
Ricettore GABA
I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.
Trovati 365 prodotti di "Ricettore GABA"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
NAP-1
CAS:NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).Formula:C20H18ClNO2Colore e forma:SolidPeso molecolare:339.82Bamaluzole
CAS:Bamaluzole is an agonist of GABA receptor.Formula:C14H12ClN3OPurezza:98%Colore e forma:SolidPeso molecolare:273.72PNU-107484A
CAS:PNU-107484A is a unique GABA(A) receptor ligand.Formula:C18H23ClN6Purezza:98%Colore e forma:SolidPeso molecolare:358.87SL-651498
CAS:SL-651498, a GABAA receptor agonist, is used potentially for the treatment of anxiety.Formula:C23H20FN3O2Purezza:98%Colore e forma:SolidPeso molecolare:389.42TB 21007
CAS:GABAA receptor inverse agonistFormula:C15H17NO2S3Purezza:98%Colore e forma:SolidPeso molecolare:339.5GABAA receptor agent 6
CAS:GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with low cellular membrane permeability (Ki = 0.56 μM) [1].Formula:C18H25N3O2Colore e forma:SolidPeso molecolare:315.41(S)-SNAP5114
CAS:<p>(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.</p>Formula:C30H35NO6Purezza:97%Colore e forma:SolidPeso molecolare:505.6GS 39783
CAS:GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement andFormula:C15H23N5O2SPurezza:99.92%Colore e forma:SolidPeso molecolare:337.44FG8119
CAS:FG8119 is a novel benzodiazepine agonist with potential anticonvulsant and antiepileptic activity for the study of neurological disorders.Formula:C17H15N5O2Purezza:>99.99%Colore e forma:SolidPeso molecolare:321.33TG41
CAS:TG41 is a GABAA receptors positive modulator.Formula:C18H13BrCl2N2O2Purezza:98%Colore e forma:SolidPeso molecolare:440.12SCH 50911
CAS:SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.Formula:C8H15NO3Purezza:98%Colore e forma:SolidPeso molecolare:173.21Anxiolytic/nonsedative agent-1
CAS:TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.Formula:C18H15N3O4Purezza:98.61%Colore e forma:SolidPeso molecolare:337.33Radequinil
CAS:<p>Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).</p>Formula:C18H14N4O3Purezza:98%Colore e forma:SolidPeso molecolare:334.33Ciclotizolam
CAS:Ciclotizolam, a thienotriazolodiazepine derivative and partial GABAA receptor agonist, has low efficacy but similar affinity as brotizolam.Formula:C20H18BrClN4SColore e forma:SolidPeso molecolare:461.81ZAPA sulfate
CAS:GABAA receptors agonistFormula:C4H8N2O6S2Purezza:98%Colore e forma:SolidPeso molecolare:244.25GABAA receptor agent 8
CAS:Compound 5e, a GABAA receptor modulator, shows potent anticonvulsant effects with low neurotoxicity for epilepsy research.Formula:C19H16N4OColore e forma:SolidPeso molecolare:316.36AZD 3043
CAS:AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.Formula:C19H29NO5Purezza:98.19% - 99.55%Colore e forma:SolidPeso molecolare:351.44SH-053-S-CH3-2'F
CAS:SH-053-S-CH3-2'F is a potent and selective agonist of GABAA receptors.Formula:C23H18FN3O2Colore e forma:SolidPeso molecolare:387.41(+)-Nipecotic acid
CAS:(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.Formula:C6H11NO2Purezza:99.38%Colore e forma:SolidPeso molecolare:129.16
