CymitQuimica logo
recettore 5-HT

recettore 5-HT

I recettori 5-HT, noti anche come recettori della serotonina, sono un gruppo di recettori accoppiati alle proteine G (GPCR) che mediano gli effetti della serotonina, un neurotrasmettitore coinvolto nella regolazione dell'umore, dell'ansia, del sonno, dell'appetito e di altri processi fisiologici. Questi recettori sono suddivisi in diversi sottotipi, ciascuno con funzioni e proprietà farmacologiche distinte. I modulatori dei recettori 5-HT sono ampiamente studiati per il loro ruolo nel trattamento della depressione, dei disturbi d'ansia e di altre condizioni neuropsichiatriche. Presso CymitQuimica, offriamo una gamma di modulatori dei recettori 5-HT di alta qualità per supportare la tua ricerca in neurofarmacologia, disturbi dell'umore e segnalazione GPCR.

Trovati 1017 prodotti per "recettore 5-HT".

Ordinare per

Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
prodotti per pagina.
  • Cariprazine

    CAS:
    Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate
    Formula:C21H32Cl2N4O
    Purezza:99.68% - 99.87%
    Colore e forma:White Solid
    Peso molecolare:427.41

    Ref: TM-T4577

    1mg
    49,00€
    5mg
    92,00€
    1mL*10mM (DMSO)
    103,00€
    10mg
    145,00€
    25mg
    281,00€
    50mg
    394,00€
    100mg
    550,00€
    200mg
    780,00€
  • Syk Inhibitor II dihydrochloride

    CAS:
    Syk inhibitor II selectively blocks Syk (IC50 = 41 nM), impacting platelet function and inflammation, with lower potency against other kinases.
    Formula:C14H17Cl2F3N6O
    Purezza:98.53%
    Colore e forma:Solid
    Peso molecolare:413.22

    Ref: TM-T4391

    1mg
    123,00€
    2mg
    200,00€
    5mg
    432,00€
    1mL*10mM (DMSO)
    432,00€
    10mg
    613,00€
    25mg
    897,00€
    50mg
    1.198,00€
    100mg
    1.611,00€
  • GR 125743

    CAS:
    GR 125743 is a novel antagonist of 5-HT1B/1D receptor.
    Formula:C25H28N4O2
    Purezza:99.76%
    Colore e forma:Solid
    Peso molecolare:416.52

    Ref: TM-T8737

    1mg
    40,00€
    2mg
    52,00€
    5mg
    84,00€
    1mL*10mM (DMSO)
    93,00€
    10mg
    113,00€
    25mg
    222,00€
    50mg
    333,00€
    100mg
    495,00€
  • SB-200646

    CAS:
    SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptor
    Formula:C15H14N4O
    Purezza:99.61%
    Colore e forma:Solid
    Peso molecolare:266.3

    Ref: TM-T8357

    1mg
    62,00€
    5mg
    122,00€
    1mL*10mM (DMSO)
    128,00€
    10mg
    177,00€
    25mg
    299,00€
    50mg
    430,00€
    100mg
    587,00€
  • MK 212 hydrochloride

    CAS:
    MK 212 hydrochloride is a 5-HT2C receptor agonist
    Formula:C8H11ClN4·HCl
    Purezza:99.88%
    Colore e forma:White Solid
    Peso molecolare:235.12

    Ref: TM-T22987

    5mg
    43,00€
    10mg
    55,00€
    25mg
    100,00€
    50mg
    161,00€
    100mg
    245,00€
    200mg
    353,00€
  • Cinitapride

    CAS:
    Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.
    Formula:C21H30N4O4
    Purezza:99.52%
    Colore e forma:Solid
    Peso molecolare:402.49

    Ref: TM-T21385

    1mg
    58,00€
    5mg
    120,00€
    1mL*10mM (DMSO)
    147,00€
    10mg
    205,00€
    25mg
    394,00€
    50mg
    573,00€
    100mg
    803,00€
  • Abaperidone Hydrochloride

    CAS:
    Abaperidone Hydrochloride is an atypical antipsychotic, potently binging to5-HT2 receptors and D2 receptors.
    Formula:C25H26ClFN2O5
    Colore e forma:Solid
    Peso molecolare:488.94

    Ref: TM-T26508

    25mg
    1.504,00€
    50mg
    1.963,00€
    100mg
    2.520,00€
  • Epinastine hydrochloride

    CAS:
    Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
    Formula:C16H15N3·HCl
    Purezza:99.26% - 99.62%
    Colore e forma:Solid
    Peso molecolare:285.77

    Ref: TM-T6488

    10mg
    37,00€
    1mL*10mM (DMSO)
    44,00€
    25mg
    52,00€
    50mg
    67,00€
    100mg
    90,00€
    200mg
    170,00€
    500mg
    305,00€
  • Alprenolol hydrochloride

