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recettore 5-HT

recettore 5-HT

I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.

Trovati 942 prodotti di "recettore 5-HT"

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  • cis-(Z)-Flupentixol dihydrochloride

    CAS:
    cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.
    Formula:C23H27Cl2F3N2OS
    Purezza:98.07%
    Colore e forma:Solid
    Peso molecolare:507.44
  • Granisetron

    CAS:
    <p>Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.</p>
    Formula:C18H24N4O
    Colore e forma:Solid
    Peso molecolare:312.41
  • Altanserin

    CAS:
    <p>Altanserin, a 5-HT2A receptor binder, is tagged with F-18 for brain PET scans.</p>
    Formula:C22H22FN3O2S
    Colore e forma:Solid
    Peso molecolare:411.49
  • Setiptiline maleate

    CAS:
    Setiptiline maleate is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist, 5-HT serotonin receptor antagonist.
    Formula:C23H23NO4
    Purezza:99.94%
    Colore e forma:Solid
    Peso molecolare:377.43
  • SB-269970 hydrochloride

    CAS:
    <p>SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits &gt;50-fold selectivity</p>
    Formula:C18H28N2O3S·HCl
    Purezza:98.45%
    Colore e forma:Solid
    Peso molecolare:388.95
  • Fluvoxamine

    CAS:
    <p>Fluvoxamine (DU-23000) is a selective, orally available 5-HT and serotonin reuptake inhibitor (SSRI) exhibiting antidepressant effects.</p>
    Formula:C15H21F3N2O2
    Colore e forma:Solid
    Peso molecolare:318.33
  • Eplivanserin (mixture)

    CAS:
    <p>Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist,</p>
    Formula:C19H21FN2O2
    Colore e forma:Solid
    Peso molecolare:328.387
  • Cefaclor

    CAS:
    Cefaclor (Panoral) is a cephalosporin antibiotic.
    Formula:C15H14ClN3O4S
    Purezza:99.03% - 99.98%
    Colore e forma:Solid
    Peso molecolare:367.81
  • Sumatriptan

    CAS:
    <p>Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.</p>
    Formula:C14H21N3O2S
    Purezza:99.93%
    Colore e forma:White To Off-White Crystalline Powder
    Peso molecolare:295.4
  • (R)-Praziquantel-d11

    CAS:
    <p>(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel.</p>
    Formula:C19H24N2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:323.47
  • Aripiprazole (D8)

    CAS:
    <p>Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).</p>
    Formula:C23H27Cl2N3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:456.44
  • 1-Phenylbiguanide HCl

    CAS:
    <p>Compound PDK0269, as 5-HT3 receptor agonists(3–100 μM, pEC50 5.05±0.06), acutely increased XII (hypoglossal) burst frequency and regularity, and decreased bursts/episode . Phenylbiguanide produced a dose-related (10-500 microM) increase in the release of dopamine (280-2000%). When nomifensine (5 microM) was included in the Ringer solution, the effect of Compound PDK0269 on the release of dopamine was ameliorated or inhibited.</p>
    Formula:C8H12ClN5
    Purezza:99.31%
    Colore e forma:Solid
    Peso molecolare:213.67
  • SB-277011 hydrochloride

    CAS:
    <p>SB-277011 hydrochloride (SB-277011A hydrochloride) is a D3R antagonist, which induces delayed ejaculation in rats.</p>
    Formula:C28H31ClN4O
    Purezza:98.54%
    Colore e forma:Solid
    Peso molecolare:475.03
  • Thioridazine

    CAS:
    <p>Thioridazine: an antipsychotic, anti-anxiety drug, blocks dopamine D2, PI3K-Akt-mTOR; halts angiogenesis, kills cancer cells, targets CSCs.</p>
    Formula:C21H26N2S2
    Colore e forma:Solid
    Peso molecolare:370.57
  • Clozapine-d8

    CAS:
    <p>Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.</p>
    Formula:C18H19ClN4
    Colore e forma:Solid
    Peso molecolare:334.87
  • Spiroxatrine

    CAS:
    <p>Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.</p>
    Formula:C22H25N3O3
    Purezza:99.94%
    Colore e forma:Solid
    Peso molecolare:379.45
  • Ziprasidone D8

    CAS:
    <p>Ziprasidone D8, deuterium-labeled, is a potent antipsychotic, antagonizing 5-HT and dopamine receptors.</p>
    Formula:C21H21ClN4OS
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:420.99
  • Agomelatine-d6

    CAS:
    Agomelatine D6 (S-20098 D6) is a deuterium-labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptors.
    Formula:C15H17NO2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:249.34
  • Quetiapine-d4 hemifumarate

    CAS:
    <p>Quetiapine D4 hemifumarate is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a agonist of 5-HT receptors and a antagonist of dopamine receptor,with ntidepressant and anxiolytic.</p>
    Formula:C25H29N3O6S
    Purezza:98%
    Colore e forma:White Solid
    Peso molecolare:503.61
  • Dehydroaripiprazole

    CAS:
    <p>Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.</p>
    Formula:C23H25Cl2N3O2
    Purezza:98.7%
    Colore e forma:Solid
    Peso molecolare:446.37