
Deidrogenasi
Le deidrogenasi sono enzimi coinvolti nelle reazioni di ossidoriduzione delle vie metaboliche, svolgendo un ruolo centrale nella produzione di energia e nella respirazione cellulare. Questi enzimi sono cruciali per processi come il ciclo dell'acido citrico, la glicolisi e l'ossidazione degli acidi grassi. Gli inibitori delle deidrogenasi sono strumenti importanti nello studio delle malattie metaboliche, del cancro e dello stress ossidativo. Presso CymitQuimica, offriamo una selezione completa di inibitori delle deidrogenasi per supportare la tua ricerca in metabolismo, biologia del cancro e biochimica.
Trovati 300 prodotti di "Deidrogenasi"
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PfDHODH-IN-2
CAS:PfDHODH-IN-2: powerful antimalarial, blocks PfDHODH (IC50: 1.11 μM), for malaria research.Formula:C13H12ClNO3SPurezza:98.9%Colore e forma:SolidPeso molecolare:297.76R162
CAS:R162 is an effective glutamate dehydrogenase 1 (GDH1) inhibitor.Formula:C17H12O3Purezza:96.21% - 98.15%Colore e forma:SolidPeso molecolare:264.28L-Allylglycine
CAS:L-Allylglycine is a potent inhibitor of the synthetic enzyme for GABA, glutamic acid decarboxylase.Formula:C5H9NO2Purezza:≥98%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:115.13Mutant IDH1-IN-1
CAS:Mutant IDH1-IN-1 is a potent mutant IDH1 R132 h inhibitor with IC50 < 0.1 uM.Formula:C30H31FN4O2Purezza:99.49% - >99.99%Colore e forma:SolidPeso molecolare:498.59BI-187004
CAS:BI-187004 is an 11β-hydroxysteroid dehydrogenase 1 inhibitor.Formula:C21H18N4OPurezza:98.63%Colore e forma:SolidPeso molecolare:342.39NCT-503
CAS:<p>NCT-503 is a phosphoglycerate dehydrogenase (PHGDH) inhibitor with no activity against other dehydrogenases. NCT-503 has antitumor activity. Cost-effective and quality-assured.</p>Formula:C20H23F3N4SPurezza:98.91% - 99.84%Colore e forma:SolidPeso molecolare:408.48Ivosidenib
CAS:Ivosidenib (AG-120) is an oral IDH1 inhibitor targeting mutated IDH1 to reduce 2-hydroxyglutarate and hinder tumor growth.Formula:C28H22ClF3N6O3Purezza:98.71% - 99.98%Colore e forma:SolidPeso molecolare:582.96Proguanil hydrochloride
CAS:Proguanil hydrochloride, a biguanide, metabolizes into cycloguanil, an anti-malaria agent that inhibits plasmodium's DNA and protein synthesis.Formula:C11H17Cl2N5Purezza:98.34% - 98.39%Colore e forma:SolidPeso molecolare:290.19BAY-1436032
CAS:BAY-1436032 is a novel, selective and orally available inhibitor of pan-mutant isocitrate dehydrogenase 1 (IDH1).Formula:C26H30F3N3O3Purezza:99.65% - 99.71%Colore e forma:SolidPeso molecolare:489.53Brequinar sodium
CAS:Bipenquinate is a potent and selective inhibitor of dihydroorotate dehydrogenase (DHODH) with IC50 of 20 nM, blocking de novo pyrimidine biosynthesis.Formula:C23H14F2NNaO2Purezza:98.16%Colore e forma:SolidPeso molecolare:397.36DS-1001b
CAS:DS-1001b is an inhibitor of mutant IDH-1 (Isocitrate Dehydrogenase-1)Formula:C29H29Cl3FN3O4Purezza:99.81%Colore e forma:SolidPeso molecolare:608.92Vidofludimus hemicalcium
CAS:Vidofludimus hemicalcium: oral DHODH inhibitor, FXR modulator, for autoimmune and fatty liver research.Formula:C20H18FNO4CaColore e forma:SolidPeso molecolare:375.4G6PDi-1
CAS:<p>G6PDi-1 is an effective G6PD inhibitor. It depletes NADPH and decreases inflammatory cytokine production.</p>Formula:C14H12N4OSPurezza:98.69%Colore e forma:SolidPeso molecolare:284.34AZD7545
CAS:AZD7545 is a potent PDHK inhibitor.Formula:C19H18ClF3N2O5SPurezza:99.12% - 99.96%Colore e forma:SolidPeso molecolare:478.87BMS-823778 hydrochloride
CAS:<p>BMS-823778 hydrochloride is a potent, selective, and orally active inhibitor of 11β-HSD1 (11β-Hydroxysteroid Dehydrogenase Type 1), demonstrating an IC50 (half</p>Formula:C18H19Cl2N3OColore e forma:SolidPeso molecolare:364.27MK-8245
CAS:MK-8245 is a liver-targeting SCD inhibitor for human SCD1 (IC50: 1 nM) and for rat/mouse SCD1 (IC50: 3 nM), with anti-diabetic and anti-dyslipidemic function.Formula:C17H16BrFN6O4Purezza:97.58% - 99%Colore e forma:SolidPeso molecolare:467.25LDHA-IN-4
CAS:LDHA-IN-4 (AZ33) is an LDHA inhibitor. Binding affinity to 6-His-tagged human LDHA expressed in E.coli BL21 (DE3) by SPR analysis with an active value of 93 nM.Formula:C25H27N3O6SPurezza:98.17% - 99.68%Colore e forma:SolidPeso molecolare:497.56NCT-505
CAS:NCT-505 is a potent and selective inhibitor of aldehyde dehydrogenase (ALDH1A1, IC50 = 7 nM) and a weak inhibitor of hALDH1A2, hALDH1A3, hALDH2, hALDH3A1 withFormula:C27H28FN5O3SPurezza:99.93%Colore e forma:SolidPeso molecolare:521.61VER-246608
CAS:VER-246608 inhibits PDK (IC50: 35-91 nM), boosts PDC, reduces glycolysis, causes cancer cell cytostasis, and enhances doxorubicin effects.Formula:C28H23ClF2N4O4Purezza:98.5%Colore e forma:SolidPeso molecolare:552.96Nifurtimox
CAS:Nifurtimox (BAY-A-2502) is an antiprotozoal agent (IC50s = 9.91, 12.28, and 10.44 μM against Taluahuén, LQ, and Brener strains of T.Formula:C10H13N3O5SPurezza:99.87% - 99.89%Colore e forma:SolidPeso molecolare:287.29
