AhR
Il recettore degli idrocarburi arilici (AhR) è un fattore di trascrizione attivato da ligandi che svolge un ruolo cruciale nella regolazione delle risposte biologiche ai contaminanti ambientali, come le diossine. AhR è coinvolto anche nel metabolismo degli xenobiotici e nella regolazione delle risposte immunitarie, della proliferazione e differenziazione cellulare. La disregolazione della segnalazione AhR è associata a diverse malattie, tra cui il cancro e i disturbi autoimmuni. Presso CymitQuimica, offriamo una gamma di inibitori di AhR per supportare la tua ricerca in tossicologia, biologia del cancro e immunologia.
Trovati 41 prodotti di "AhR"
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GNF351
CAS:GNF351: Full AHR antagonist, inhibits DRE-dependent/independent activity, low toxicity, binds AHR (IC50: 62 nM).Formula:C24H25N7Purezza:98.43%Colore e forma:SolidPeso molecolare:411.5Diosmin
CAS:Diosmin (Venosmine) is a bioflavonoid that strengthens vascular walls.Formula:C28H32O15Purezza:97.90%Colore e forma:Greyish-Yellow Or Light Yellow Hygroscopic PowderPeso molecolare:608.54Mexiletine hydrochloride
CAS:Mexiletine hydrochloride is a lidocaine-like antiarrhythmic (Class IB) and anesthetic, stabilizing heartbeats by inhibiting sodium in cardiac cells.Formula:C11H18ClNOPurezza:99.88%Colore e forma:White To Off-White SolidPeso molecolare:215.72BAY 2416964
CAS:BAY 2416964 is a small molecule inhibitor that selectively targets aromatic receptor (AhR) and is commonly used in tumor research. Cost-effective and quality-assured.Formula:C18H18ClN5O3Purezza:99.15% - 99.85%Colore e forma:SolidPeso molecolare:387.82Leflunomide
CAS:Leflunomide (HWA486) is an immunomodulatory agent used in the therapy of rheumatoid arthritis and psoriatic arthritis.Formula:C12H9F3N2O2Purezza:99.52% - 99.96%Colore e forma:Off White Crystalline SolidPeso molecolare:270.21StemRegenin 1 Hydrochloride
CAS:StemRegenin 1 Hydrochloride is an AhR antagonist (IC₅₀ = 127 nM) that inhibits RANKL-induced osteoclast generation and differentiation.Formula:C24H24ClN5OSPurezza:99.94%Colore e forma:SolidPeso molecolare:466KYN-101
CAS:<p>KYN-101 is an and aryl hydrocarbon receptor (AHR) inhibitor with anticancer activity. KYN-101 is used for the study of breast cancer and acute myeloid leukemia.</p>Formula:C22H19FN6Purezza:98.35%Colore e forma:SolidPeso molecolare:386.43MeBIO
CAS:MeBIO is an agonist of aryl hydrocarbon receptor, with IC50 of 44 and 55 μM for GSK-3 and CDK1/CyclinB, respectively. MeBIO does not affect GSK-3β.Formula:C17H12BrN3O2Purezza:99.64%Colore e forma:SolidPeso molecolare:370.2WAY-605471
CAS:WAY-605471 is a AHR antagonist with IC50 of 0.5 - 1 μM.Formula:C14H15NO3S2Purezza:99.62%Colore e forma:SolidPeso molecolare:309.4AHR Inhibitor I-103
CAS:AHR Inhibitor I-103 is an aryl hydrocarbon receptor (AHR) inhibitor with anticancer activity used in the study of breast cancer and acute myeloid leukemia.Formula:C21H17FN6Purezza:98.70%Colore e forma:SoildPeso molecolare:372.43',4'-Dimethoxyflavone
CAS:3',4'-Dimethoxyflavone is a standard compound of flavonoids with numerous medicinal activities.Formula:C17H14O4Purezza:98.05%Colore e forma:SolidPeso molecolare:282.29L-Kynurenine
CAS:L-Kynurenine ((S)-Kynurenine)) is an endogenous agonist of aryl hydrocarbon receptor (AHR) ,inhibits allogeneic T cell proliferation. High-Quality, Low-Cost!Formula:C10H12N2O3Purezza:98.44% - 99.91%Colore e forma:Light Yellow CrystallinePeso molecolare:208.21YL-109
CAS:<p>YL-109, a novel anticancer agent, can inhibit breast Y cell growth and invasiveness in vitro and in vivo.</p>Formula:C14H11NO2SPurezza:99.77% - ≥95%Colore e forma:SolidPeso molecolare:257.31ITE
CAS:ITE is a potent endogenous agonist of aryl hydrocarbon receptor (AhR) (Ki : 3 nM), has immunosuppressive activity.Formula:C14H10N2O3SPurezza:97.91% - 99.14%Colore e forma:SolidPeso molecolare:286.31PDM11
CAS:PDM11 (1-[2-(4-Chloro-phenyl)-vinyl]-3,5-diMeth) is an antagonist of aryl hydrocarbon receptor (AhR)Formula:C16H15ClO2Purezza:99.88%Colore e forma:SolidPeso molecolare:274.74Benzyl butyl phthalate
CAS:<p>Benzyl butyl phthalate (1,2-benzenedicarboxylic acid) is used as a plasticizer for PVC.</p>Formula:C19H20O4Purezza:99.02%Colore e forma:Colourless Liquid Oily LiquidPeso molecolare:312.36Indole-3-pyruvic acid
CAS:Indole-3-pyruvic acid is a precursor for the plant growth hormone indole-3-acetic acid.Formula:C11H9NO3Purezza:98.89% - 99.21%Colore e forma:Off White CrystalsPeso molecolare:203.19Tapinarof
CAS:Tapinarof (Benvitimod) is targeted as a topical cream treatment for psoriasis, a chronic autoimmune skin disease.Formula:C17H18O2Purezza:99.64% - >99.99%Colore e forma:SolidPeso molecolare:254.32PD98059
CAS:PD98059 is an MEK inhibitor that inhibits MEK1 and MEK2 (IC50=2/50 μM) and is non-ATP-competitive.Formula:C16H13NO3Purezza:98.63% - >99.99%Colore e forma:Yellow SolidPeso molecolare:267.28Carbidopa
CAS:<p>Carbidopa (Lodosyn) is an aromatic-L-amino-acid decarboxylase inhibitor (IC50: 29±2 μM).</p>Formula:C10H14N2O4Purezza:98.01% - ≥98%Colore e forma:SolidPeso molecolare:226.23
