Fosfolipasi
Le fosfolipasi sono un gruppo di enzimi che idrolizzano i fosfolipidi in acidi grassi e altre sostanze lipofile, svolgendo un ruolo critico nella biologia delle membrane e nella generazione di molecole segnalatrici. Gli inibitori delle fosfolipasi vengono utilizzati per studiare il loro ruolo nelle malattie infiammatorie, nei disturbi cardiovascolari e nella neurodegenerazione. Questi inibitori sono anche preziosi per esplorare le vie di segnalazione lipidica e le loro implicazioni nei meccanismi delle malattie. Presso CymitQuimica, offriamo una varietà di inibitori delle fosfolipasi per supportare la tua ricerca in infiammazione, metabolismo lipidico e segnalazione cellulare.
Trovati 83 prodotti di "Fosfolipasi"
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Omeprazole
CAS:Omeprazole (Losec) is a proton pump inhibitor (PPI), Omeprazole(Losec) is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor.Formula:C17H19N3O3SPurezza:98.43% - 98.48%Colore e forma:White SolidPeso molecolare:345.42Niflumic acid
CAS:<p>Niflumic acid (Nifluril) is a Ca2+-activated Cl- channel blocker and an analgesic and anti-inflammatory agent used in the therapy of rheumatoid arthritis.</p>Formula:C13H9F3N2O2Purezza:99.47%Colore e forma:SolidPeso molecolare:282.22Tris(2,4-di-tert-butylphenyl)phosphate
CAS:Tris(2,4-di-tert-butylphenyl)phosphate (TDTBPP) inhibits secretory phospholipase A2 (sPLA2) with anti-inflammatory effect. Cost-effective and quality-assured.Formula:C42H63O4PPurezza:99.73%Colore e forma:SolidPeso molecolare:662.92Lp-PLA2-IN-1
CAS:<p>Lp-PLA2-IN-1 suppresses Lp-PLA2, aiding in treating atherosclerosis and Alzheimer's.</p>Formula:C21H17F5N4O3Purezza:99.60%Colore e forma:SolidPeso molecolare:468.38Lansoprazole
CAS:Lansoprazole (A-65006) is a 2, 2, 2-trifluoroethoxypyridyl derivative of timoprazole that is used in the therapy of STOMACH ULCERS and ZOLLINGER-ELLISONFormula:C16H14F3N3O2SPurezza:99.18% - 99.84%Colore e forma:White Crystalline PowderPeso molecolare:369.36ML349
CAS:ML349 is an inhibitor of LYPLA2 (IC50: 144 nM). ML349 is an effective and specific acyl protein thioesterase 2 (APT-2) inhibitor (Ki: 120 nM).Formula:C23H22N2O4S2Purezza:99.59% - 99.88%Colore e forma:SolidPeso molecolare:454.561-Myristoyl-2-Linoleoyl-sn-glycero-3-PC
CAS:1-Myristoyl-2-Linoleoyl-sn-glycero-3-PC is a phospholipid identified in human plasma, characterized by the presence of Myristic acid and Linoleic acid at the sn-1 and sn-2 positions, respectively.Formula:C40H76NO8PColore e forma:SolidPeso molecolare:730.01VU533
CAS:VU533 is a NAPE-PLD activator, EC50=0.30 µM, boosts macrophage activity, potential in cardiometabolic diseases.Formula:C21H22FN3O3S2Purezza:99.87%Colore e forma:SolidPeso molecolare:447.55AACOCF3
CAS:AACOCF3 (Arachidonyl trifluoromethyl ketone) is a cell-permeable trifluoromethyl ketone analog of arachidonic acid.Formula:C21H31F3OPurezza:99% - 99%Colore e forma:Yellow LiquidPeso molecolare:356.47A3373
