculine, an irreversible GABA-T inhibitor (Ki: 2.9 μM), impacts plastid development and affects DPOR/GluTR levels.Formula:C7H10ClNO2Colore e forma:SolidPeso molecolare:175.61S-8510 phosphate
CAS:S-8510 phosphate is an agonist of inverse Benzodiazepine (BDZ) receptor(Kis of 34.6 nM, 36.2 nM for –GABA and +GABA respectively).Formula:C12H13N4O6PPurezza:98%Colore e forma:SolidPeso molecolare:340.23Fletazepam
CAS:Fletazepam, a benzodiazepine derivative, exhibits sedative, anti-anxiety, and muscle-relaxant properties. It is utilized in neurological research.Formula:C17H13ClF4N2Colore e forma:SolidPeso molecolare:356.74EF1502 free base
CAS:EF1502 is a potent and selective GABA transporter inhibitor.Formula:C22H26N2O2S2Purezza:98%Colore e forma:SolidPeso molecolare:414.58GABAA receptor agonist 1
Compound 3e, a potent GABAA agonist, targets GABA sites and has potential anti-depressive effects in mice.Formula:C20H30O3Colore e forma:SolidPeso molecolare:318.45Moxetomidate
CAS:Moxetomidate is a GABAA receptor (GABAA receptor) agonist with hypnotic properties.
Formula:C15H18N2O3Colore e forma:SolidPeso molecolare:274.315Cyproflanilide
CAS:Cyproflanilide is a GABAR antagonist that exhibits high activity against a variety of pests, including those from the Lepidoptera, Coleoptera, and Thysanoptera orders.Formula:C28H17BrF12N2O2Colore e forma:SolidPeso molecolare:721.33BGT1-IN-1
CAS:BGT1-IN-1 (compound 9) is an effective inhibitor of BGT1, demonstrating IC50 values of 13.9 µM for hBGT1 and 58.3 µM for GAT3. It exhibits no cytotoxic effects and possesses neuroprotective activity.Formula:C6H9NO2Colore e forma:SolidPeso molecolare:127.14(-)-Bicuculline methobromide
CAS:(-)-Bicuculline methobromide is a potent antagonist of GABAA receptor .Formula:C21H20BrNO6Colore e forma:WhitePeso molecolare:462.29Alfadolone acetate
CAS:Alfadolone acetate is a gamma-aminobutyric acid (GABA) receptor agonist.Formula:C23H34O5Colore e forma:SolidPeso molecolare:390.512-AEMP TFA
CAS:2-AEMP TFA is a potent and rapidly acting antagonist of GABA(A)-ρ1 receptors. 2-AEMP is an analog of GABA.Formula:C3H10NO3PPurezza:98%Colore e forma:SolidPeso molecolare:139.0913-Methylglutaconic acid
CAS:3-Methylglutaconic acid, a primary metabolite accumulating in 3-Methylglutaconic aciduria (MGTA), induces lipid and protein oxidation, while diminishing non-enzymatic antioxidant defenses in cerebral cortex supernatants, thereby promoting oxidative stress in the cerebral cortex. This compound is utilized in research concerning brain damage diseases [1].Formula:C6H8O4Purezza:98%Colore e forma:SolidPeso molecolare:144.13Pazinaclone
CAS:Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.Formula:C25H23ClN4O4Purezza:97.79% - 98.65%Colore e forma:SolidPeso molecolare:478.93CGP 44532
CAS:CGP 44532 a GABAB receptor agonist.Formula:C4H12NO3PPurezza:98%Colore e forma:SolidPeso molecolare:153.12Ref: TM-T26991
Prodotto fuori produzionePipequaline
CAS:Pipequaline (PK-8165) is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It possesses a novel chemical structure that is not closely related to other drugs of this type. The drug has a similar pharmacological profile to the benzodiazepine family of drugs, but with mainly anxiolytic properties and very little sedative, amnestic or anticonvulsant effects, and so is classified as a nonbenzodiazepine anxiolytic.Formula:C22H24N2Purezza:98%Colore e forma:SolidPeso molecolare:316.44CGP 56999A
CAS:CGP 56999A is a GABA(B) receptor antagonist; it boosts BDNF and reduces dopamine loss in rat striatum.Formula:C19H30NO5PPurezza:98%Colore e forma:SolidPeso molecolare:383.42Ref: TM-T26993
Prodotto fuori produzioneXilmenolone
CAS:Xilmenolone acts as a positive allosteric modulator of the GABA_A receptor [1].
Formula:C26H37N3O2Purezza:98%Colore e forma:SolidPeso molecolare:423.59Ref: TM-T78670
Prodotto fuori produzione
