Ricettore GABA
I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.
Trovati 365 prodotti di "Ricettore GABA"
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Ro 22-8515
CAS:Ro 22-8515 is the ligand of benzodiazepine receptor.Formula:C18H12Cl2N2OColore e forma:SolidPeso molecolare:343.21Ro15-4513
CAS:Ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. Ro15-4513 is an effective ethanol antagonist.Formula:C15H14N6O3Purezza:98%Colore e forma:SolidPeso molecolare:326.31ZK-91296
CAS:ZK-91296: GABA agonist, lowers anxiety without sedation, may target specific BZ receptor subtype.Formula:C23H22N2O4Purezza:98%Colore e forma:SolidPeso molecolare:390.432-Hydroxysaclofen
CAS:2-Hydroxysaclofen is a GABAB receptor antagonist.Formula:C9H12ClNO4SPurezza:98%Colore e forma:White SolidPeso molecolare:265.71SCH-50910 free base
CAS:SCH-50910 is an antagonist of GABAB receptor.Formula:C8H15NO3Colore e forma:SolidPeso molecolare:173.21CGS 20625
CAS:partial agonist for the benzodiazepine binding site of the GABAA receptorFormula:C18H19N3O2Purezza:99.61%Colore e forma:SolidPeso molecolare:309.36Profadol hydrochloride
CAS:Profadol hydrochloride acts as a mixed agonist-antagonist of the μ-opioid receptor with analgesic activity.Formula:C14H22ClNOPurezza:98%Colore e forma:SolidPeso molecolare:255.78SX-3228
CAS:SX-3228 is a selective agonist of benzodiazepine1 (BZ1) receptor(IC50 of 17 nM).Formula:C18H18N4O3Purezza:98%Colore e forma:SolidPeso molecolare:338.36Ro 14-7437
CAS:Ro 14-7437 is an antagonist of GABA-benzodiazepine receptor.Formula:C15H15N3O3Colore e forma:SolidPeso molecolare:285.3Adinazolam Mesylate
CAS:Adinazolam Mesylate is an anxiolytic and antidepressant agent. Adinazolam Mesylate binds to peripheral-type benzodiazepine receptors that interact allosterically with GABA receptors as an agonist to produce inhibitory effects.Formula:C20H22ClN5O3SPurezza:98%Colore e forma:SolidPeso molecolare:447.94Ro 15-1310
CAS:Ro 15-3505, a benzodiazepine receptor partial inverse agonist, has shown the ability to improve impaired recent memory of aged mice.Formula:C15H14ClN3O3Colore e forma:SolidPeso molecolare:319.74CP-457920
CAS:CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.Formula:C18H17N3O3Purezza:99.06% - 99.74%Colore e forma:SolidPeso molecolare:323.35Org 20599
CAS:GABAA receptor agonistFormula:C25H40ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:438.04U-101017
CAS:U-101017 is a partial benzodiazepine receptor and GABAA receptor agonist.Formula:C23H27ClN4O3Purezza:98%Colore e forma:SolidPeso molecolare:442.94TPA-023B
CAS:TPA-023B: oral GABAA α2/α3 agonist (Kis: 0.73/2 nM), α1 antagonist (Ki: 1.8 nM), non-sedating anxiolytic.Formula:C21H15F2N5OPurezza:98%Colore e forma:SolidPeso molecolare:391.37CGP 7930
CAS:Positive allosteric modulator of GABAB receptorsFormula:C19H32O2Purezza:98%Colore e forma:SolidPeso molecolare:292.46BHF-177
CAS:BHF-177 is a positive allosteric modulator of the GABAB receptor. BHF-177 reduces self-administration of nicotine in animal studies.Formula:C19H20F3N3Colore e forma:SolidPeso molecolare:347.38CGS8216
CAS:CGS8216 shows analgesic activity at high doses, has anxiolytic activity, and can be used to study immune system disorders.Formula:C16H11N3OPurezza:98.53%Colore e forma:SolidPeso molecolare:261.28SCH 50911 hydrochloride
CAS:SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).Formula:C8H16ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:209.67DS2
CAS:Positive allosteric modulator of δ-subunit containing GABAA receptorsFormula:C18H12ClN3OSPurezza:98%Colore e forma:SolidPeso molecolare:353.83(±)-Homoproline Hydrochloride
CAS:(±)-Homoproline Hydrochloride. Affordable Excellence: Reliable Quality You Can TrustFormula:C6H12ClNO2Purezza:99.69%Colore e forma:SolidPeso molecolare:165.62MK-0343
CAS:MK0343 is an orally bioavailable GABAA receptor subtype-selective partial agonist and is a non-sedating anxiolytic.Formula:C19H17F2N7OPurezza:98%Colore e forma:SolidPeso molecolare:397.3817-PA
