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Deidrogenasi

Deidrogenasi

Le deidrogenasi sono enzimi coinvolti nelle reazioni di ossidoriduzione delle vie metaboliche, svolgendo un ruolo centrale nella produzione di energia e nella respirazione cellulare. Questi enzimi sono cruciali per processi come il ciclo dell'acido citrico, la glicolisi e l'ossidazione degli acidi grassi. Gli inibitori delle deidrogenasi sono strumenti importanti nello studio delle malattie metaboliche, del cancro e dello stress ossidativo. Presso CymitQuimica, offriamo una selezione completa di inibitori delle deidrogenasi per supportare la tua ricerca in metabolismo, biologia del cancro e biochimica.

Trovati 300 prodotti di "Deidrogenasi"

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  • PfDHODH-IN-2

    CAS:
    PfDHODH-IN-2: powerful antimalarial, blocks PfDHODH (IC50: 1.11 μM), for malaria research.
    Formula:C13H12ClNO3S
    Purezza:98.9%
    Colore e forma:Solid
    Peso molecolare:297.76
  • R162

    CAS:
    R162 is an effective glutamate dehydrogenase 1 (GDH1) inhibitor.
    Formula:C17H12O3
    Purezza:96.21% - 98.15%
    Colore e forma:Solid
    Peso molecolare:264.28
  • L-Allylglycine

    CAS:
    L-Allylglycine is a potent inhibitor of the synthetic enzyme for GABA, glutamic acid decarboxylase.
    Formula:C5H9NO2
    Purezza:≥98%
    Colore e forma:White To Off-White Crystalline Powder
    Peso molecolare:115.13
  • Mutant IDH1-IN-1

    CAS:
    Mutant IDH1-IN-1 is a potent mutant IDH1 R132 h inhibitor with IC50 < 0.1 uM.
    Formula:C30H31FN4O2
    Purezza:99.49% - >99.99%
    Colore e forma:Solid
    Peso molecolare:498.59
  • BI-187004

    CAS:
    BI-187004 is an 11β-hydroxysteroid dehydrogenase 1 inhibitor.
    Formula:C21H18N4O
    Purezza:98.63%
    Colore e forma:Solid
    Peso molecolare:342.39
  • NCT-503

    CAS:
    <p>NCT-503 is a phosphoglycerate dehydrogenase (PHGDH) inhibitor with no activity against other dehydrogenases. NCT-503 has antitumor activity. Cost-effective and quality-assured.</p>
    Formula:C20H23F3N4S
    Purezza:98.91% - 99.84%
    Colore e forma:Solid
    Peso molecolare:408.48
  • Ivosidenib

    CAS:
    Ivosidenib (AG-120) is an oral IDH1 inhibitor targeting mutated IDH1 to reduce 2-hydroxyglutarate and hinder tumor growth.
    Formula:C28H22ClF3N6O3
    Purezza:98.71% - 99.98%
    Colore e forma:Solid
    Peso molecolare:582.96
  • Proguanil hydrochloride

    CAS:
    Proguanil hydrochloride, a biguanide, metabolizes into cycloguanil, an anti-malaria agent that inhibits plasmodium's DNA and protein synthesis.
    Formula:C11H17Cl2N5
    Purezza:98.34% - 98.39%
    Colore e forma:Solid
    Peso molecolare:290.19
  • BAY-1436032

    CAS:
    BAY-1436032 is a novel, selective and orally available inhibitor of pan-mutant isocitrate dehydrogenase 1 (IDH1).
    Formula:C26H30F3N3O3
    Purezza:99.65% - 99.71%
    Colore e forma:Solid
    Peso molecolare:489.53
  • Brequinar sodium

    CAS:
    Bipenquinate is a potent and selective inhibitor of dihydroorotate dehydrogenase (DHODH) with IC50 of 20 nM, blocking de novo pyrimidine biosynthesis.
    Formula:C23H14F2NNaO2
    Purezza:98.16%
    Colore e forma:Solid
    Peso molecolare:397.36
  • DS-1001b

    CAS:
    DS-1001b is an inhibitor of mutant IDH-1 (Isocitrate Dehydrogenase-1)
    Formula:C29H29Cl3FN3O4
    Purezza:99.81%
    Colore e forma:Solid
    Peso molecolare:608.92
  • Vidofludimus hemicalcium

    CAS:
    Vidofludimus hemicalcium: oral DHODH inhibitor, FXR modulator, for autoimmune and fatty liver research.
    Formula:C20H18FNO4Ca
    Colore e forma:Solid
    Peso molecolare:375.4
  • G6PDi-1

    CAS:
    <p>G6PDi-1 is an effective G6PD inhibitor. It depletes NADPH and decreases inflammatory cytokine production.</p>
    Formula:C14H12N4OS
    Purezza:98.69%
    Colore e forma:Solid
    Peso molecolare:284.34
  • AZD7545

    CAS:
    AZD7545 is a potent PDHK inhibitor.
    Formula:C19H18ClF3N2O5S
    Purezza:99.12% - 99.96%
    Colore e forma:Solid
    Peso molecolare:478.87
  • BMS-823778 hydrochloride

    CAS:
    <p>BMS-823778 hydrochloride is a potent, selective, and orally active inhibitor of 11β-HSD1 (11β-Hydroxysteroid Dehydrogenase Type 1), demonstrating an IC50 (half</p>
    Formula:C18H19Cl2N3O
    Colore e forma:Solid
    Peso molecolare:364.27
  • MK-8245

    CAS:
    MK-8245 is a liver-targeting SCD inhibitor for human SCD1 (IC50: 1 nM) and for rat/mouse SCD1 (IC50: 3 nM), with anti-diabetic and anti-dyslipidemic function.
    Formula:C17H16BrFN6O4
    Purezza:97.58% - 99%
    Colore e forma:Solid
    Peso molecolare:467.25
  • LDHA-IN-4

    CAS:
    LDHA-IN-4 (AZ33) is an LDHA inhibitor. Binding affinity to 6-His-tagged human LDHA expressed in E.coli BL21 (DE3) by SPR analysis with an active value of 93 nM.
    Formula:C25H27N3O6S
    Purezza:98.17% - 99.68%
    Colore e forma:Solid
    Peso molecolare:497.56
  • NCT-505

    CAS:
    NCT-505 is a potent and selective inhibitor of aldehyde dehydrogenase (ALDH1A1, IC50 = 7 nM) and a weak inhibitor of hALDH1A2, hALDH1A3, hALDH2, hALDH3A1 with
    Formula:C27H28FN5O3S
    Purezza:99.93%
    Colore e forma:Solid
    Peso molecolare:521.61
  • VER-246608

    CAS:
    VER-246608 inhibits PDK (IC50: 35-91 nM), boosts PDC, reduces glycolysis, causes cancer cell cytostasis, and enhances doxorubicin effects.
    Formula:C28H23ClF2N4O4
    Purezza:98.5%
    Colore e forma:Solid
    Peso molecolare:552.96
  • Nifurtimox

    CAS:
    Nifurtimox (BAY-A-2502) is an antiprotozoal agent (IC50s = 9.91, 12.28, and 10.44 μM against Taluahuén, LQ, and Brener strains of T.
    Formula:C10H13N3O5S
    Purezza:99.87% - 99.89%
    Colore e forma:Solid
    Peso molecolare:287.29