CAS:A3373 is a novel inhibitor targeting both Phospholipase D1 (PLD1) and Phospholipase D2 (PLD2), demonstrating half maximal inhibitory concentrations (IC50) ofFormula:C17H9F7N2OPurezza:98%Colore e forma:SoildPeso molecolare:390.26Compound 48/80 trihydrochloride
CAS:<p>Compound 48/80 trihydrochloride (C48/80 trihydrochloride) 是 N-甲基对甲氧基苯乙胺和甲醛发生缩合反应后的混合物。Compound 48/80 trihydrochloride 是一种肥大细胞 (mast cell) 脱颗粒剂和组胺 (histamine) 释放剂。Compound 48/80 trihydrochloride 对人血小板磷脂酰肌醇特异性磷脂酶 C (phosphatidylinositol-specific phospholipase C) 活性有抑制作用。</p>Formula:C32H48Cl3N3O3Purezza:98%Colore e forma:SolidPeso molecolare:629.1DPTIP
CAS:<p>DPTIP is an effective inhibitor of neutral sphingomyelinase 2 with an IC50 value of 30 nM.</p>Formula:C21H18N2O3SPurezza:99.88%Colore e forma:SolidPeso molecolare:378.44BIRM 271
CAS:<p>BIRM 271 is a novel arachidonic acid release inhibitor that blocks leukotriene B4 and platelet-activating factor biosynthesis in human neutrophils.</p>Formula:C21H25N3OPurezza:99.64%Colore e forma:SoildPeso molecolare:335.44SB-435495
CAS:SB-435495 is a compound characterized by its potent, selective, reversible, and non-covalent inhibition of Lp-PLA2, demonstrating an IC50 value of 0.06 nM.Formula:C38H40F4N6O2SPurezza:99.07%Colore e forma:SolidPeso molecolare:720.82DPTIP hydrochloride
CAS:DPTIP hydrochloride is a potent inhibitor of neutral sphingomyelinase (N-SMase 2) that can cross the blood-brain barrier. It acts as an exosome inhibitor with an IC50 value of 30 nM.Formula:C21H19ClN2O3SColore e forma:SolidPeso molecolare:414.91PLA2-IN-1
PLA2-IN-1 (Compound 7) is a potent and selective inhibitor of phospholipase A (PLA2) with an IC50 value of 1 nM. It effectively inhibits PLA2-induced coagulation disorders in vitro and shows potential for use as an antidote for snake bites caused by cobra venom.Colore e forma:Odour SolidnSMase2-IN-1
nSMase2-IN-1 is an orally active inhibitor of Neutral sphingomyelinase 2 (nSMase2) with a potent IC50 value of 0.13 ± 0.06 μM.Formula:C12H17N5OPurezza:98%Colore e forma:SolidPeso molecolare:247.3A4333
A4333, a biotinylated derivative of A3373, selectively inhibits Phospholipase D1 (PLD1) while sparing PLD2.Purezza:98%Colore e forma:Odour SolidLEI110
CAS:LEI110 inhibits PLA2G16 and HRASLS enzymes, Ki 20 nM, selectively targets related thiol hydrolases.Formula:C25H23F3N2O3Purezza:98.66% - 98.8%Colore e forma:SolidPeso molecolare:456.46ASM-IN-3
CAS:ASM-IN-3 (Compound 21b) is a selective acid sphingomyelinase (ASM) inhibitor that can penetrate the blood-brain barrier, with an IC50 of 3.37 μM against purified human ASM. By inhibiting ASM activity in the hippocampus and promoting neurogenesis, ASM-IN-3 alleviates depressive-like behavior in reserpine-induced depressive rats.Formula:C17H13ClN2O4Colore e forma:SolidPeso molecolare:344.75BMS493
CAS:BMS493 is an inverse agonist of RAR that inhibits retinoic acid-induced differentiation and inhibits the increase in phospholipase A2 activity.Formula:C29H24O2Purezza:99.12% - >99.99%Colore e forma:SolidPeso molecolare:404.5Bromoenol lactone
