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recettore 5-HT

recettore 5-HT

I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.

Trovati 942 prodotti di "recettore 5-HT"

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  • p-MPPF

    CAS:
    <p>p-MPPF is a 5-HT antagonist that can be used to study neurological diseases.</p>
    Formula:C25H27FN4O2
    Purezza:99.92%
    Colore e forma:Solid
    Peso molecolare:434.51
  • R 50595

    CAS:
    <p>R 50595 is a selective non-competitive cisapride antagonist.</p>
    Formula:C30H35Cl2F2N3O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:594.52
  • Alverine hydrochloride

    CAS:
    <p>Alverine hydrochloride is a parasympatholytic.</p>
    Formula:C20H28ClN
    Colore e forma:Solid
    Peso molecolare:317.9
  • PF-03382792

    CAS:
    <p>PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.</p>
    Formula:C23H32FN3O4
    Purezza:99.64%
    Colore e forma:Solid
    Peso molecolare:433.52
  • LP 12 hydrochloride

    CAS:
    <p>LP 12 hydrochloride is a selective 5-HT7 receptor agonist (Ki=0.13 nM).</p>
    Formula:C32H40ClN3O
    Colore e forma:Solid
    Peso molecolare:518.14
  • Minesapride

    CAS:
    <p>Minesapride: novel 5-HT4 partial agonist, may treat constipation-predominant IBS.</p>
    Formula:C21H31ClN4O5
    Purezza:99.85% - 99.88%
    Colore e forma:Solid
    Peso molecolare:454.95
  • 4-Hydroxy MET

    CAS:
    4-Hydroxy MET (4-HO-MET) is a tryptamine-based new psychoactive substance (NPS), structurally similar to the endogenous neurotransmitter serotonin. It has hallucinogenic properties that affect mood, movement, and cognitive functions.
    Formula:C13H18N2O
    Colore e forma:Solid
    Peso molecolare:218.3
  • Xaliproden

    CAS:
    Xaliproden is a biochemical.
    Formula:C24H22F3N
    Colore e forma:Solid
    Peso molecolare:381.43
  • SB 699551

    CAS:
    <p>SB 699551 is a selective 5-HT5A antagonist (Ki=6.31 nM) that enhances 5-HT neuronal function. It inhibits SERT (Ki=25.12 nM),inhibit breast cancer.</p>
    Formula:C34H45N3O
    Purezza:99.83%
    Peso molecolare:511.74
  • Ethylpropyltryptamine

    CAS:
    <p>Ethylpropyltryptamine (EPT) is an orally active novel psychoactive substance. It is predicted to act as a partial agonist of the 5-HT2A receptor.</p>
    Formula:C15H22N2
    Colore e forma:Solid
    Peso molecolare:230.35
  • Naratriptan D3 Hydrochloride

    CAS:
    Naratriptan D3 Hydrochloride is the deuterium labeled Naratriptan, is a selective agonist of 5-HT1 receptor subtype.
    Formula:C17H26ClN3O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:374.94
  • LEK 8804

    CAS:
    <p>LEK 8804 is a 5-HT(2) receptor antagonist and 5-HT(1A) receptor agonist.</p>
    Formula:C19H19N3O
    Colore e forma:Solid
    Peso molecolare:305.37
  • 5-methoxy-α-Ethyltryptamine

    CAS:
    <p>5-Methoxy-alpha-ethyltryptamine is a psychoactive substance that can cause various effects. It belongs to the tryptamine chemical class and can be used for various psychoactive and stimulant effects. </p>
    Formula:C13H18N2O
    Purezza:98.25%
    Colore e forma:Solid
    Peso molecolare:218.29
  • Minaprine

    CAS:
    <p>Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.</p>
    Formula:C17H22N4O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:298.38
  • 4-Iodoamphetamine hydrochloride

    CAS:
    <p>4-Iodoamphetamine (p-Iodoamphetamine) hydrochloride is a halogenated phenethylamine characterized by the presence of an iodine atom at the para position of the phenyl group. It selectively induces serotonin release and inhibits reuptake in rat brain synaptosomes.</p>
    Formula:C9H13ClIN
    Colore e forma:Solid
    Peso molecolare:297.56
  • 2,6-DMA hydrochloride

    CAS:
    <p>2,6-DMA hydrochloride is a phenethylamine and acts as an agonist of the serotonin 5-HT2 receptor, with a pA2 value of 5.09.</p>
    Formula:C11H18ClNO2
    Colore e forma:Solid
    Peso molecolare:231.72
  • MRS7925


    <p>MRS7925 (Compound 43) serves as a potent antagonist of the 5-HT2B receptor, with an inhibition constant (Ki) of 17 nM, and is utilized in the study of fibrosis</p>
    Formula:C20H26IN5O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:511.36
  • Cariprazine D6

    CAS:
    <p>Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).</p>
    Formula:C21H26D6Cl2N4O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:433.45
  • Alosetron D3 Hydrochloride

    CAS:
    <p>Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.</p>
    Formula:C17H19ClN4O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:333.83
  • Altanserin

    CAS:
    <p>Altanserin, a 5-HT2A receptor binder, is tagged with F-18 for brain PET scans.</p>
    Formula:C22H22FN3O2S
    Colore e forma:Solid
    Peso molecolare:411.49