    CAS:
    Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.
    Formula:C15H24ClNO2
    Purezza:99.79%
    Colore e forma:White Solid
    Peso molecolare:285.81

    Ref: TM-T22236

    1mL*10mM (DMSO)
    34,00€
    50mg
    39,00€
    100mg
    62,00€
    500mg
    190,00€
  • Temanogrel hydrochloride

    CAS:
    Temanogrel hydrochloride is a serotonin antagonist and anti-platelet agent.
    Formula:C24H29ClN4O4
    Colore e forma:Solid
    Peso molecolare:472.97

    Ref: TM-T68237

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Dolasetron Mesylate hydrate

    CAS:
    Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.
    Formula:C20H26N2O7S
    Purezza:99.86% - 99.99%
    Colore e forma:White Solid
    Peso molecolare:438.49

    Ref: TM-T2589

    5mg
    33,00€
    10mg
    44,00€
    1mL*10mM (DMSO)
    48,00€
    25mg
    62,00€
    50mg
    86,00€
  • Zacopride

    CAS:
    Zacopride is a selective agonist of inward rectifier potassium current (I K1) channel, inhibiting ventricular arrhythmias without affecting atrial arrhythmias.
    Formula:C15H20ClN3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:309.79

    Ref: TM-T5336L

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Cariprazine hydrochloride

    CAS:
    Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)
    Formula:C21H33Cl3N4O
    Purezza:99.78% - >99.99%
    Colore e forma:Solid
    Peso molecolare:463.87

    Ref: TM-T8382

    5mg
    34,00€
    10mg
    49,00€
    25mg
    79,00€
    50mg
    108,00€
    100mg
    161,00€
    500mg
    385,00€
  • LY310762

    CAS:
    LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.
    Formula:C24H27FN2O2·HCl
    Purezza:99.8%
    Colore e forma:Solid
    Peso molecolare:430.94

    Ref: TM-T2688

    5mg
    33,00€
    1mL*10mM (DMSO)
    33,00€
    10mg
    48,00€
    25mg
    92,00€
    50mg
    132,00€
    100mg
    207,00€
    200mg
    313,00€
  • Melitracen hydrochloride

    CAS:
    Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.
    Formula:C21H26ClN
    Purezza:99.99%
    Colore e forma:Crystalline Solid
    Peso molecolare:327.90

    Ref: TM-T4274

    10mg
    44,00€
    1mL*10mM (DMSO)
    48,00€
    25mg
    64,00€
    50mg
    93,00€
    100mg
    110,00€
    200mg
    161,00€
    500mg
    264,00€
  • Metergoline

    CAS:
    Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.
    Formula:C25H29N3O2
    Purezza:99.83% - 99.97%
    Colore e forma:Solid
    Peso molecolare:403.52

    Ref: TM-T4008

    25mg
    Prezzo su richiesta
    50mg
    Prezzo su richiesta
    1mL*10mM (DMSO)
    33,00€
    10mg
    37,00€
  • Rotigotine-

    CAS:
    Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.
    Formula:C19H25NOS
    Purezza:98.08% - 99.59%
    Colore e forma:Solid
    Peso molecolare:315.47

    Ref: TM-T6647

    5mg
    50,00€
    1mL*10mM (DMSO)
    52,00€
    10mg
    73,00€
    25mg
    138,00€
    50mg
    241,00€
    100mg
    358,00€
    200mg
    523,00€
    500mg
    822,00€
  • Buclizine dihydrochloride

    CAS:
    Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and
    Formula:C28H33ClN2·2HCl
    Purezza:98.05%
    Colore e forma:Solid
    Peso molecolare:505.95

    Ref: TM-T6426

    50mg
    34,00€
    100mg
    47,00€
    1mL*10mM (DMSO)
    50,00€
    500mg
    90,00€
    1g
    116,00€
  • Renzapride hydrochloride

    CAS:
    Renzapride is a 5-HT3 antagonist and 5-HT4 agonist. Renzapride also functions as a 5-HT2B antagonist and has some affinity for the 5-HT2A and 5-HT2C receptors.
    Formula:C16H23Cl2N3O2
    Colore e forma:Solid
    Peso molecolare:360.28

    Ref: TM-T28517

    25mg
    1.504,00€
    50mg
    1.963,00€
    100mg
    2.520,00€
  • Vortioxetine hydrobromide

    CAS:
    Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33
    Formula:C18H22N2S·HBr
    Purezza:98.85% - 99.98%
    Colore e forma:White Solid
    Peso molecolare:379.36

    Ref: TM-T2395L

    1mL*10mM (DMSO)
    33,00€
    25mg
    39,00€
    50mg
    55,00€
    100mg
    79,00€
    500mg
    198,00€