CAS:NeurokininBromoenol lactone ((6E)-Bromoenol lactone) is an iPLA2β and serine protease inhibitor that attenuates nicotine-induced breast cancer cell proliferation.Formula:C16H13BrO2Colore e forma:SolidPeso molecolare:317.18PACOCF3
CAS:PACOCF3, a phospholipase A2 inhibitor, hinders Ca2+ signaling with an IC50 of 3.8 μM in renal cells.Formula:C17H31F3OPurezza:99.93%Colore e forma:SolidPeso molecolare:308.42LEI-401
CAS:LEI-401 is a NAPE-PLD inhibitor.LEI-401 reduces the level of n-acyl ethanolamines in the brain of free-ranging mice and modulates their emotional behaviour.Formula:C24H31N5O2Purezza:99.79% - 99.79%Colore e forma:SolidPeso molecolare:421.54MJ33 lithium salt
CAS:MJ33 lithium salt is an inhibitor of NADPH oxidase type 2-mediated ROS generation, inhibits PLA2 activity, and can be used to study acute lung injury.Formula:C22H43F3LiO6PPurezza:99%Colore e forma:SolidPeso molecolare:498.48AA26-9
CAS:AA26-9 is an effective and broad-spectrum inhibitor of serine hydrolase.Formula:C7H10N4OPurezza:99.88%Colore e forma:SolidPeso molecolare:166.18Ref: TM-T3990
1mg37,00€2mg52,00€5mg79,00€10mg119,00€25mg210,00€50mg350,00€100mg522,00€1mL*10mM (DMSO)87,00€N-(p-amylcinnamoyl) Anthranilic Acid
CAS:N-(p-amylcinnamoyl) Anthranilic Acid (ACA) is a broad spectrum Phospholipase A2 (PLA2) inhibitor and TRP channel blocker.Formula:C21H23NO3Purezza:99.35% - 99.67%Colore e forma:SolidPeso molecolare:337.41Rhamnetin
CAS:Rhamnetin (beta-Rhamnocitrin), a quercetin derivative found in Coriandrum sativum, has antioxidant and anti-inflammatory activities.Formula:C16H12O7Purezza:99.61% - 99.905%Colore e forma:SolidPeso molecolare:316.26Ref: TM-TN1419
1mg64,00€5mg137,00€10mg210,00€25mg356,00€50mg525,00€100mg747,00€1mL*10mM (DMSO)144,00€hnps-PLA Inhibitor
CAS:<p>Hnps-PLA Inhibitor is an inhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA).</p>Formula:C21H21N3O4Purezza:99.68%Colore e forma:SolidPeso molecolare:379.41Varespladib
CAS:Varespladib (LY315920) inhibits hnsPLA2 effectively (IC50=7 nM), studied for sickle cell, VOC, and acute coronary syndrome.Formula:C21H20N2O5Purezza:99.97%Colore e forma:SolidPeso molecolare:380.39Ref: TM-T2044
1mg46,00€5mg87,00€10mg144,00€25mg227,00€50mg338,00€100mg487,00€200mg705,00€1mL*10mM (DMSO)81,00€BAPTA
CAS:BAPTA is a neuroprotective agent in cerebral ischemia, acting as an intercellular Ca2+ chelator.Formula:C22H24N2O10Purezza:97.21% - ≥95%Colore e forma:White SolidPeso molecolare:476.43Rapanone
CAS:Rapanone (2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone) is a natural benzoquinone that is a potent and selective inhibitor of human synovial PLA2.Formula:C19H30O4Purezza:99.56%Colore e forma:SolidPeso molecolare:322.44U-73343
CAS:<p>U-73343 is an inactive analog of U-73122 and can be used as a negative control. U-73122 dose-dependently inhibits acid secretion irrespective of the stimulant.</p>Formula:C29H42N2O3Purezza:99.06%Colore e forma:SolidPeso molecolare:466.66Tanshinone I
