
CETP
La CETP è una proteina plasmatica che facilita il trasferimento di esteri del colesterolo e trigliceridi tra le lipoproteine, svolgendo un ruolo chiave nel metabolismo lipidico e nella salute cardiovascolare. L'inibizione della CETP è stata esplorata come strategia terapeutica per aumentare i livelli di colesterolo HDL e ridurre il rischio di malattie cardiovascolari. Presso CymitQuimica, offriamo inibitori della CETP per supportare la tua ricerca nel metabolismo lipidico, nelle malattie cardiovascolari e nello sviluppo terapeutico.
Trovati 20 prodotti di "CETP"
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3-Pyridinemethanol
CAS:<p>3-Pyridinemethanol (Roniacol) is an alcohol analog of nicotinic acid which is a peripheral vasodilator that causes flushing and may decrease blood pressure.</p>Formula:C6H7NOPurezza:98.9% - 99.30%Colore e forma:Clear Light Yellow To Yellow LiquidPeso molecolare:109.13CETP-IN-4
CAS:CETP-IN-4 is a cholesteryl ester transfer protein (CETP) inhibitor.Formula:C36H28F9N3O4Colore e forma:SolidPeso molecolare:737.623MK-8262
CAS:MK-8262: oral CETP inhibitor, potent (IC50 = 53 nM, log D = 5.3), may impact HDL/LDL and CHD research.Formula:C35H25F9N2O5Colore e forma:SolidPeso molecolare:724.58α-Amyl cinnamaldehyde
CAS:<p>alpha-Amyl cinnamaldehyde is a common additive in the perfume and cosmetic industry as an aroma substance.</p>Formula:C14H18OColore e forma:Colorless Liquid LiquidPeso molecolare:202.29Anti-CETP Antibody (2H481)
Anti-CETP Antibody (2H481) is an antibody targeting CETP. Anti-CETP Antibody (2H481) can be used in ELISA, IHC.Colore e forma:Odour LiquidTorcetrapib
CAS:Torcetrapib (CP-529414), a CETP inhibitor, curbs cholesteryl ester movement from HDL to LDL/VLDL; failed Phase III trials due to mortality increase.Formula:C26H25F9N2O4Purezza:98% - 99.59%Colore e forma:LipidPeso molecolare:600.47Evacetrapib
CAS:Evacetrapib (LY2484595) inhibits CETP strongly (IC50=5.5 nM), raises HDL cholesterol, no rise in aldosterone/blood pressure. Phase 3.Formula:C31H36F6N6O2Purezza:98.53%Colore e forma:SolidPeso molecolare:638.65Dalcetrapib
CAS:Dalcetrapib (RO4607381), a rhCETP inhibitor (IC50=0.2 μM), increases the plasma HDL cholesterol.Formula:C23H35NO2SPurezza:97.98% - >99.99%Colore e forma:SolidPeso molecolare:389.59Anacetrapib
CAS:Anacetrapib (MK-0859) inhibits rhCETP/CETP(C13S) (IC50: 7.9/11.8 nM), boosts HDL, lowers LDL cholesterol.Formula:C30H25F10NO3Purezza:98.40% - 99.87%Colore e forma:SolidPeso molecolare:637.51CP-532623
CAS:CP-532623, a close structural analog of Torcetrapib, is a CETP inhibitor with highly lipophilic properties. It elevates high-density lipoprotein cholesterol.Formula:C27H27F9N2O3Purezza:98%Colore e forma:SolidPeso molecolare:598.520-HC-Me-Pyrrolidine
<p>20-HC-Me-Pyrrolidine is a potent Aster protein inhibitor that blocks the ability of Aster proteins to bind and transfer cholesterol.</p>Formula:C28H47NO2Purezza:99.99%Colore e forma:SolidPeso molecolare:429.68Azacosterol hydrochloride
CAS:Azacosterol, a diaza cholesterol derivative, reduces cholesterol by inhibiting 24-DHCR and other biosynthesis steps, also affecting bird fertility.Formula:C25H46Cl2N2OColore e forma:SolidPeso molecolare:461.56BMS-795311
CAS:Potent CETP inhibitor, boosts HDL-C levels, orally active; IC50=4nM.Formula:C33H23F10NO3Colore e forma:SolidPeso molecolare:671.52CETP-IN-3
CAS:CETP-IN-3 is an inhibitor of the plasma glycoprotein cholesterol ester transfer protein (CETP), elevating HDL-C through inhibition of CETP.Formula:C30H24F12N2O4Purezza:98%Colore e forma:SolidPeso molecolare:704.5CKD-519
CAS:CKD-519: A CETP inhibitor with an IC50 of 2.3 nM, blocking cholesteryl ester transfer in serum.Formula:C31H34F7NO3Colore e forma:SolidPeso molecolare:601.6Canosimibe
CAS:Canosimibe is a cholesterol absorption inhibitorFormula:C44H60FN3O10Colore e forma:SolidPeso molecolare:809.96CP 524515
CAS:<p>CP 524515 is a potent inhibitor of cholesterol ester transfer protein (CETP), which results in increased levels of high-density lipoprotein cholesterol.</p>Formula:C27H27F9N2O4Colore e forma:SolidPeso molecolare:614.5Implitapide
CAS:Implitapide is an inhibitor of microsomal triglyceride transfer protein (MTP).Formula:C35H37N3O2Purezza:98%Colore e forma:SolidPeso molecolare:531.69TAP311
TAP311 is an inhibitor of cholesteryl ester transfer protein (CETP)(IC50 of 62 nM).Formula:C34H40F6N6O4Purezza:98%Colore e forma:SolidPeso molecolare:710.71Obicetrapib
CAS:<p>Obicetrapib (AMG-899) is an inhibitor of cholesteryl ester transfer protein.</p>Formula:C32H31F9N4O5Purezza:99.26% - >99.99%Colore e forma:SolidPeso molecolare:722.6

