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CETP

CETP

La CETP è una proteina plasmatica che facilita il trasferimento di esteri del colesterolo e trigliceridi tra le lipoproteine, svolgendo un ruolo chiave nel metabolismo lipidico e nella salute cardiovascolare. L'inibizione della CETP è stata esplorata come strategia terapeutica per aumentare i livelli di colesterolo HDL e ridurre il rischio di malattie cardiovascolari. Presso CymitQuimica, offriamo inibitori della CETP per supportare la tua ricerca nel metabolismo lipidico, nelle malattie cardiovascolari e nello sviluppo terapeutico.

Trovati 20 prodotti di "CETP"

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  • 3-Pyridinemethanol

    CAS:
    <p>3-Pyridinemethanol (Roniacol) is an alcohol analog of nicotinic acid which is a peripheral vasodilator that causes flushing and may decrease blood pressure.</p>
    Formula:C6H7NO
    Purezza:98.9% - 99.30%
    Colore e forma:Clear Light Yellow To Yellow Liquid
    Peso molecolare:109.13
  • CETP-IN-4

    CAS:
    CETP-IN-4 is a cholesteryl ester transfer protein (CETP) inhibitor.
    Formula:C36H28F9N3O4
    Colore e forma:Solid
    Peso molecolare:737.623
  • MK-8262

    CAS:
    MK-8262: oral CETP inhibitor, potent (IC50 = 53 nM, log D = 5.3), may impact HDL/LDL and CHD research.
    Formula:C35H25F9N2O5
    Colore e forma:Solid
    Peso molecolare:724.58
  • α-Amyl cinnamaldehyde

    CAS:
    <p>alpha-Amyl cinnamaldehyde is a common additive in the perfume and cosmetic industry as an aroma substance.</p>
    Formula:C14H18O
    Colore e forma:Colorless Liquid Liquid
    Peso molecolare:202.29
  • Anti-CETP Antibody (2H481)


    Anti-CETP Antibody (2H481) is an antibody targeting CETP. Anti-CETP Antibody (2H481) can be used in ELISA, IHC.
    Colore e forma:Odour Liquid
  • Torcetrapib

    CAS:
    Torcetrapib (CP-529414), a CETP inhibitor, curbs cholesteryl ester movement from HDL to LDL/VLDL; failed Phase III trials due to mortality increase.
    Formula:C26H25F9N2O4
    Purezza:98% - 99.59%
    Colore e forma:Lipid
    Peso molecolare:600.47
  • Evacetrapib

    CAS:
    Evacetrapib (LY2484595) inhibits CETP strongly (IC50=5.5 nM), raises HDL cholesterol, no rise in aldosterone/blood pressure. Phase 3.
    Formula:C31H36F6N6O2
    Purezza:98.53%
    Colore e forma:Solid
    Peso molecolare:638.65
  • Dalcetrapib

    CAS:
    Dalcetrapib (RO4607381), a rhCETP inhibitor (IC50=0.2 μM), increases the plasma HDL cholesterol.
    Formula:C23H35NO2S
    Purezza:97.98% - >99.99%
    Colore e forma:Solid
    Peso molecolare:389.59
  • Anacetrapib

    CAS:
    Anacetrapib (MK-0859) inhibits rhCETP/CETP(C13S) (IC50: 7.9/11.8 nM), boosts HDL, lowers LDL cholesterol.
    Formula:C30H25F10NO3
    Purezza:98.40% - 99.87%
    Colore e forma:Solid
    Peso molecolare:637.51
  • CP-532623

    CAS:
    CP-532623, a close structural analog of Torcetrapib, is a CETP inhibitor with highly lipophilic properties. It elevates high-density lipoprotein cholesterol.
    Formula:C27H27F9N2O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:598.5
  • 20-HC-Me-Pyrrolidine


    <p>20-HC-Me-Pyrrolidine is a potent Aster protein inhibitor that blocks the ability of Aster proteins to bind and transfer cholesterol.</p>
    Formula:C28H47NO2
    Purezza:99.99%
    Colore e forma:Solid
    Peso molecolare:429.68
  • Azacosterol hydrochloride

    CAS:
    Azacosterol, a diaza cholesterol derivative, reduces cholesterol by inhibiting 24-DHCR and other biosynthesis steps, also affecting bird fertility.
    Formula:C25H46Cl2N2O
    Colore e forma:Solid
    Peso molecolare:461.56
  • BMS-795311

    CAS:
    Potent CETP inhibitor, boosts HDL-C levels, orally active; IC50=4nM.
    Formula:C33H23F10NO3
    Colore e forma:Solid
    Peso molecolare:671.52
  • CETP-IN-3

    CAS:
    CETP-IN-3 is an inhibitor of the plasma glycoprotein cholesterol ester transfer protein (CETP), elevating HDL-C through inhibition of CETP.
    Formula:C30H24F12N2O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:704.5
  • CKD-519

    CAS:
    CKD-519: A CETP inhibitor with an IC50 of 2.3 nM, blocking cholesteryl ester transfer in serum.
    Formula:C31H34F7NO3
    Colore e forma:Solid
    Peso molecolare:601.6
  • Canosimibe

    CAS:
    Canosimibe is a cholesterol absorption inhibitor
    Formula:C44H60FN3O10
    Colore e forma:Solid
    Peso molecolare:809.96
  • CP 524515

    CAS:
    <p>CP 524515 is a potent inhibitor of cholesterol ester transfer protein (CETP), which results in increased levels of high-density lipoprotein cholesterol.</p>
    Formula:C27H27F9N2O4
    Colore e forma:Solid
    Peso molecolare:614.5
  • Implitapide

    CAS:
    Implitapide is an inhibitor of microsomal triglyceride transfer protein (MTP).
    Formula:C35H37N3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:531.69
  • TAP311


    TAP311 is an inhibitor of cholesteryl ester transfer protein (CETP)(IC50 of 62 nM).
    Formula:C34H40F6N6O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:710.71
  • Obicetrapib

    CAS:
    <p>Obicetrapib (AMG-899) is an inhibitor of cholesteryl ester transfer protein.</p>
    Formula:C32H31F9N4O5
    Purezza:99.26% - >99.99%
    Colore e forma:Solid
    Peso molecolare:722.6