CAS:Tanshinone I (Tanshinone A), an active principle isolated from the herbal medicine Salvia miltiorrhiza, displays cytotoxicity against tumor cells.Formula:C18H12O3Purezza:98.31% - 98.70%Colore e forma:SolidPeso molecolare:276.29ML348
CAS:ML348 (GNF-Pf-1127) is a selective and reversible lysophospholipase 1 (LYPLA1) inhibitor (IC50 = 210 nM).Formula:C18H17ClF3N3O3Purezza:99% - 99.88%Colore e forma:SolidPeso molecolare:415.79Ref: TM-T3439
2mg47,00€5mg69,00€10mg97,00€25mg227,00€50mg354,00€100mg567,00€200mg792,00€500mg1.198,00€FIPI
CAS:<p>FIPI, a halopemide derivative, strongly blocks PLD1 and PLD2 (IC50s: 25 nM, 20 nM) and hinders PLD-mediated cell activity.</p>Formula:C23H24FN5O2Purezza:97.21% - 98.68%Colore e forma:SolidPeso molecolare:421.47ML-298
CAS:ML-298 (CID53393915) is a potent, specific inhibitor of Phospholipase D2 (PLD2, IC50 of 355 nM).Formula:C22H23F3N4O2Purezza:99.35%Colore e forma:SolidPeso molecolare:432.441-Naphthaleneacetic acid
CAS:1-Naphthaleneacetic acid, an auxin-like synthetic plant hormone, boosts rooting in horticulture.Formula:C12H10O2Purezza:98.67%Colore e forma:Needles From Water White To Off White CrystalsPeso molecolare:186.21ST271
CAS:<p>ST271 is an effective protein tyrosine kinase (PTK) inhibitor.</p>Formula:C16H20N2O2Purezza:98.94%Colore e forma:SolidPeso molecolare:272.34Darapladib
CAS:Darapladib (SB-480848) is a lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor with an IC50 value of 0.25 nM.Cost-effective and quality-assured.Formula:C36H38F4N4O2SPurezza:99.82% - >99.99%Colore e forma:SolidPeso molecolare:666.77Ref: TM-T6109
1mg42,00€2mg52,00€5mg87,00€10mg125,00€25mg180,00€50mg309,00€100mg499,00€200mgPrezzo su richiesta1mL*10mM (DMSO)116,00€RHC 80267
CAS:RHC 80267 (U-57908) is a selective inhibitor of DAGL (IC50 : 4 μM in canine platelets)Formula:C20H34N4O4Purezza:99.54%Colore e forma:White SolidPeso molecolare:394.51GW4869
CAS:GW4869 (GW69A) is a selective and non-competitive inhibitor of neutral sphingomyelinase N-SMase (IC50=1 μM).Formula:C30H30Cl2N6O2Purezza:98.12% - 98.47%Colore e forma:SolidPeso molecolare:577.5RPI-1
CAS:<p>RPI-1 is a competitive, potent ATP-dependent Ret kinase inhibitor.</p>Formula:C17H15NO4Purezza:98.91% - ≥95%Colore e forma:SolidPeso molecolare:297.31Anti-Inflammatory Peptide 1 Acetate
Anti-Inflammatory Peptide 1 Acetate (C45H82N12O14S2) inhibits PLA2 to reduce inflammation and pain.Formula:C47H86N12O16S2Purezza:98.95%Colore e forma:SolidPeso molecolare:1139.39Ref: TM-T21606L
2mg46,00€5mg64,00€10mg96,00€25mg138,00€50mg202,00€100mg301,00€200mg452,00€1mL*10mM (DMSO)150,00€1-Linoleoyl Glycerol
CAS:1-Linoleoyl Glycerol (Monolinolein) is fatty acid glycerol that has been isolated from Saururus Chinensis roots.Formula:C21H38O4Purezza:98.95% - 99.15%Colore e forma:Less Oil Colourless OilPeso molecolare:354.52ONO-RS-082
