
recettore 5-HT
I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.
Trovati 942 prodotti di "recettore 5-HT"
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cis-(Z)-Flupentixol dihydrochloride
CAS:cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.Formula:C23H27Cl2F3N2OSPurezza:98.07%Colore e forma:SolidPeso molecolare:507.44Granisetron
CAS:<p>Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.</p>Formula:C18H24N4OColore e forma:SolidPeso molecolare:312.41Altanserin
CAS:<p>Altanserin, a 5-HT2A receptor binder, is tagged with F-18 for brain PET scans.</p>Formula:C22H22FN3O2SColore e forma:SolidPeso molecolare:411.49Setiptiline maleate
CAS:Setiptiline maleate is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist, 5-HT serotonin receptor antagonist.Formula:C23H23NO4Purezza:99.94%Colore e forma:SolidPeso molecolare:377.43SB-269970 hydrochloride
CAS:<p>SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivity</p>Formula:C18H28N2O3S·HClPurezza:98.45%Colore e forma:SolidPeso molecolare:388.95Fluvoxamine
CAS:<p>Fluvoxamine (DU-23000) is a selective, orally available 5-HT and serotonin reuptake inhibitor (SSRI) exhibiting antidepressant effects.</p>Formula:C15H21F3N2O2Colore e forma:SolidPeso molecolare:318.33Eplivanserin (mixture)
CAS:<p>Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist,</p>Formula:C19H21FN2O2Colore e forma:SolidPeso molecolare:328.387Cefaclor
CAS:Cefaclor (Panoral) is a cephalosporin antibiotic.Formula:C15H14ClN3O4SPurezza:99.03% - 99.98%Colore e forma:SolidPeso molecolare:367.81Sumatriptan
CAS:<p>Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.</p>Formula:C14H21N3O2SPurezza:99.93%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:295.4(R)-Praziquantel-d11
CAS:<p>(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel.</p>Formula:C19H24N2O2Purezza:98%Colore e forma:SolidPeso molecolare:323.47Aripiprazole (D8)
CAS:<p>Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).</p>Formula:C23H27Cl2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:456.441-Phenylbiguanide HCl
CAS:<p>Compound PDK0269, as 5-HT3 receptor agonists(3–100 μM, pEC50 5.05±0.06), acutely increased XII (hypoglossal) burst frequency and regularity, and decreased bursts/episode . Phenylbiguanide produced a dose-related (10-500 microM) increase in the release of dopamine (280-2000%). When nomifensine (5 microM) was included in the Ringer solution, the effect of Compound PDK0269 on the release of dopamine was ameliorated or inhibited.</p>Formula:C8H12ClN5Purezza:99.31%Colore e forma:SolidPeso molecolare:213.67SB-277011 hydrochloride
CAS:<p>SB-277011 hydrochloride (SB-277011A hydrochloride) is a D3R antagonist, which induces delayed ejaculation in rats.</p>Formula:C28H31ClN4OPurezza:98.54%Colore e forma:SolidPeso molecolare:475.03Thioridazine
CAS:<p>Thioridazine: an antipsychotic, anti-anxiety drug, blocks dopamine D2, PI3K-Akt-mTOR; halts angiogenesis, kills cancer cells, targets CSCs.</p>Formula:C21H26N2S2Colore e forma:SolidPeso molecolare:370.57Clozapine-d8
CAS:<p>Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.</p>Formula:C18H19ClN4Colore e forma:SolidPeso molecolare:334.87Spiroxatrine
CAS:<p>Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.</p>Formula:C22H25N3O3Purezza:99.94%Colore e forma:SolidPeso molecolare:379.45Ziprasidone D8
CAS:<p>Ziprasidone D8, deuterium-labeled, is a potent antipsychotic, antagonizing 5-HT and dopamine receptors.</p>Formula:C21H21ClN4OSPurezza:98%Colore e forma:SolidPeso molecolare:420.99Agomelatine-d6
CAS:Agomelatine D6 (S-20098 D6) is a deuterium-labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptors.Formula:C15H17NO2Purezza:98%Colore e forma:SolidPeso molecolare:249.34Quetiapine-d4 hemifumarate
CAS:<p>Quetiapine D4 hemifumarate is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a agonist of 5-HT receptors and a antagonist of dopamine receptor,with ntidepressant and anxiolytic.</p>Formula:C25H29N3O6SPurezza:98%Colore e forma:White SolidPeso molecolare:503.61Dehydroaripiprazole
CAS:<p>Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.</p>Formula:C23H25Cl2N3O2Purezza:98.7%Colore e forma:SolidPeso molecolare:446.37