CAS:17-PA is a GABAA receptor antagonist.Formula:C25H34OPurezza:98%Colore e forma:SolidPeso molecolare:350.54Bifenazate
CAS:Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.Formula:C17H20N2O3Purezza:99.62%Colore e forma:Solid CrystallinePeso molecolare:300.35CGP11952
CAS:CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.Formula:C21H21Cl2N5O2Purezza:98%Colore e forma:SolidPeso molecolare:446.33E2730
CAS:E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.Formula:C9H8F4N2O2SPurezza:98.22% - 98.54%Colore e forma:SolidPeso molecolare:284.23U-89843A
CAS:U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].Formula:C16H24ClN5Purezza:98%Colore e forma:SolidPeso molecolare:321.85(R)-Baclofen hydrochloride
CAS:Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.Formula:C10H13Cl2NO2Purezza:98%Colore e forma:SolidPeso molecolare:250.12NO 711
CAS:NO 711（NNC-711 free acid） is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.Formula:C21H22N2O3Purezza:99.70%Colore e forma:SolidPeso molecolare:350.41AZD 3043
CAS:AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.Formula:C19H29NO5Purezza:98.19% - 99.55%Colore e forma:SolidPeso molecolare:351.44mGAT3/4-IN-1
CAS:mGAT3/4-IN-1 inhibits mGAT3/4 with pIC50: 5.31/5.24, reduces neuropathic pain in diabetic mice.Formula:C26H31ClN2O2S2Colore e forma:SolidPeso molecolare:503.12GABAA receptor agent 4
CAS:<p>Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.</p>Formula:C17H24N2OColore e forma:SolidPeso molecolare:272.39Ro 19-4603
CAS:Benzodiazepine inverse agonistFormula:C15H17N3O3SPurezza:98%Colore e forma:SolidPeso molecolare:319.38TG41
CAS:TG41 is a GABAA receptors positive modulator.Formula:C18H13BrCl2N2O2Purezza:98%Colore e forma:SolidPeso molecolare:440.12FG8119
CAS:FG8119 is a novel benzodiazepine agonist with potential anticonvulsant and antiepileptic activity for the study of neurological disorders.Formula:C17H15N5O2Purezza:>99.99%Colore e forma:SolidPeso molecolare:321.33GABAA receptor agent 6
CAS:GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with low cellular membrane permeability (Ki = 0.56 μM) [1].Formula:C18H25N3O2Colore e forma:SolidPeso molecolare:315.41TB 21007
CAS:GABAA receptor inverse agonistFormula:C15H17NO2S3Purezza:98%Colore e forma:SolidPeso molecolare:339.5SL-651498
CAS:SL-651498, a GABAA receptor agonist, is used potentially for the treatment of anxiety.Formula:C23H20FN3O2Purezza:98%Colore e forma:SolidPeso molecolare:389.42Bamaluzole
CAS:Bamaluzole is an agonist of GABA receptor.Formula:C14H12ClN3OPurezza:98%Colore e forma:SolidPeso molecolare:273.72ZAPA sulfate
CAS:GABAA receptors agonistFormula:C4H8N2O6S2Purezza:98%Colore e forma:SolidPeso molecolare:244.25Lesogaberan
CAS:Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity (Ki 1.4 μM).Formula:C3H9FNO2PPurezza:98%Colore e forma:SolidPeso molecolare:141.08NAP-1
CAS:NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).Formula:C20H18ClNO2Colore e forma:SolidPeso molecolare:339.82GABAA receptor agent 7
CAS:Compound 5c, a GABAA receptor modulator with anticonvulsant properties and low neurotoxicity, is promising for epilepsy research.Formula:C18H13ClN4OColore e forma:SolidPeso molecolare:336.77MRK-623
CAS:MRK-623 (14k) is an oral GABA A agonist with high affinity for α1/α2/α3/α5 subunits and anxiolytic properties.Formula:C20H17FN4OColore e forma:SolidPeso molecolare:348.37GABAA receptor agent 8
CAS:Compound 5e, a GABAA receptor modulator, shows potent anticonvulsant effects with low neurotoxicity for epilepsy research.Formula:C19H16N4OColore e forma:SolidPeso molecolare:316.36Etbicyphat
CAS:Etbicyphat: potent GABA(A) antagonist, induces epileptiform activity, binds to GABA/benzodiazepine receptors.Formula:C6H11O4PColore e forma:SolidPeso molecolare:178.12NCS-382
CAS:γ-Hydroxybutyric acid antagonistFormula:C13H14O3Purezza:98%Colore e forma:SolidPeso molecolare:218.25TCS 1105
CAS:TCS 1105 is a GABAA BZR ligand, blocking Sema3A and altering mouse anxiety, aggression, and social dominance.Formula:C17H13FN2O2Purezza:99.75%Colore e forma:SolidPeso molecolare:296.3