CAS:ONO-RS-082 is a Ca2+-independent phospholipase A2 inhibitor.Formula:C21H22ClNO3Purezza:99.35%Colore e forma:SolidPeso molecolare:371.86Ref: TM-T21815
2mg42,00€5mg62,00€10mg92,00€25mg170,00€50mg283,00€100mg424,00€200mg612,00€1mL*10mM (DMSO)67,00€ML-211
CAS:<p>ML-211 is a carbamate-based dual inhibitor of LYPLA1 (IC50 = 17 nM) and the related LYPLA2 (IC50 = 30 nM)</p>Formula:C25H30N4O2Purezza:97.07%Colore e forma:SolidPeso molecolare:418.531-Naphthaleneacetic acid potassium salt
CAS:1-Naphthaleneacetic acid potassium salt (1-NAA Potassium Salt) is a synthetic phytogrowth hormone that promotes plant growth and a PLA2 inhibitor.Formula:C12H9O2·KPurezza:97.68%Colore e forma:Off-White To Beige PowderPeso molecolare:224.3Difluprednate
CAS:<p>Difluprednate (Myser)(Durezol) is a corticosteroid, approved for the treatment of post-operative ocular inflammation and pain.</p>Formula:C27H34F2O7Purezza:99.23% - 99.86%Colore e forma:SolidPeso molecolare:508.55Cambinol
CAS:Cambinol is a SIRT1/2 inhibitor (IC50: 56/59 μM), non-competitive with NAD, weak on SIRT5, and prompts apoptosis in lymphoma cells.Formula:C21H16N2O2SPurezza:98.02% - 99.83%Colore e forma:SolidPeso molecolare:360.43Ref: TM-T4019
1mg40,00€2mg52,00€5mg85,00€10mg124,00€25mg219,00€50mg350,00€100mg522,00€500mg1.130,00€1mL*10mM (DMSO)66,00€CAY10594
CAS:CAY10594, a PLD2 inhibitor, mitigates acetaminophen liver damage via the p-GSK-3β/JNK pathway.Formula:C26H28N4O2Purezza:98%Colore e forma:SolidPeso molecolare:428.53trans-Benzylideneacetone
CAS:trans-Benzylideneacetone (Acetocinnamone) is used in various synthetic preparations.Formula:C10H10OPurezza:97.48%Colore e forma:Light Yellow Low Melting Crystalline MassPeso molecolare:146.19Aristolochic acid C
CAS:<p>Aristolochic acid C is a derivative of Aristolochic acid which is a phospholipase A2 inhibitor.</p>Formula:C16H9NO7Purezza:99.8%Colore e forma:White PowderPeso molecolare:327.25CAY10650
CAS:CAY10650 is an effective inhibitor of cytosolic phospholipase A2α (cPLA2α, IC50: 12 nM).Formula:C28H25NO6Purezza:97.33%Colore e forma:SolidPeso molecolare:471.5Ref: TM-TQ0105
1mg51,00€5mg120,00€10mg175,00€25mg354,00€50mg494,00€100mg655,00€1mL*10mM (DMSO)125,00€U-73122
CAS:U-73122 (U73122) , an effective PLC inhibitor, reduces agonist-induced Ca2+ increases in platelets and PMN.Formula:C29H40N2O3Purezza:97.50%Colore e forma:Solid Off-WhitePeso molecolare:464.64m-3M3FBS
CAS:m-3M3FBS is a phospholipase C (PLC) activator.Formula:C16H16F3NO2SPurezza:99.66%Colore e forma:SolidPeso molecolare:343.36Melittin
CAS:Melittin: principal bee venom toxin, 26 amino acids, activates low-weight PLA2, not high-weight PLA2.Formula:C131H229N39O31Purezza:98.37% - 99.92%Colore e forma:SolidPeso molecolare:2846.46Neomycin sulfate
CAS:Neomycin sulfate (Framycin sulfate) is a broad-spectrum aminoglycoside antibiotic that blocks the synthesis of bacterial proteins in order to exertFormula:C23H46N6O13·3H2SO4Purezza:99.4% - 99.88%Colore e forma:Tan PowderPeso molecolare:908.87VU0155056
