
recettore 5-HT
I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.
Trovati 1017 prodotti per "recettore 5-HT".
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Cariprazine
CAS:Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderateFormula:C21H32Cl2N4OPurezza:99.68% - 99.87%Colore e forma:White SolidPeso molecolare:427.41Ref: TM-T4577
1mg49,00€5mg92,00€1mL*10mM (DMSO)103,00€10mg145,00€25mg281,00€50mg394,00€100mg550,00€200mg780,00€Syk Inhibitor II dihydrochloride
CAS:Syk inhibitor II selectively blocks Syk (IC50 = 41 nM), impacting platelet function and inflammation, with lower potency against other kinases.Formula:C14H17Cl2F3N6OPurezza:98.53%Colore e forma:SolidPeso molecolare:413.22Ref: TM-T4391
1mg123,00€2mg200,00€5mg432,00€1mL*10mM (DMSO)432,00€10mg613,00€25mg897,00€50mg1.198,00€100mg1.611,00€GR 125743
CAS:GR 125743 is a novel antagonist of 5-HT1B/1D receptor.Formula:C25H28N4O2Purezza:99.76%Colore e forma:SolidPeso molecolare:416.52Ref: TM-T8737
1mg40,00€2mg52,00€5mg84,00€1mL*10mM (DMSO)93,00€10mg113,00€25mg222,00€50mg333,00€100mg495,00€SB-200646
CAS:SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptorFormula:C15H14N4OPurezza:99.61%Colore e forma:SolidPeso molecolare:266.3MK 212 hydrochloride
CAS:MK 212 hydrochloride is a 5-HT2C receptor agonistFormula:C8H11ClN4·HClPurezza:99.88%Colore e forma:White SolidPeso molecolare:235.12Cinitapride
CAS:Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.Formula:C21H30N4O4Purezza:99.52%Colore e forma:SolidPeso molecolare:402.49Ref: TM-T21385
1mg58,00€5mg120,00€1mL*10mM (DMSO)147,00€10mg205,00€25mg394,00€50mg573,00€100mg803,00€Abaperidone Hydrochloride
CAS:Abaperidone Hydrochloride is an atypical antipsychotic, potently binging to5-HT2 receptors and D2 receptors.Formula:C25H26ClFN2O5Colore e forma:SolidPeso molecolare:488.94Epinastine hydrochloride
CAS:Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.Formula:C16H15N3·HClPurezza:99.26% - 99.62%Colore e forma:SolidPeso molecolare:285.77Alprenolol hydrochloride
CAS:Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.Formula:C15H24ClNO2Purezza:99.79%Colore e forma:White SolidPeso molecolare:285.81Temanogrel hydrochloride
CAS:Temanogrel hydrochloride is a serotonin antagonist and anti-platelet agent.Formula:C24H29ClN4O4Colore e forma:SolidPeso molecolare:472.97Dolasetron Mesylate hydrate
CAS:Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.Formula:C20H26N2O7SPurezza:99.86% - 99.99%Colore e forma:White SolidPeso molecolare:438.49Zacopride
CAS:Zacopride is a selective agonist of inward rectifier potassium current (I K1) channel, inhibiting ventricular arrhythmias without affecting atrial arrhythmias.Formula:C15H20ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:309.79Cariprazine hydrochloride
CAS:Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Formula:C21H33Cl3N4OPurezza:99.78% - >99.99%Colore e forma:SolidPeso molecolare:463.87LY310762
CAS:LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.Formula:C24H27FN2O2·HClPurezza:99.8%Colore e forma:SolidPeso molecolare:430.94Melitracen hydrochloride
CAS:Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.Formula:C21H26ClNPurezza:99.99%Colore e forma:Crystalline SolidPeso molecolare:327.90Ref: TM-T4274
10mg44,00€1mL*10mM (DMSO)48,00€25mg64,00€50mg93,00€100mg110,00€200mg161,00€500mg264,00€Metergoline
CAS:Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Formula:C25H29N3O2Purezza:99.83% - 99.97%Colore e forma:SolidPeso molecolare:403.52Rotigotine-
CAS:Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Formula:C19H25NOSPurezza:98.08% - 99.59%Colore e forma:SolidPeso molecolare:315.47Ref: TM-T6647
5mg50,00€1mL*10mM (DMSO)52,00€10mg73,00€25mg138,00€50mg241,00€100mg358,00€200mg523,00€500mg822,00€Buclizine dihydrochloride
CAS:Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic andFormula:C28H33ClN2·2HClPurezza:98.05%Colore e forma:SolidPeso molecolare:505.95Renzapride hydrochloride
CAS:Renzapride is a 5-HT3 antagonist and 5-HT4 agonist. Renzapride also functions as a 5-HT2B antagonist and has some affinity for the 5-HT2A and 5-HT2C receptors.Formula:C16H23Cl2N3O2Colore e forma:SolidPeso molecolare:360.28Vortioxetine hydrobromide
CAS:Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33Formula:C18H22N2S·HBrPurezza:98.85% - 99.98%Colore e forma:White SolidPeso molecolare:379.36
