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Ricettore GABA

Ricettore GABA

I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.

Trovati 365 prodotti di "Ricettore GABA"

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  • GABA-IN-2
    Targetmol
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    GABA-IN-2

    CAS:
    GABA-IN-2 (Compound 5), a GABA inhibitor, exhibits both larvicidal and insecticidal properties, achieving an 87% mortality rate at a concentration of 50 mg/L [1
    Formula:C12H4Cl2F6N4Se
    Colore e forma:Solid
    Peso molecolare:468.04

    Ref: TM-T82355

  • TPA 023
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    TPA 023

    CAS:
    <p>TPA 023 is a selective agonist of GABAA α2/α3 subtype (Kis = 0.19 - 0.41 nM).</p>
    Formula:C20H22FN7O
    Purezza:99.75%
    Colore e forma:Solid
    Peso molecolare:395.43

    Ref: TM-T17144

  • CGP 55845
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    CGP 55845

    CAS:
    CGP 55845: potent, selective GABAB blocker, IC50=5 nM, hinders agonist binding, reduces GABA/glutamate release.
    Formula:C18H22Cl2NO3P
    Colore e forma:Solid
    Peso molecolare:402.25

    Ref: TM-T70531

  • CGP-54626 free base
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    CGP-54626 free base

    CAS:
    CGP-54626 is a selective antagonist of the GABAB receptor (IC50 = 4 nM ).
    Formula:C18H28Cl2NO3P
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:408.3

    Ref: TM-T26998

  • Afizagabar
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    Afizagabar

    CAS:
    Afizagabar, a first-in-class α5-GABAAR antagonist, IC50: 585 nM, Ki: 66 nM, may boost memory.
    Formula:C19H12FN3O2S
    Colore e forma:Solid
    Peso molecolare:365.38

    Ref: TM-T37388

  • mGAT-IN-1
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    mGAT-IN-1

    CAS:
    mGAT-IN-1 is a potent, non-selective GAT inhibitor that inhibits mGAT3 activity well (IC50: 2.5 μM, pIC50: 5.61).
    Formula:C28H34ClN3O2S2
    Colore e forma:Solid
    Peso molecolare:544.17

    Ref: TM-T63832

  • CGP 54626 hydrochloride
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    CGP 54626 hydrochloride

    CAS:
    CGP 54626 hydrochloride is a GABAB receptor antagonist.
    Formula:C18H29Cl3NO3P
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:444.76

    Ref: TM-T22651

  • Piperidine-4-sulfonic acid
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    Piperidine-4-sulfonic acid

    CAS:
    Piperidine-4-sulfonic acid is a potent GABA agonist, demonstrating an IC50 value of 0.034 μM for the inhibition of H-GABA binding [1].
    Formula:C5H11NO3S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:165.21

    Ref: TM-T78642

  • SCS
    Targetmol
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    SCS

    CAS:
    SCS is a GABAA receptor antagonist.
    Formula:C14H12N2O3
    Purezza:99.73%
    Colore e forma:Solid
    Peso molecolare:256.26

    Ref: TM-T23339

  • CGP36216 hydrochloride
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    CGP36216 hydrochloride

    CAS:
    CGP36216 hydrochloride acts as a selective antagonist at the presynaptic GABA receptor, specifically binding to the GABAB receptor with a Ki value of 0.3 μM. This compound is leveraged in research focused on anxiety and trauma-related disorders [1] [2].
    Formula:C5H15ClNO2P
    Colore e forma:Solid
    Peso molecolare:187.6

    Ref: TM-T84878

  • NO-711ME
    Targetmol
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    NO-711ME

    CAS:
    NO-711ME (N-O711 Methyl ester) is a prodrug of NO-711. It also is a potent and selective GABA uptake inhibitor.
    Formula:C22H24N2O3
    Purezza:99.54%
    Colore e forma:Solid
    Peso molecolare:364.44

    Ref: TM-T24540

  • U 89843A
    Targetmol
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    U 89843A

    CAS:
    <p>U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.</p>
    Formula:C16H23N5
    Purezza:99.62%
    Colore e forma:Solid
    Peso molecolare:285.39

    Ref: TM-T23481

  • PZ-II-029
    Targetmol
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    PZ-II-029

    CAS:
    <p>PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.</p>
    Formula:C18H15N3O3
    Purezza:99.79%
    Colore e forma:Solid
    Peso molecolare:321.33

    Ref: TM-T28479

  • (-)-Bicuculline methochloride
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    (-)-Bicuculline methochloride

    CAS:
    <p>(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.</p>
    Formula:C21H20ClNO6
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:417.84

    Ref: TM-T12044

  • L 663581
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    L 663581

    CAS:
    L 663581 is the benzodiazepine receptor partial agonist.
    Formula:C17H16ClN5O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:357.79

    Ref: TM-T24317

  • 6,2'-Dihydroxyflavone
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    6,2'-Dihydroxyflavone

    CAS:
    6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.
    Formula:C15H10O4
    Purezza:99.44% - 99.67%
    Colore e forma:Solid
    Peso molecolare:254.24

    Ref: TM-T8268

  • NCS-382 sodium
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    NCS-382 sodium

    CAS:
    NCS-382 (sodium) is a potent antagonist of the GABA receptor, exhibiting anti-sedative and anti-hypnotic properties, with applications in neurological disease
    Formula:C13H13NaO3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:240.23

    Ref: TM-T78111

  • COR659
    Targetmol
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    COR659

    CAS:
    COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.
    Formula:C16H16ClNO3S
    Purezza:99.75%
    Colore e forma:Solid
    Peso molecolare:337.82

    Ref: TM-T36520

  • Logo CymitQuimica
    Targetmol
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    GABAA receptor agonist 2

    Compound 4c, a potent GABAA agonist with anti-depressive effects in mouse FST/TST, shows promise in depression research.
    Formula:C22H36O5
    Colore e forma:Solid
    Peso molecolare:380.52

    Ref: TM-T61625

  • SGE-516
    Targetmol
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    SGE-516

    CAS:
    <p>SGE516: neuroactive steroid, enhances GABAA, lowers neuronal activity, protects from seizures.</p>
    Formula:C23H35N3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:385.54

    Ref: TM-T28766