CAS:VU0155056 is a dual PLD1/2 inhibitor with IC50 < 1 µM in cellular assays, inhibits breast cancer cell invasion.Formula:C25H26N4O2Purezza:98.6% - 99.15%Colore e forma:SolidPeso molecolare:414.5LCL521
CAS:LCL521 inhibits lysosomal acid sphingomyelinase (ASMase).LCL521 is an acid ceramidase (ACDase) inhibitor.Formula:C31H52N4O7Purezza:98%Colore e forma:SolidPeso molecolare:592.77Omeprazole Sodium
CAS:Omeprazole Sodium is a proton pump inhibitor(PPI) and suppresses gastric acid secretion.Formula:C17H18N3NaO3SPurezza:99.84%Colore e forma:Clear In WaterPeso molecolare:367.42-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide
CAS:2-Decenoylaminoethyl cyclohexylethyl sulfide prevents stress ulcers, stabilizes phospholipase A2 and prostaglandin E2.Formula:C20H37NOSPurezza:98%Colore e forma:SolidPeso molecolare:339.58ML299
CAS:ML299 (VU0463568) is a dual PLD1/2 inhibitor (PLD1 and PLD2, IC50 of 6 nM, 20 nM, respectively).Formula:C23H26BrFN4O2Purezza:98%Colore e forma:SolidPeso molecolare:489.38Lp-PLA2-IN-3
CAS:Lp-PLA2-IN-3: Potent oral inhibitor of human Lp-PLA2 with a 14 nM IC50.Formula:C20H13ClF3N3O3SPurezza:99.84%Colore e forma:SolidPeso molecolare:467.85Ref: TM-T11874
1mg96,00€2mg139,00€5mg227,00€10mg359,00€25mg595,00€50mg842,00€100mg1.121,00€500mg2.262,00€1mL*10mM (DMSO)233,00€ASM-IN-1
CAS:ASM-IN-1: Oral acid sphingomyelinase inhibitor, IC50 = 1.5 µM; reduces lipid plaques, plasma ceramide, Ox-LDL.Formula:C16H12BrN3O4Purezza:98%Colore e forma:SolidPeso molecolare:390.19GK187
CAS:GK187 is a selective and potent Group VIA calcium-independent phospholipase A2 (GVIA iPLA2) inhibitor, used in the study of neurological disorders.Formula:C14H15F5O2Colore e forma:SolidPeso molecolare:310.26Ref: TM-T37221
1mg84,00€5mg175,00€10mg283,00€25mg538,00€50mg847,00€100mg1.378,00€1mL*10mM (DMSO)188,00€Halopemide
CAS:Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).Formula:C21H22ClFN4O2Purezza:96.57%Colore e forma:SolidPeso molecolare:416.88Giripladib
CAS:<p>Giripladib (PLA695/PLX-695) blocks radiation-boosted phosphorylation of ERK and Akt in endothelial cells.</p>Formula:C41H36ClF3N2O4SPurezza:99.64%Colore e forma:SolidPeso molecolare:745.25VU0155069
CAS:VU0155069, a selective PLD1 inhibitor (IC50: 46 nM), halts cancer cell migration in transwell assays.Formula:C26H27ClN4O2Purezza:99.5%Colore e forma:SolidPeso molecolare:462.97VU0364739
CAS:VU0364739, a selective phospholipase D2 (PLD2) inhibitor with an IC50 of 22 nM, effectively reduces cancer cell proliferation [1].Formula:C26H27FN4O2Purezza:98%Colore e forma:SolidPeso molecolare:446.52Lp-PLA2-IN-13
CAS:Lp-PLA2-IN-13 (compound 15), a potent Lp-PLA2 inhibitor, holds potential for research in neurodegenerative-related diseases [1].Formula:C22H17F5N4O4Purezza:98%Colore e forma:SolidPeso molecolare:496.39Lp-PLA2-IN-2
CAS:Lp-PLA2-IN-2 is a selective and potent lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor, with an IC50 0f 120 nM for recombinant human Lp-PLA2.Formula:C19H23FN2O4SPurezza:98%Colore e forma:SolidPeso molecolare:394.46Lp-PLA2-IN-14
