
Ricettore GABA
I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.
Trovati 365 prodotti di "Ricettore GABA"
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Pipequaline hydrochloride
CAS:<p>Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative.</p>Formula:C22H25ClN2Purezza:99.46%Colore e forma:SolidPeso molecolare:352.9Gabazine free base
CAS:Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.Formula:C15H17N3O3Colore e forma:SolidPeso molecolare:287.31p-Hydroxybenzaldehyde
CAS:1.Formula:C7H6O2Purezza:99.05% - 99.86%Colore e forma:SolidPeso molecolare:122.12Piperazine citrate
CAS:<p>Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.</p>Formula:C24H46N6O14Purezza:99.8%Colore e forma:Crystals IndicationPeso molecolare:642.65Baclofen hydrochloride
CAS:Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.Formula:C10H13Cl2NO2Purezza:99.55%Colore e forma:SolidPeso molecolare:250.122(-)-Securinine
CAS:(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.Formula:C13H15NO2Purezza:99.58% - 99.87%Colore e forma:SolidPeso molecolare:217.26(2S)-6-Prenylnaringenin
CAS:(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.Formula:C20H20O5Purezza:99.47%Colore e forma:SolidPeso molecolare:340.37SSD114 HCl
CAS:<p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>Formula:C18H21ClF3N3OPurezza:99.03% - 99.95%Colore e forma:SolidPeso molecolare:387.83Aminooxyacetic acid hemihydrochloride
CAS:Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABAFormula:C2H5NO3·5HClPurezza:98.03%Colore e forma:Light Beige Crystalline PowderPeso molecolare:109.3Loreclezole hydrochloride
CAS:Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.Formula:C10H7Cl4N3Colore e forma:SolidPeso molecolare:310.99α-Thujone
CAS:α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.Formula:C10H16OPurezza:97.02% - 98.41%Colore e forma:Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)Peso molecolare:152.23Cholesterol myristate
CAS:<p>Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.</p>Formula:C41H72O2Purezza:99.65%Colore e forma:SolidPeso molecolare:597.01Fipronil
CAS:Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.Formula:C12H4Cl2F6N4OSPurezza:97.21%Colore e forma:Solid PowderPeso molecolare:437.15Acetoxyvalerensre
CAS:<p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>Formula:C17H24O4Purezza:98.22%Colore e forma:SolidPeso molecolare:292.37α-Asarone
CAS:alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.Formula:C12H16O3Purezza:99.64% - 99.64%Colore e forma:Monoclinic Needles From Water Monoclinic Needles From WaterPeso molecolare:208.25Tiagabine hydrochloride hydrate
CAS:Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.Formula:C20H28ClNO3S2Colore e forma:SolidPeso molecolare:430.02(+)-Kavain
CAS:(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.Formula:C14H14O3Purezza:97% - ≥95%Colore e forma:White Fine PowderPeso molecolare:230.26Cyclothiazide
CAS:<p>Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).</p>Formula:C14H16ClN3O4S2Purezza:98.23% - 99.49%Colore e forma:Crystals From Dilute Alcohol SolidPeso molecolare:389.88Pikamilone
CAS:Pikamilone (Picamilon) is an intelligent medicine.Formula:C10H12N2O3Purezza:99.38%Colore e forma:White Crystalline PowderPeso molecolare:208.21AZD-6280
CAS:AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.Formula:C20H22N4O3Purezza:98.99%Colore e forma:SolidPeso molecolare:366.41