CAS:Lp-PLA2-IN-14 (Compound 19), an inhibitor of rhLp-PLA2, exhibits a potent inhibitory effect with a pIC50 value of 8.4.Formula:C16H14F3N3O3Purezza:98%Colore e forma:SolidPeso molecolare:353.37,7-Dimethyl-(5Z,8Z)-eicosadienoic acid
CAS:7,7-Dimethyl-(5Z,8Z)-eicosadienoic acid (DEDA, 5 μM) significantly impacts the response to βA(25-35) stimulation. It reduces the formation of ROS.Formula:C22H40O2Colore e forma:SolidPeso molecolare:336.55Varespladib methyl
CAS:Varespladib methyl (LY333013), a bioavailable prodrug of Varespladib, is a selective group II secretory phospholipase A2 inhibitor.Formula:C22H22N2O5Purezza:99.42% - 99.97%Colore e forma:SolidPeso molecolare:394.42Ref: TM-T17218
1mg87,00€2mg130,00€5mg210,00€10mg338,00€25mg557,00€50mg770,00€100mg1.054,00€200mg1.406,00€1mL*10mM (DMSO)233,00€Ecopladib
CAS:<p>Ecopladib inhibits cPLA2α with IC50 of 0.15 μM (micelles) & 0.11 μM (rat blood).</p>Formula:C39H33Cl3N2O5SPurezza:95.15%Colore e forma:SolidPeso molecolare:748.11Rilapladib
CAS:Rilapladib (SB 659032) is a selective inhibitor of Lipoprotein-Associated Phospholipase A2(Lp-PLA2, IC50 = 230 pM) and an antagonist of the platelet activatingFormula:C40H38F5N3O3SPurezza:99.92%Colore e forma:SolidPeso molecolare:735.8Ref: TM-T16751
1mg93,00€5mg227,00€10mg369,00€25mg567,00€50mg787,00€100mg1.169,00€200mg1.586,00€1mL*10mM (DMSO)368,00€MAFP
CAS:MAFP (Methyl Arachidonyl Fluorophosphonate) is an effective irreversible inhibitor of anandamide amidase.Formula:C21H36FO2PColore e forma:SolidPeso molecolare:370.48GK420
CAS:GK420 (AVX420) is a potent inhibitor of cytoplasmic phospholipase A2α (cPLA2α), with an XI(50) value of 0.0016. It effectively inhibits the release of arachidonic acid, with an EC50 of 0.09 μM. GK420 plays a significant role in cancer research.Formula:C20H25NO5SColore e forma:SolidPeso molecolare:391.481Ro 23-9358
CAS:Ro 23-9358 is a potent inhibitor of secretory phospholipase A2, exhibiting anti-inflammatory properties.Formula:C30H51NO6Colore e forma:SolidPeso molecolare:521.729Lp-PLA2-IN-16
CAS:<p>Lp-PLA2-IN-16 (Example 1) is an inhibitor of lipoprotein-associated phospholipase A2 (Lp-PLA2) with potential applications in Alzheimer's disease research [1].</p>Formula:C22H17F5N4O3Purezza:98%Colore e forma:SolidPeso molecolare:480.39Ref: TM-T79076
Prodotto fuori produzioneLp-PLA2-IN-12
CAS:<p>Lp-PLA2-IN-12 (compound 19), an Lp-PLA2 inhibitor, is utilized in researching neurodegenerative diseases including Alzheimer's disease (AD), glaucoma, age-</p>Formula:C24H23F2N5O3Purezza:98%Colore e forma:SolidPeso molecolare:467.47Ref: TM-T79010
Prodotto fuori produzioneLp-PLA2-IN-15
CAS:<p>Lp-PLA2-IN-15 (example 2) is an inhibitor of lipoprotein-associated phospholipase A2 (Lp-PLA2) with potential application in Alzheimer's disease research [1].</p>Formula:C22H17F5N4O3Purezza:98%Colore e forma:SolidPeso molecolare:480.39Ref: TM-T79075
Prodotto fuori produzione
